Search Count: 13
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Type-Iii C-Met Inhibitor Enabled By Free-Energy Perturbation Calculations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2026-05-27 Classification: TRANSFERASE Ligands: A1C9B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-27
Ligands: A1C9B
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Crystal Structure Of Egfr(L858R/T790M/C797S) In Complex With Aur-3418
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2025-03-05 Classification: TRANSFERASE/INHIBITOR Ligands: A1A5V, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-05
Ligands: A1A5V, CL
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Crystal Structure Of Egfr(L858R/T790M/C797S) In Complex With Aur-8250
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2025-03-05 Classification: TRANSFERASE/INHIBITOR Ligands: A1A5L, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-05
Ligands: A1A5L, CL
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Crystal Structure Of Dlk With Inhibitor Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2025-02-19 Classification: TRANSFERASE/INHIBITOR Ligands: A1AZP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1AZP
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Crystal Structure Of Dlk With Inhibitor Bound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2025-02-19 Classification: TRANSFERASE/INHIBITOR Ligands: A1AZ8, MG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-19
Ligands: A1AZ8, MG, EDO
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Identification Of Gdc-1971 (Rly-1971), A Shp2 Inhibitor Designed For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2023-10-11 Classification: HYDROLASE Ligands: SO4, YR2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-11
Ligands: SO4, YR2
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Identification Of Gdc-1971 (Rly-1971), A Shp2 Inhibitor Designed For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2023-10-11 Classification: HYDROLASE Ligands: SO4, YT2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-11
Ligands: SO4, YT2
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Identification Of Gdc-1971 (Rly-1971), A Shp2 Inhibitor Designed For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2023-10-11 Classification: HYDROLASE Ligands: ZH5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-11
Ligands: ZH5
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Identification Of Gdc-1971 (Rly-1971), A Shp2 Inhibitor Designed For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2023-10-11 Classification: HYDROLASE/INHIBITOR Ligands: ZJX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-10-11
Ligands: ZJX
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Cryo-Em Structure Of Human Atp-Citrate Lyase In Complex With Inhibitor Ndi-091143
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2019-04-17 Classification: ligase/ligase inhibitor Ligands: LBG, ADP |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2019-04-17
Ligands: LBG, ADP
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Thrombin In Complex With Inhibitor
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2006-10-24 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-10-24
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Crystal Structure Of Human Beta Secretase Complexed With Nvp-Aur200
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2006-01-17 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-01-17
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Crystal Structure Of Human Beta Secretase Complexed With Nvp-Amk640
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2006-01-17 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-01-17
