Search Count: 24
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Sarm1 Tir Domain In Complex With Compound 7-Adpr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: A1IW3, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1IW3, EDO
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Sarm1 Tir Domain In Complex With Compound 7-Adpr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: A1IWL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1IWL
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Sarm1 Tir Domain In Complex With Compound 28-Adpr
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2025-12-24 Classification: HYDROLASE Ligands: A1IWN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-12-24
Ligands: A1IWN
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Egfr Kinase Domain In Complex With 2-(6,7-Dihydro-5H-Pyrrolo[1,2-C]Imidazol-1-Yl)-2-[6-[2-[4-[[4-(Hydroxymethyl)-1-Piperidyl]Methyl]Phenyl]Ethynyl]-1-Oxo-4-(Trifluoromethyl)Isoindolin-2-Yl]-N-Thiazol-2-Yl-Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.07 Å Release Date: 2022-10-19 Classification: TRANSFERASE Ligands: EDO, KY9, NO3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-19
Ligands: EDO, KY9, NO3
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Egfr Kinase Domain In Complex With 2-(6,7-Dihydro-5H-Pyrrolo[1,2-C]Imidazol-1-Yl)-2-[6-[2-[4-[[4-(Hydroxymethyl)-1-Piperidyl]Methyl]Phenyl]Ethynyl]-1-Oxo-4-(Trifluoromethyl)Isoindolin-2-Yl]-N-Thiazol-2-Yl-Acetamide (Form 2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2022-10-19 Classification: TRANSFERASE Ligands: KY9, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-19
Ligands: KY9, SO4
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Egfr Kinase Domain (L858R/V948R) In Complex With 2-(6,7-Dihydro-5H-Pyrrolo[1,2-C]Imidazol-1-Yl)-2-[6-[2-[4-[[4-(Hydroxymethyl)-1-Piperidyl]Methyl]Phenyl]Ethynyl]-1-Oxo-4-(Trifluoromethyl)Isoindolin-2-Yl]-N-Thiazol-2-Yl-Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2022-10-19 Classification: TRANSFERASE Ligands: KY9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-19
Ligands: KY9
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Egfr Kinase Domain (L858R/V948R) In Complex With 2-[4-(Difluoromethyl)-6-[2-[4-[[4-(Hydroxymethyl)-1-Piperidyl]Methyl]Phenyl]Ethynyl]-7-Methyl-Indazol-2-Yl]-2-Spiro[6,7-Dihydropyrrolo[1,2-C]Imidazole-5,1'-Cyclopropane]-1-Yl-N-Thiazol-2-Yl-Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.11 Å Release Date: 2022-10-19 Classification: TRANSFERASE Ligands: EDO, MES, KXY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-10-19
Ligands: EDO, MES, KXY
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Crystal Structure Of Streptomyces Hygroscopicus Bialaphos Resistance (Bar) Protein In Complex With Acetyl Coenzyme A
Organism: Streptomyces hygroscopicus
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2017-06-07 Classification: TRANSFERASE Ligands: ACO, ACT |
Organism: Streptomyces hygroscopicus
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: ACO, ACT
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Crystal Structure Of Streptomyces Hygroscopicus Bialaphos Resistance (Bar) Protein In Complex With Coenzyme A And L-Phosphinothricin
Organism: Streptomyces hygroscopicus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2017-06-07 Classification: TRANSFERASE Ligands: COA, PPQ, BNG |
Organism: Streptomyces hygroscopicus
Method: X-RAY DIFFRACTION
Release Date: 2017-06-07
Ligands: COA, PPQ, BNG
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Crystal Structure Of Spleen Tyrosine Kinase Complexed With 2-(3,4,5-Trimethoxy-Phenyl)-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid Isopropylamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2013-10-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1B4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-30
Ligands: 1B4
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Crystal Structure Of Spleen Tyrosine Kinase Complexed With 2-(6-Chloro-1-Methyl-1H-Indazol-3-Yl)-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid Isopropylamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2013-10-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1B5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-30
Ligands: 1B5
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Crystal Structure Of Spleen Tyrosine Kinase Complexed With 2-(5,6,7,8-Tetrahydro-Imidazo[1,5-A]Pyridin-1-Yl)-5H-Pyrrolo[2,3-B]Pyrazine-7-Carboxylic Acid Tert-Butylamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2013-10-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1B6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-10-30
Ligands: 1B6
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Hepatitis C Virus Polymerase Ns5B Genotype 1B (Bk) In Complex With Inhibitor 2 (3-(3-Tert-Butyl-4-Methoxyphenyl)Pyridin-2(1H)-One)
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2013-10-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: MG, DMS, 28O |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2013-10-09
Ligands: MG, DMS, 28O
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Hepatitis C Virus Polymerase Ns5B Genotype 1B (Bk) In Complex With Inhibitor 4 (N-(4-{2-[3-Tert-Butyl-2-Methoxy-5-(2-Oxo-1,2-Dihydropyridin-3-Yl)Phenyl]Ethyl}Phenyl)Methanesulfonamide)
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2013-10-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: DMS, 28Q, GOL |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2013-10-09
Ligands: DMS, 28Q, GOL
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Hepatitis C Virus Polymerase Ns5B Genotype 1B (Bk) In Complex With Inhibitor 12 (N-{2-[3-Tert-Butyl-2-Methoxy-5-(2-Oxo-1,2-Dihydropyridin-3-Yl)Phenyl]-1,3-Benzoxazol-5-Yl}Methanesulfonamide)
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2013-10-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 28R, GOL |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2013-10-09
Ligands: 28R, GOL
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Hepatitis C Virus Polymerase Ns5B Genotype 1B (Bk) In Complex With Inhibitor 13 (N-{2-[3-Tert-Butyl-2-Methoxy-5-(2-Oxo-1,2-Dihydropyridin-3-Yl)Phenyl]-1,3-Benzoxazol-5-Yl}Methanesulfonamide)
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2013-10-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, 2AY, DMS |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2013-10-09
Ligands: GOL, 2AY, DMS
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Hepatitis C Virus Polymerase Ns5B Genotype 1B (Bk) In Complex With Inhibitor 14 (N-(4-{(E)-2-[3-Tert-Butyl-2-Methoxy-5-(3-Oxo-2,3-Dihydropyridazin-4-Yl)Phenyl]Ethenyl}Phenyl)Methanesulfonamide)
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2013-10-09 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 28V |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2013-10-09
Ligands: 28V
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Crystal Structure Of Jak3 Kinase Domain In Complex With An Indazole Substituted Pyrrolopyrazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2013-09-25 Classification: TRANSFERASE Ligands: VFC, PEG, CL, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-25
Ligands: VFC, PEG, CL, PG4
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Cis Form Of A Photoswitchable Pdz Domain Crosslinked With An Azobenzene Derivative
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2013-07-03 Classification: HYDROLASE Ligands: 33B |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2013-07-03
Ligands: 33B
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Trans Form Of A Photoswitchable Pdz Domain Crosslinked With An Azobenzene Derivative
Organism: Homo sapiens
Method: SOLUTION NMR Release Date: 2013-07-03 Classification: HYDROLASE Ligands: 33B |
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2013-07-03
Ligands: 33B
