Search Count: 26
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Quinazolinone-Pyrrolodihydropyrrolone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-01-16 Classification: TRANSFERASE Ligands: JYG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-16
Ligands: JYG, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With An Imidazopyridazine Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-11-09 Classification: transferase/transferase inhibitor Ligands: 6YN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: 6YN
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Crystal Structure Of Panitumumab In Complex With Epidermal Growth Factor Receptor Domain 3.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2016-10-05 Classification: TRANSFERASE/IMMUNE SYSTEM Ligands: SO4, GOL, 1PE, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-05
Ligands: SO4, GOL, 1PE, EDO
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Crystal Structure Of Panitumumab In Complex With Epidermal Growth Factor Receptor Domain 3 Mutant S468R.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-10-05 Classification: TRANSFERASE/IMMUNE SYSTEM Ligands: SO4, GOL, EDO, 1PE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-05
Ligands: SO4, GOL, EDO, 1PE
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Quinazolinone-Pyrrolopyrrolone Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-06-22 Classification: transferase/transferase inhibitor Ligands: 6CD, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-22
Ligands: 6CD, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Macrocyclic Quinoxaline-Pyrrolodihydropiperidinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-05-04 Classification: transferase/transferase inhibitor Ligands: 5QO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 5QO, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Thiazolamine-Indazole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-02-11 Classification: transferase/transferase inhibitor Ligands: 3U5, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
Ligands: 3U5, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With A Thiadiazolamine-Indole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2015-02-11 Classification: transferase/transferase inhibitor Ligands: 3U6, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-11
Ligands: 3U6, GOL
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Co-Crystal Structure Of Pim1 With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2015-02-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3UR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: 3UR
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Crystal Structure Of Human Pim-1 Kinase In Complex With An Aminooxadiazole-Indole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2015-02-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 38W, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: 38W, GOL
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Crystal Structure Of Human Pim-1 Kinase In Complex With An Azaspiro Pyrazinyl-Indazole Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-02-04 Classification: transferase/transferase inhibitor Ligands: GOL, 3U1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-04
Ligands: GOL, 3U1
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Crystal Structure Of Human Pi3K-Gamma In Complex With (S)-N-(1-(7-Fluoro-2-(Pyridin-2-Yl)Quinolin-3-Yl)Ethyl)-9H-Purin-6-Amine Amg319 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2014-12-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 3VC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: SO4, 3VC
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Crystal Structure Of Human Pi3K-Gamma In Complex With Phenylquinoline Inhibitor N-{(1S)-1-[8-Chloro-2-(3-Fluorophenyl)Quinolin-3-Yl]Ethyl}-9H-Purin-6-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2014-12-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 3VD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: SO4, 3VD
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Crystal Structure Of Human Pi3K-Gamma In Complex With Pyridinylquinoline Inhibitor N-{(1S)-1-[8-Chloro-2-(2-Methylpyridin-3-Yl)Quinolin-3-Yl]Ethyl}-9H-Purin-6-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2014-12-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 3VE, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-12-17
Ligands: SO4, 3VE, GOL
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Crystal Structure Of Human Ire1 Cytoplasmic Domains In Complex With A Sulfonamide Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2014-10-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3E4, SO4, EDO, EPE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: 3E4, SO4, EDO, EPE
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Crystal Structure Of Human Jnk3 In Complex With A Benzenesulfonamide Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2014-10-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3EL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-08
Ligands: 3EL
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Crystal Structure Of P38A Mitogen-Activated Protein Kinase In Complex With A Triazolopyridazinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2012-08-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 09J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-08-29
Ligands: 09J
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Crystal Structure Of P38A Mitogen-Activated Protein Kinase In Complex With A Pyrazolopyridinone Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.31 Å Release Date: 2010-04-14 Classification: TRANSFERASE Ligands: LHJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-04-14
Ligands: LHJ
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Crystal Structure Of P38A Mitogen-Activated Protein Kinase In Complex With A Pyrazolopyridazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2010-03-02 Classification: TRANSFERASE Ligands: P66 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: P66
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Crystal Structure Of The Vegfr2 Kinase Domain In Complex With Motesanib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2009-09-15 Classification: TRANSFERASE Ligands: 706 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-09-15
Ligands: 706