Search Count: 50
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An Rorgt Inverse Agonist For Treatment Of Psoriasis
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2025-04-30 Classification: NUCLEAR PROTEIN Ligands: A1BW2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-30
Ligands: A1BW2
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Factor Xia In Complex With Compound 2A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-08-03 Classification: Blood Clotting, Hydrolase Ligands: OQ6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: OQ6
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Factor Xia In Complex With Compound 2D
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: OQI, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: OQI, CIT
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Factor Xia In Complex With Compound 2E
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.47 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, hydrolase Ligands: OQO, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: OQO, CIT
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Factor Xia In Complex With Compound 2F
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: OR0, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: OR0, CIT
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Factor Xia In Complex With Compound 2G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, ORF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, ORF
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Factor Xia In Complex With Compound 2H
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, ORU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, ORU
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Factor Xia In Complex With Compound 2I
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, OSX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, OSX
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Factor Xia In Complex With Compound 2J
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.51 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, OT7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, OT7
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Factor Xia In Complex With Compound 2K
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, OTL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, OTL
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Factor Xia In Complex With Compound 3F
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2022-08-03 Classification: BLOOD CLOTTING, Hydrolase Ligands: CIT, OTX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: CIT, OTX
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Structure Of A Hit For G Protein Coupled Receptor Kinase 2 (Grk2) Inhibitor For The Potential Treatment Of Heart Failure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2020-10-28 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: MG, W4D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: MG, W4D
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Structure Of A Hit For G Protein Coupled Receptor Kinase 2 (Grk2) Inhibitor For The Potential Treatment Of Heart Failure
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2020-10-28 Classification: SIGNALING PROTEIN,TRANSFERASE/INHIBITOR Ligands: W4G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-28
Ligands: W4G
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Optimization And Biological Evaluation Of Thiazole-Bis-Amide Inverse Agonists Of Rorgt
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2020-05-13 Classification: NUCLEAR PROTEIN Ligands: RG7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-05-13
Ligands: RG7
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Identification And Biological Evaluation Of Tertiary Alcohol-Based Inverse Agonists Of Rorgt
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2019-05-08 Classification: NUCLEAR PROTEIN Ligands: KHY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-05-08
Ligands: KHY
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Identification And Biological Evaluation Of Thiazole-Based Inverse Agonists Of Rorgt
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2018-04-25 Classification: NUCLEAR PROTEIN Ligands: FJG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-25
Ligands: FJG
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Structure Of Rorgt Bound To A Tertiary Alcohol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2017-12-27 Classification: NUCLEAR PROTEIN Ligands: 9WD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: 9WD
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Structure Of Rorgt Bound To A Tertiary Alcohol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2017-12-27 Classification: NUCLEAR PROTEIN Ligands: 9WA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-27
Ligands: 9WA
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Prommp-9Desfnii
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2017-09-13 Classification: HYDROLASE Ligands: ZN, CA, SO4, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-13
Ligands: ZN, CA, SO4, TRS
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Prommp-9Desfnii Complexed To Jnj0966 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2017-09-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, CA, SO4, 5XQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-13
Ligands: ZN, CA, SO4, 5XQ
