Search Count: 73
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Co-Crystal Structure Of P. Aeruginosa Lpxc-50067 Complex
Organism: Pseudomonas aeruginosa pao1
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2019-07-17 Classification: HYDROLASE/INHIBITOR Ligands: MG, JWM |
Organism: Pseudomonas aeruginosa pao1
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: MG, JWM
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Co-Crystal Structure Of P. Aeruginosa Lpxc-50228 Complex
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-07-17 Classification: HYDROLASE/INHIBITOR Ligands: JWP, MG |
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Co-Crystal Structure Of P. Aeruginosa Lpxc-50432 Complex
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-07-17 Classification: HYDROLASE/INHIBITOR Ligands: MG, JWV, GOL |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: MG, JWV, GOL
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Co-Crystal Structure Of P. Aeruginosa Lpxc-Achn975 Complex
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-07-17 Classification: HYDROLASE/INHIBITOR Ligands: ZN, A5F |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2019-07-17
Ligands: ZN, A5F
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Crystal Structure Of T110A Mutant Human Glutamate Oxaloacetate Transaminase 1 (Got1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2018-11-14 Classification: TRANSFERASE Ligands: PG4, PLP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-14
Ligands: PG4, PLP
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Crystal Structure Of T110A:S256A Mutant Human Glutamate Oxaloacetate Transaminase 1 (Got1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2018-11-14 Classification: TRANSFERASE Ligands: PG4, GOL, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-14
Ligands: PG4, GOL, PO4
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Crystal Structure Of Wild-Type (Wt) Human Glutamate Oxaloacetate Transaminase 1 (Got1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-11-14 Classification: TRANSFERASE Ligands: PG4, PLP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-11-14
Ligands: PG4, PLP
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Glycogen Synthase Kinase 3 Beta Complexed With Brd0209
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VK
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Glycogen Synthase Kinase 3 Beta Complexed With Brd0705
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VL
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Glycogen Synthase Kinase 3 Beta Complexed With Brd3731
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.69 Å Release Date: 2018-03-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6VM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: 6VM
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Exploiting An Asp-Glu Switch In Glycogen Synthase Kinase 3 To Design Paralog Selective Inhibitors For Use In Acute Myeloid Leukemia
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2018-02-21 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 6VL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-21
Ligands: 6VL
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Tryptophan 5-Hydroxylase In Complex With Inhibitor (3~{S})-8-[2-Azanyl-6-[(1~{R})-1-(4-Chloranyl-2-Phenyl-Phenyl)-2,2,2-Tris(Fluoranyl)Ethoxy]Pyrimidin-4-Yl]-2,8-Diazaspiro[4.5]Decane-3-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-01-25 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: FE, 6Z4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: FE, 6Z4
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Optimization Of Spirocyclic Proline Tryptophanhydroxylase-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2017-01-25 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor Ligands: FE, TRS, CCN, 7H5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: FE, TRS, CCN, 7H5
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Selective Inhibition Of Autotaxin Is Effective In Mouse Models Of Liver Fibrosis
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2016-11-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NAG, ZN, CA, 6Y7, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-09
Ligands: NAG, ZN, CA, 6Y7, PO4
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Discovery Of Acyl Guanidine Tryptophan Hydroxylase-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2016-05-25 Classification: OXIDOREDUCTASE/INHIBITOR Ligands: FE, TRS, GOL, 6H5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: FE, TRS, GOL, 6H5
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Structural Basis For Inhibition Of Human Autotaxin By Four Novel Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-10-14 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, CA, NA, GOL, 4NY, SCN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-14
Ligands: ZN, CA, NA, GOL, 4NY, SCN
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Structural Basis For Inhibition Of Human Autotaxin By Four Novel Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2015-10-14 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, CA, NA, 4O0, NKN, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-14
Ligands: ZN, CA, NA, 4O0, NKN, GOL, CL
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Structural Basis For Inhibition Of Human Autotaxin By Four Novel Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.95 Å Release Date: 2015-10-14 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, CA, NA, 4O2, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-14
Ligands: ZN, CA, NA, 4O2, EDO
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Structural Basis For Inhibition Of Human Autotaxin By Four Novel Compounds
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2015-10-14 Classification: Hydrolase/Hydrolase Inhibitor Ligands: ZN, CA, EDO, SCN, ACD, 4O3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-14
Ligands: ZN, CA, EDO, SCN, ACD, 4O3
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The Crystal Structure Of Lin0861 From Listeria Innocua To 2.8A
Organism: Listeria innocua
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2010-09-29 Classification: Structural Genomics, Unknown function Ligands: SO4 |
Organism: Listeria innocua
Method: X-RAY DIFFRACTION
Release Date: 2010-09-29
Ligands: SO4