Search Count: 21
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Monkey Tlr7 Ectodomain With Small Molecule Agonist 9
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2025-03-05 Classification: IMMUNE SYSTEM Ligands: NAG, CL, A1BLT, CIT |
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION
Release Date: 2025-03-05
Ligands: NAG, CL, A1BLT, CIT
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Human Tlr8 Ectodomain With Small Molecule Agonist 9
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2025-03-05 Classification: IMMUNE SYSTEM Ligands: NAG, NI, A1BLT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-05
Ligands: NAG, NI, A1BLT
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Human Tlr8 Ectodomain With Small Molecule Agonist 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2025-03-05 Classification: IMMUNE SYSTEM Ligands: NAG, A1BLO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-05
Ligands: NAG, A1BLO
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Human Tlr8 Ectodomain With Small Molecule Agonist 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2025-03-05 Classification: IMMUNE SYSTEM Ligands: NAG, SO4, A1BLN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-05
Ligands: NAG, SO4, A1BLN
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Crystal Structure Of Monkey Tlr7 Ectodomain With Compound 14
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2024-02-07 Classification: IMMUNE SYSTEM Ligands: NAG, ZWV, SO4 |
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: NAG, ZWV, SO4
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Crystal Structure Of Monkey Tlr7 Ectodomain With Compound 5
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2024-02-07 Classification: IMMUNE SYSTEM Ligands: NAG, QEC, SO4 |
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: NAG, QEC, SO4
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Crystal Structure Of Monkey Tlr7 Ectodomain With Compound 20
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION Resolution:3.14 Å Release Date: 2024-02-07 Classification: IMMUNE SYSTEM Ligands: NAG, SO4, QCX |
Organism: Macaca mulatta
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: NAG, SO4, QCX
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Crystal Structure Of Glycogen Synthase Kinase 3 Beta Complexed With 2-[(4-Cyanophenyl)Amino]-N-(4-Phenylpyridin-3-Yl)Pyrimidine-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2023-06-07 Classification: TRANSFERASE/INHIBITOR Ligands: XV0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: XV0
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Crystal Structure Of Glycogen Synthase Kinase 3 Beta Complexed With (4S)-N-{4-[(2S)-2-Methylmorpholin-4-Yl] Pyridin-3-Yl}-2-Phenylimidazo[1,2-B]Pyridazine-8-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2023-03-22 Classification: TRANSFERASE/INHIBITOR Ligands: UAU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-22
Ligands: UAU
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Crystal Structure Of Glycogen Synthase Kinase 3 Beta Complexed With 3-[(Cyclopropylmethyl)Amino] -N-(4-Phenylpyridin-3-Yl)Imidazo[1,2-B]Pyridazine-8-Carbox Amide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2023-03-22 Classification: TRANSFERASE/INHIBITOR Ligands: U6S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-03-22
Ligands: U6S
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Crystal Structure Of Hiv-1 Integrase Complexed With (2S)-2-(Tert-Butoxy)-2-(5-{2-[(2-Chloro-6-M Ethylphenyl)Methyl]-1,2,3,4-Tetrahydroisoquinolin-6-Yl}-4- (4,4-Dimethylpiperidin-1-Yl)-2-Methylpyridin-3-Yl)Acetic Acid
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2022-07-06 Classification: TRANSFERASE Ligands: O20, SO4 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2022-07-06
Ligands: O20, SO4
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Crystal Structure Of Hiv-1 Integrase Complexed With Compound-2A Aka (2S)-2-(Tert-Butoxy)-2-[7-(4,4-Dimethylpipe Ridin-1-Yl)-8-{4-[2-(4-Fluorophenyl)Ethoxy]Phenyl}-2,5-Dim Ethylimidazo[1,2-A]Pyridin-6-Yl]Acetic Acid
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2022-06-08 Classification: DNA BINDING PROTEIN, viral protein Ligands: KZD, SO4 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2022-06-08
Ligands: KZD, SO4
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Hiv Integrase In Complex With Compound-15
Organism: human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2022-04-06 Classification: DNA BINDING PROTEIN, Viral protein Ligands: MG, GE7 |
Organism: human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2022-04-06
Ligands: MG, GE7
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Hiv Integrase In Complex With Compound-25
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2022-04-06 Classification: DNA BINDING PROTEIN, Viral Protein Ligands: SO4, GEI, GOL |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2022-04-06
Ligands: SO4, GEI, GOL
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Structure Of Human Pregnane X Receptor Ligand Binding Domain Bound Tethered With Src Co-Activator Peptide In Complex With (S,S)-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2020-09-23 Classification: NUCLEAR PROTEIN Ligands: QCG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: QCG, GOL
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Hiv Integrase In Complex With Compound-14
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2020-03-04 Classification: TRANSFERASE,Hydrolase Ligands: 1PE, PEG, QCG, SO4 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2020-03-04
Ligands: 1PE, PEG, QCG, SO4
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Crystal Structure Of Gsk3B In Complex With Compound 15: 2-[(Cyclopropylcarbonyl)Amino]-N-(4-Methoxypyridin-3-Yl)Pyridine-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2016-02-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3UO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 3UO
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Crystal Structure Of Gsk3B In Complex With Compound 18: 2-[(Cyclopropylcarbonyl)Amino]-N-(4-Phenylpyridin-3-Yl)Pyridine-4-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2016-02-03 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 3UP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-03
Ligands: 3UP
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Structure Of A Carboxamide Compound (3) (2-{2-[(Cyclopropylcarbonyl)Amino]Pyridin-4-Yl}-4-Oxo-4H-1Lambda~4~,3-Thiazole-5-Carboxamide) To Gsk3B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.71 Å Release Date: 2015-04-08 Classification: transferase/transferase inhibitor Ligands: 2WE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-08
Ligands: 2WE
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Structure Of A Carvoxamide Compound (15) (N-[4-(Isoquinolin-7-Yl)Pyridin-2-Yl]Cyclopropanecarboxamide) To Gsk3B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2015-04-08 Classification: transferase/transferase inhibitor Ligands: 2WF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-08
Ligands: 2WF
