Search Count: 18
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Human Sting With Diabzi Agonist 15
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2023-07-26 Classification: IMMUNE SYSTEM/AGONIST Ligands: WWU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-26
Ligands: WWU
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Human Sting With Agonist Xmt-1616
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2023-07-26 Classification: IMMUNE SYSTEM/AGONIST Ligands: WX8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-26
Ligands: WX8
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Chk1 Kinase In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2018-01-17 Classification: TRANSFERASE Ligands: SO4, D4Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: SO4, D4Q
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Chk1 Kinase In Complex With Compound 44
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2018-01-17 Classification: TRANSFERASE Ligands: D58, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: D58, SO4
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Chk1 Kinase In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-01-17 Classification: TRANSFERASE Ligands: D4Z, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: D4Z, SO4
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Human Jak1 Kinase In Complex With Compound 30 At 2.30 Angstroms Resolution
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-11-25 Classification: TRANSFERASE Ligands: PEG, 5JG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-25
Ligands: PEG, 5JG
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Irreversible Inhibition Of Tak1 Kinase By 5Z-7-Oxozeaenol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2013-01-23 Classification: Transferase/Transferase inhibitor Ligands: EDO, 1FM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-23
Ligands: EDO, 1FM
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Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2012-04-04 Classification: TRANSFERASE Ligands: SO4, YDI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-04
Ligands: SO4, YDI
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Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-04-04 Classification: TRANSFERASE Ligands: SO4, GOL, YDK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-04
Ligands: SO4, GOL, YDK
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Synthesis And Evaluation Of Triazolones As Checkpoint Kinase 1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2012-03-14 Classification: TRANSFERASE Ligands: TQ1, SO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-14
Ligands: TQ1, SO4, EDO
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Synthesis And Evaluation Of Triazolones As Checkpoint Kinase 1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2012-03-14 Classification: TRANSFERASE Ligands: GOL, YEX, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-14
Ligands: GOL, YEX, SO4
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Discovery Of Checkpoint Kinase Inhibitor Azd7762 By Structure Based Design And Optimization Of Thiophene Carboxamide Ureas
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2012-01-25 Classification: TRANSFERASE Ligands: YDJ, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-25
Ligands: YDJ, PO4
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Jnk1 In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2011-12-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, CFK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-12-14
Ligands: SO4, CFK
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Discovery Of A Novel Class Of Triazolones As Checkpoint Kinase Inhibitors - Hit To Lead Exploration
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2010-08-11 Classification: TRANSFERASE Ligands: X8D, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-08-11
Ligands: X8D, SO4
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Discovery Of A Novel Class Of Triazolones As Checkpoint Kinase Inhibitors - Hit To Lead Exploration
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-08-11 Classification: TRANSFERASE Ligands: X8E, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-08-11
Ligands: X8E, SO4
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Discovery Of A Novel Class Of Triazolones As Checkpoint Kinase Inhibitors - Hit To Lead Exploration
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2010-08-11 Classification: TRANSFERASE Ligands: X8I, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-08-11
Ligands: X8I, SO4, GOL
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Structure-Based Design Of Protein Tyrosine Phosphatase-1B Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2005-05-04 Classification: HYDROLASE Ligands: T1D, CL, PO4, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-05-04
Ligands: T1D, CL, PO4, NA
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Structure-Based Design Of Protein Tyrosine Phosphatase-1B Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2005-05-04 Classification: HYDROLASE Ligands: T2D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2005-05-04
Ligands: T2D
