Search Count: 28
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Factor Xia In Complex With Compound 2A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-08-03 Classification: Blood Clotting, Hydrolase Ligands: OQ6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: OQ6
 |
Factor Xia In Complex With Compound 2D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: OQI, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: OQI, CIT
 |
Factor Xia In Complex With Compound 2E
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, hydrolase Ligands: OQO, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: OQO, CIT
 |
Factor Xia In Complex With Compound 2F
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: OR0, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: OR0, CIT
 |
Factor Xia In Complex With Compound 2G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, ORF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, ORF
 |
Factor Xia In Complex With Compound 2H
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, ORU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, ORU
 |
Factor Xia In Complex With Compound 2I
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, OSX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, OSX
 |
Factor Xia In Complex With Compound 2J
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, OT7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, OT7
 |
Factor Xia In Complex With Compound 2K
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, OTL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, OTL
 |
Factor Xia In Complex With Compound 3F
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, OTX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, OTX
 |
Structure Of A Hit For G Protein Coupled Receptor Kinase 2 (Grk2) Inhibitor For The Potential Treatment Of Heart Failure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2020-10-28 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: MG, W4D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: MG, W4D
 |
Structure Of A Hit For G Protein Coupled Receptor Kinase 2 (Grk2) Inhibitor For The Potential Treatment Of Heart Failure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2020-10-28 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: W4G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: W4G
 |
Discovery And Clinical Evaluation Of Rwj-671818, A Thrombin Inhibitor With An Oxyguanidine P1 Motif
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2011-08-10 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: NLI |
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION
Release Date: 2011-08-10
Ligands: NLI
 |
Cyanofluorophenylacetamides As Orally Efficacious Thrombin Inhibitors
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2009-02-17 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: DKK |
Organism: Homo sapiens, Hirudo medicinalis
Method: X-RAY DIFFRACTION
Release Date: 2009-02-17
Ligands: DKK
 |
Potent, Nonpeptide Inhibitors Of Human Mast Cell Tryptase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2008-12-09 Classification: HYDROLASE Ligands: 11M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-12-09
Ligands: 11M
 |
Potent, Nonpeptide Inhibitors Of Human Mast Cell Tryptase
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2008-12-09 Classification: HYDROLASE Ligands: 11N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-12-09
Ligands: 11N
 |
Crystal Structure Of Human Tryptase With Potent Non-Peptide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-02-26 Classification: HYDROLASE Ligands: 2FF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-02-26
Ligands: 2FF
 |
C-Fms Tyrosine Kinase In Complex With A Quinolone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2006-11-28 Classification: TRANSFERASE Ligands: SO4, 6C3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-11-28
Ligands: SO4, 6C3
 |
Cfms Tyrosine Kinase (Fgf Kid) In Complex With An Arylamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2006-11-28 Classification: TRANSFERASE Ligands: 5CN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-11-28
Ligands: 5CN
 |
Cfms Tyrosine Kinase (Tie2 Kid) In Complex With An Arylamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2006-11-28 Classification: TRANSFERASE Ligands: 5CN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2006-11-28
Ligands: 5CN