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9VLJ image
Crystal Structure Of Fgfr1 In Complex With Covalent Inhibitor 10A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.81 Å Release Date: 2026-05-06
Classification: TRANSFERASE
Ligands: A1ESP, SO4

9VLM image
The X-Ray Co-Crystal Structure Of Human Fgfr2 And Covalent Inhibitor 10A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.26 Å Release Date: 2026-05-06
Classification: TRANSFERASE
Ligands: A1ESP, GOL

9VM9 image
Crystal Structure Of Fgfr3 In Complex With 10S
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.65 Å Release Date: 2026-05-06
Classification: TRANSFERASE
Ligands: A1ESW, MG, GOL

9VMB image
The X-Ray Co-Crystal Structure Of Human Fgfr3 And Compound 10T
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.97 Å Release Date: 2026-05-06
Classification: TRANSFERASE
Ligands: A1ESX, MG, GOL

9U7E image
Fgfr2 Kinase Domain With A Macrocyclic Compound 8G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2026-01-21
Classification: TRANSFERASE
Ligands: A1EOH, SO4

9U7S image
Fgfr2 Kinase Domain With A Macrocyclic Compound 8R
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.99 Å Release Date: 2026-01-21
Classification: TRANSFERASE
Ligands: A1EOJ, SO4

9UHC image
Fgfr1 Kinase Domain With A Covalent Inhibitor 9P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.88 Å Release Date: 2025-09-24
Classification: TRANSFERASE
Ligands: A1EPE, SO4

9UHI image
Fgfr1 Kinase Domain With A Covalent Inhibitor 9O
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.76 Å Release Date: 2025-09-24
Classification: TRANSFERASE
Ligands: A1EPF, SO4

8XB1 image
Crystal Structure Of Flt3 In Complex With A Pyrazinamide Macrocycle Derivative
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.85 Å Release Date: 2024-12-11
Classification: TRANSFERASE/TRANSFERASE INHIBITOR
Ligands: ZX3

8KH6 image
Crystal Structure Of Fgfr4 Kinase Domain With 8R
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.62 Å Release Date: 2024-07-31
Classification: TRANSFERASE/INHIBITOR
Ligands: SO4, VVI, EDO

8KH7 image
Crystal Structure Of Fgfr4 Kinase Domain With 8Zc
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.52 Å Release Date: 2024-07-31
Classification: TRANSFERASE/INHIBITOR
Ligands: SO4, VVW, EDO

8KH8 image
Crystal Structure Of Fgfr4(V550L) Kinase Domain With 8Z
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.49 Å Release Date: 2024-07-31
Classification: TRANSFERASE/INHIBITOR
Ligands: SO4, VVW, EDO

8KH9 image
Crystal Structure Of Fgfr4(V550M) Kinase Domain With 8Z
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.42 Å Release Date: 2024-07-31
Classification: TRANSFERASE/INHIBITOR
Ligands: EDO, SO4, VVW

8W5C image
Crystal Structure Of Fgfr4 Kinase Domain In Complex With 8K
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2024-07-31
Classification: TRANSFERASE
Ligands: VZO

8XZ7 image
Fgfr1 Kinase Domain With A Covalent Inhibitor 10H
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.75 Å Release Date: 2024-06-26
Classification: TRANSFERASE
Ligands: SO4, A1LWW

8Y22 image
Fgfr1 Kinase Domain With A Covalent Inhibitor 9G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.79 Å Release Date: 2024-06-26
Classification: TRANSFERASE
Ligands: A1LW9, SO4

8IKR image
Crystal Structure Of Dpaa
Organism: Escherichia coli 908519
Method: X-RAY DIFFRACTION
Resolution:2.90 Å Release Date: 2023-10-11
Classification: HYDROLASE

8J5W image
The Crystal Structure Of Trka(F589L) Kinase In Complex With N-(3-Cyclopropyl-5-((4-Methylpiperazin-1-Yl)Methyl)Phenyl)-4^6-Methyl-14-Oxo-5-Oxa-13-Aza-1(3,6)-Imidazo[1,2-B]Pyridazina-4(1,3)-Benzenacyclotetradecaphan-2-Yne-4^5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.28 Å Release Date: 2023-09-20
Classification: TRANSFERASE
Ligands: A4U

8J5X image
The Crystal Structure Of Trka(G595R) Kinase In Complex With N-(3-Cyclopropyl-5-((4-Methylpiperazin-1-Yl)Methyl)Phenyl)-4^6-Methyl-14-Oxo-5-Oxa-13-Aza-1(3,6)-Imidazo[1,2-B]Pyridazina-4(1,3)-Benzenacyclotetradecaphan-2-Yne-4^5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.09 Å Release Date: 2023-09-20
Classification: TRANSFERASE
Ligands: A4U

8J61 image
The Crystal Structure Of Trka Kinase In Complex With 4^6-Methyl-N-(3-(4-Methyl-1H-Imidazol-1-Yl)-5-(Trifluoromethyl)Phenyl)-14-Oxo-5-Oxa-13-Aza-1(3,6)-Imidazo[1,2-B]Pyridazina-4(1,3)-Benzenacyclotetradecaphan-2-Yne-4^5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.05 Å Release Date: 2023-09-20
Classification: TRANSFERASE
Ligands: A0X
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