Search Count: 10
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First Bromodomain Of Brdt Liganded With Inhibitor Gxh-Iv-076 (Compound 33)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2026-07-29 Classification: TRANSCRIPTION/INHIBITOR Ligands: ZNJ, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-29
Ligands: ZNJ, EDO, CL
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Brd4 Bd1 Liganded With Macrocyclic Compound 2B (Jj-Ii-352A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2025-03-19 Classification: TRANSCRIPTION Ligands: A1AAL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-19
Ligands: A1AAL, EDO
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Brd4 Bd1 Liganded With Macrocyclic Compound 2D (Jj-Ii-363A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.22 Å Release Date: 2024-12-18 Classification: TRANSCRIPTION Ligands: YPB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: YPB, EDO
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Crystal Structure Of The First Bromodomain (Bd1) Of Human Brd4 Bound To Gxh-Ii-076
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2022-05-11 Classification: GENE REGULATION Ligands: ZNJ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-11
Ligands: ZNJ, EDO
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Anthrax Toxin Lethal Factor With Hydroxamic Acid Inhibitor
Organism: Bacillus anthracis
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2015-11-11 Classification: Hydrolase/hydrolase inhibitor Ligands: 56Q, ZN |
Organism: Bacillus anthracis
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: 56Q, ZN
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Anthrax Toxin Lethal Factor With Hydroxamic Acid Inhibitor
Organism: Bacillus anthracis
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2015-11-11 Classification: hydrolase/hydrolase inhibitor Ligands: ZN, 56R |
Organism: Bacillus anthracis
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: ZN, 56R
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Anthrax Toxin Lethal Factor With Hydroxamic Acid Inhibitor
Organism: Bacillus anthracis
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2015-11-11 Classification: Hydrolase/hydrolase inhibitor Ligands: 56P, ZN |
Organism: Bacillus anthracis
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: 56P, ZN
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Anthrax Toxin Lethal Factor With Bound Small Molecule Inhibitor Mk-31
Organism: Bacillus anthracis
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2015-09-09 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: ZN, 407, EDO |
Organism: Bacillus anthracis
Method: X-RAY DIFFRACTION
Release Date: 2015-09-09
Ligands: ZN, 407, EDO
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First-In-Class Small Molecule Inhibitors Of The Single-Strand Dna Cytosine Deaminase Apobec3G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2012-02-01 Classification: HYDROLASE Ligands: ZN, PQR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-01
Ligands: ZN, PQR
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First-In-Class Small Molecule Inhibitors Of The Single-Strand Dna Cytosine Deaminase Apobec3G
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2012-01-25 Classification: HYDROLASE Ligands: CL, MG, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-01-25
Ligands: CL, MG, ZN
