Search Count: 54
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Cereblon In Complex With Ddb1, Gspt1 And Compound-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.90 Å Release Date: 2025-10-22 Classification: ONCOPROTEIN Ligands: ZN, A1IWG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-10-22
Ligands: ZN, A1IWG
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Sars-Cov-2 Main Protease With Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2025-10-22 Classification: VIRAL PROTEIN, HYDROLASE Ligands: A1B3B, BTB, EDO |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2025-10-22
Ligands: A1B3B, BTB, EDO
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Sars-Cov-2 Main Protease With Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2025-09-10 Classification: VIRAL PROTEIN Ligands: A1A3N |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1A3N
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Sars-Cov-2 Main Protease With Inhibitor
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2025-09-10 Classification: VIRAL PROTEIN Ligands: A1A3O |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2025-09-10
Ligands: A1A3O
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The Limk1 Kinase Domain Bound To Lijtf500025
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2020-12-23 Classification: SIGNALING PROTEIN Ligands: RXN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-23
Ligands: RXN
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The Limk1 Kinase Domain Bound To Lijtf500127
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2020-11-25 Classification: SIGNALING PROTEIN Ligands: RXQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-25
Ligands: RXQ
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P38 In Complex With T-3220137
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-11-20 Classification: TRANSFERASE/INHIBITOR Ligands: MKP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-20
Ligands: MKP
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Identification Of Novel, Potent And Selective Gcn2 Inhibitors As First-In-Class Anti-Tumor Agents
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2019-10-09 Classification: transferase/transferase inhibitor Ligands: KAV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: KAV
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Identification Of Novel, Potent And Selective Gcn2 Inhibitors As First-In-Class Anti-Tumor Agents
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.01 Å Release Date: 2019-10-09 Classification: transferase/transferase inhibitor Ligands: KA4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: KA4
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Identification Of Novel, Potent And Selective Gcn2 Inhibitors As First-In-Class Anti-Tumor Agents
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-10-09 Classification: transferase/transferase inhibitor Ligands: KA7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-09
Ligands: KA7
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Structure Of Rorgt In Complex With A Novel Inverse Agonist.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2019-07-17 Classification: nuclear protein/agonist Ligands: SO4, MPD, HQ7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: SO4, MPD, HQ7
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Structure Of Rorgt In Complex With A Novel Agonist.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-06-12 Classification: nuclear protein/agonist Ligands: EDO, HOJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-12
Ligands: EDO, HOJ
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Structure-Based Design, Synthesis, And Biological Evaluation Of Imidazo[4,5-B]Pyridine-2-One Based P38 Map Kinase Inhibitors By Scaffold Hopping: Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-04-17 Classification: TRANSFERASE Ligands: J8S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-17
Ligands: J8S
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Structure-Based Design, Synthesis, And Biological Evaluation Of Imidazo[4,5-B]Pyridine-2-One Based P38 Map Kinase Inhibitors By Scaffold Hopping - Compound 10
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2019-04-17 Classification: TRANSFERASE/INHIBITOR Ligands: J9G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-04-17
Ligands: J9G
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Structure-Based Design, Synthesis, And Biological Evaluation Of Imidazo[1,2-B]Pyridazine-Based P38 Map Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2018-01-17 Classification: Transferase/Transferase Inhibitor Ligands: AQY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: AQY
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Structure-Based Design, Synthesis, And Biological Evaluation Of Imidazo[1,2-B]Pyridazine-Based P38 Map Kinase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-01-17 Classification: TRANSFERASE Ligands: T75 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
Ligands: T75
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Compound 1A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2017-08-16 Classification: Transcription/Inhibitor Ligands: 80R, EDO, K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-16
Ligands: 80R, EDO, K
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Crystal Structure Of The Bcl6 Btb Domain In Complex With Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2017-08-16 Classification: Transcription/Inhibitor Ligands: 80L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-08-16
Ligands: 80L
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Crystal Structure Of Human Kinase Domain Of B-Raf With A Dfg-Out Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2014-01-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0T2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-01-08
Ligands: 0T2
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Crystal Structure Of Human B-Raf Bound To A Dfg-Out Inhibitor Tak-632
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.93 Å Release Date: 2013-07-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1SU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-24
Ligands: 1SU