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Search Count: 28

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9TDA image
Erap1 In Complex With 1-[2-(5-Bromo-7-Fluoro-2-Oxo-2,3-Dihydro-1,3-Benzothiazol-3-Yl)Acetamido]-4,4-Difluorocyclohexane-1-Carboxylic Acid

9TD3 image
Erap1 In Complex With 1-[2-(6-Bromo-2,2-Difluoro-3-Oxo-3,4-Dihydro-2H-1,4-Benzoxazin-4-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid

9TD4 image
Erap1 In Complex With 1-[2-(2-Oxo-5-Phenyl-2,3-Dihydro-1,3-Benzoxazol-3-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid

9TD5 image
Erap1 In Complex With 1-[2-(5-Chloro-2-Oxo-2,3-Dihydro-1,3-Benzothiazol-3-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid

9TD7 image
Erap1 In Complex With 1-[2-(3-Oxo-6-Phenyl-3,4-Dihydro-2H-1,4-Benzoxazin-4-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid

8ZLD image
Crystal Structure Of Pfho From Plasmodium Falciparum At 2.78 A

7AX4 image
Human Tyk2 Pseudokinase Domain (575-869) In Complex With 5-(4-Fluoro-Phenyl)-2-Ureido-Thiophene-3-Carboxylic Acid Amide.

5NA5 image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) Apo Structure

5NAB image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With 3-(5-Chloro-6-Methyl-2-Oxo-2,3-Dihydro-1,3-Benzoxazol-3-Yl)Propanoic Acid

5NAE image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With 3-{5-Chloro-2-Oxo-6-[(1R)-1-(Pyridin-2-Yl)Ethoxy]-2,3-Dihydro-1,3-Benzoxazol-3-Yl}Propanoic Acid

5NAG image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With 3-{5-Chloro-6-[(1R)-1-(Pyridin-2-Yl)Ethoxy]-1,2-Benzoxazol-3-Yl}Propanoic Acid

5NAH image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With 3-{5-Chloro-6-[(1R)-1-(6-Methylpyridazin-3-Yl)Ethoxy]-1,2-Benzoxazol-3-Yl}Propanoic Acid

5NAK image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With The Enzyme Substrate L-Kynurenine

5N7T image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With 3-(5,6-Dichloro-2-Oxo-2,3-Dihydro-1,3-Benzoxazol-3-Yl)Propanoic Acid

5MZC image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With 3-(5-Chloro-6-Ethoxy-2-Oxo-2,3-Dihydro-1,3-Benzoxazol-3-Yl)Propanoic Acid

5MZI image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With 3-(5-Chloro-6-Cyclopropoxy-2-Oxo-2,3-Dihydro-1,3-Benzoxazol-3-Yl)Propanoic Acid

5MZK image
Pseudomonas Fluorescens Kynurenine 3-Monooxygenase (Kmo) In Complex With 3-[5-Chloro-6-(Cyclobutylmethoxy)-2-Oxo-2,3-Dihydro-1,3-Benzoxazol-3-Yl]Propanoic Acid

5FP7 image
Crystal Structure Of Human Kdm4D In Complex With 3-4-Methylthiophen-2- Yl Methylaminopyridine-4-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2016-11-09
Classification: INHIBITOR
Ligands: ZN, FE2, GOL, YC8, SO4

5FP3 image
Cell Penetrant Inhibitors Of The Jmjd2 (Kdm4) And Jarid1 (Kdm5) Families Of Histone Lysine Demethylases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.05 Å Release Date: 2016-01-27
Classification: OXIDOREDUCTASE
Ligands: YC8, ZN, MG, BCN, CO

5FP4 image
Crystal Structure Of Human Kdm4D In Complex With 3-(4- Phenylbutanamido)Pyridine-4-Carboxylic Acid
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