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9HQ0 image
Sarm1 Tir Domain In Complex With Compound 7-Adpr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.13 Å Release Date: 2025-12-24
Classification: HYDROLASE
Ligands: A1IW3, EDO

9HQF image
Sarm1 Tir Domain In Complex With Compound 7-Adpr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.73 Å Release Date: 2025-12-24
Classification: HYDROLASE
Ligands: A1IWL

9HQH image
Sarm1 Tir Domain In Complex With Compound 28-Adpr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.99 Å Release Date: 2025-12-24
Classification: HYDROLASE
Ligands: A1IWN

8A27 image
Egfr Kinase Domain In Complex With 2-(6,7-Dihydro-5H-Pyrrolo[1,2-C]Imidazol-1-Yl)-2-[6-[2-[4-[[4-(Hydroxymethyl)-1-Piperidyl]Methyl]Phenyl]Ethynyl]-1-Oxo-4-(Trifluoromethyl)Isoindolin-2-Yl]-N-Thiazol-2-Yl-Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.07 Å Release Date: 2022-10-19
Classification: TRANSFERASE
Ligands: EDO, KY9, NO3

8A2A image
Egfr Kinase Domain In Complex With 2-(6,7-Dihydro-5H-Pyrrolo[1,2-C]Imidazol-1-Yl)-2-[6-[2-[4-[[4-(Hydroxymethyl)-1-Piperidyl]Methyl]Phenyl]Ethynyl]-1-Oxo-4-(Trifluoromethyl)Isoindolin-2-Yl]-N-Thiazol-2-Yl-Acetamide (Form 2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.43 Å Release Date: 2022-10-19
Classification: TRANSFERASE
Ligands: KY9, SO4

8A2B image
Egfr Kinase Domain (L858R/V948R) In Complex With 2-(6,7-Dihydro-5H-Pyrrolo[1,2-C]Imidazol-1-Yl)-2-[6-[2-[4-[[4-(Hydroxymethyl)-1-Piperidyl]Methyl]Phenyl]Ethynyl]-1-Oxo-4-(Trifluoromethyl)Isoindolin-2-Yl]-N-Thiazol-2-Yl-Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.69 Å Release Date: 2022-10-19
Classification: TRANSFERASE
Ligands: KY9

8A2D image
Egfr Kinase Domain (L858R/V948R) In Complex With 2-[4-(Difluoromethyl)-6-[2-[4-[[4-(Hydroxymethyl)-1-Piperidyl]Methyl]Phenyl]Ethynyl]-7-Methyl-Indazol-2-Yl]-2-Spiro[6,7-Dihydropyrrolo[1,2-C]Imidazole-5,1'-Cyclopropane]-1-Yl-N-Thiazol-2-Yl-Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.11 Å Release Date: 2022-10-19
Classification: TRANSFERASE
Ligands: EDO, MES, KXY

5T7D image
Crystal Structure Of Streptomyces Hygroscopicus Bialaphos Resistance (Bar) Protein In Complex With Acetyl Coenzyme A

5T7E image
Crystal Structure Of Streptomyces Hygroscopicus Bialaphos Resistance (Bar) Protein In Complex With Coenzyme A And L-Phosphinothricin

4I0R image
Crystal Structure Of Spleen Tyrosine Kinase Complexed With 2-(3,4,5-Trimethoxy-Phenyl)-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid Isopropylamide

4I0S image
Crystal Structure Of Spleen Tyrosine Kinase Complexed With 2-(6-Chloro-1-Methyl-1H-Indazol-3-Yl)-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid Isopropylamide

4I0T image
Crystal Structure Of Spleen Tyrosine Kinase Complexed With 2-(5,6,7,8-Tetrahydro-Imidazo[1,5-A]Pyridin-1-Yl)-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid Tert-Butylamide

4MK7 image
Hepatitis C Virus Polymerase Ns5B Genotype 1B (Bk) In Complex With Inhibitor 2 (3-(3-Tert-Butyl-4-Methoxyphenyl)Pyridin-2(1H)-One)

4MK8 image
Hepatitis C Virus Polymerase Ns5B Genotype 1B (Bk) In Complex With Inhibitor 4 (N-(4-{2-[3-Tert-Butyl-2-Methoxy-5-(2-Oxo-1,2-Dihydropyridin-3-Yl)Phenyl]Ethyl}Phenyl)Methanesulfonamide)

4MK9 image
Hepatitis C Virus Polymerase Ns5B Genotype 1B (Bk) In Complex With Inhibitor 12 (N-{2-[3-Tert-Butyl-2-Methoxy-5-(2-Oxo-1,2-Dihydropyridin-3-Yl)Phenyl]-1,3-Benzoxazol-5-Yl}Methanesulfonamide)

4MKA image
Hepatitis C Virus Polymerase Ns5B Genotype 1B (Bk) In Complex With Inhibitor 13 (N-{2-[3-Tert-Butyl-2-Methoxy-5-(2-Oxo-1,2-Dihydropyridin-3-Yl)Phenyl]-1,3-Benzoxazol-5-Yl}Methanesulfonamide)

4MKB image
Hepatitis C Virus Polymerase Ns5B Genotype 1B (Bk) In Complex With Inhibitor 14 (N-(4-{(E)-2-[3-Tert-Butyl-2-Methoxy-5-(3-Oxo-2,3-Dihydropyridazin-4-Yl)Phenyl]Ethenyl}Phenyl)Methanesulfonamide)

3ZC6 image
Crystal Structure Of Jak3 Kinase Domain In Complex With An Indazole Substituted Pyrrolopyrazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.42 Å Release Date: 2013-09-25
Classification: TRANSFERASE
Ligands: VFC, PEG, CL, PG4

2M0Z image
Cis Form Of A Photoswitchable Pdz Domain Crosslinked With An Azobenzene Derivative

2M10 image
Trans Form Of A Photoswitchable Pdz Domain Crosslinked With An Azobenzene Derivative
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