Search Count: 26
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Crystal Structure Of Human Pkmyt1 Protein Kinase Domain With Naphthyridinone Inhibitor Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2026-03-25 Classification: TRANSFERASE Ligands: A1E5A, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-03-25
Ligands: A1E5A, SO4
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Crystal Structure Of Human Pkmyt1 Protein Kinase Domain With Naphthyridinone Inhibitor Compound 16
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2026-03-25 Classification: TRANSFERASE Ligands: A1E5J, DMS, EDO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-03-25
Ligands: A1E5J, DMS, EDO, SO4
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Crystal Structure Of H5N1 Influenza Polymerase Pb2 Domain In Complex With Compound 3
Organism: Influenza a virus (a/duck/shantou/4610/2003(h5n1))
Method: X-RAY DIFFRACTION Resolution:0.91 Å Release Date: 2026-01-28 Classification: TRANSFERASE Ligands: A1JV9, SO4 |
Organism: Influenza a virus (a/duck/shantou/4610/2003(h5n1))
Method: X-RAY DIFFRACTION
Release Date: 2026-01-28
Ligands: A1JV9, SO4
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 1 In Complex With Atp Competitive Inhibitor 29
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2025-06-25 Classification: TRANSFERASE Ligands: SO4, TF3, EDO, GOL, A1EQH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-25
Ligands: SO4, TF3, EDO, GOL, A1EQH
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 2 In Complex With Atp Competitive Inhibitor 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2025-06-25 Classification: TRANSFERASE Ligands: EDO, TF3, GOL, A1EQJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-25
Ligands: EDO, TF3, GOL, A1EQJ
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 2 In Complex With Atp Competitive Inhibitor 22
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2025-06-11 Classification: TRANSFERASE Ligands: TF3, A1EQI, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-11
Ligands: TF3, A1EQI, DMS
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Crystal Structure Of Human Pkmyt1 Protein Kinase Domain With Naphthyridinone Inhibitor Compound 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2025-05-14 Classification: TRANSFERASE Ligands: A1EJW, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1EJW, EDO, CL
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Crystal Structure Of Human Pkmyt1 Protein Kinase Domain With Naphthyridinone Inhibitor Compound 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2025-05-14 Classification: TRANSFERASE Ligands: A1EJX, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1EJX, SO4
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Crystal Structure Of Human Pkmyt1 Protein Kinase Domain With Naphthyridinone Inhibitor Compound 40
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2025-04-16 Classification: TRANSFERASE Ligands: A1EJU, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-16
Ligands: A1EJU, SO4
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Crystal Structure Of Human Pkmyt1 Protein Kinase Domain With Naphthyridinone Inhibitor Compound 11
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2025-04-16 Classification: TRANSFERASE Ligands: TLA, A1EJV, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-16
Ligands: TLA, A1EJV, EDO
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 1 In Complex With Atp Competitive Inhibitor 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2025-04-02 Classification: TRANSFERASE Ligands: K, A1EMR, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-02
Ligands: K, A1EMR, GOL
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Crystal Structure Of Human Pyruvate Dehydrogenase Kinase Isoform 1 In Complex With Atp Competitive Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.01 Å Release Date: 2025-04-02 Classification: TRANSFERASE Ligands: K, SZ6, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-02
Ligands: K, SZ6, GOL
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Hepatitis B Virus Core Protein Y132A Mutant In Complex With Thpp Derivatives 48
Organism: Hepatitis b virus adw/991
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2023-10-25 Classification: VIRAL PROTEIN Ligands: IPA, VX0, GOL |
Organism: Hepatitis b virus adw/991
Method: X-RAY DIFFRACTION
Release Date: 2023-10-25
Ligands: IPA, VX0, GOL
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Hepatitis B Virus Core Protein Y132A Mutant In Complex With Linvencorvir (Rg7907), A Hepatitis B Virus (Hbv) Core Protein Allosteric Modulator (Cpam)
Organism: Hepatitis b virus subtype adyw
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2023-03-22 Classification: VIRAL PROTEIN Ligands: CL, IPA, GOL, OTI, DMS |
Organism: Hepatitis b virus subtype adyw
Method: X-RAY DIFFRACTION
Release Date: 2023-03-22
Ligands: CL, IPA, GOL, OTI, DMS
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The Dna Gyrase B Atp Binding Domain Of Pseudomonas Aeruginosa In Complex With Compound 12X
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2020-09-02 Classification: ISOMERASE Ligands: DMS, SO4, NA, EZ6 |
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION
Release Date: 2020-09-02
Ligands: DMS, SO4, NA, EZ6
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The Dna Gyrase B Atp Binding Domain Of Pseudomonas Aeruginosa In Complex With Compound 12O
Organism: Pseudomonas aeruginosa (strain atcc 15692 / dsm 22644 / cip 104116 / jcm 14847 / lmg 12228 / 1c / prs 101 / pao1)
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2020-09-02 Classification: ISOMERASE Ligands: EZ9, SO4, CL |
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Crystal Structure Of Tead2 Bound To Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2020-06-24 Classification: Transcription/Transcription Inhibitor Ligands: GOL, QSJ, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-24
Ligands: GOL, QSJ, TRS
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Crystal Structure Of Tead2 Bound To Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2020-06-24 Classification: TRANSCRIPTION/INHIBITOR Ligands: QLV, TRS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-24
Ligands: QLV, TRS
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Structure Of Aldosterone Synthase (Cyp11B2) In Complex With N-[(1R)-1-[5-(6-Chloro-1,1-Dimethyl-3-Oxo-Isoindolin-2-Yl)-3-Pyridyl]Ethyl]Methanesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2020-06-24 Classification: OXIDOREDUCTASE Ligands: HEC, O4T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-24
Ligands: HEC, O4T
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Structure Of Aldosterone Synthase (Cyp11B2) In Complex With 5-Chloro-3,3-Dimethyl-2-[5-[1-(1-Methylpyrazole-4-Carbonyl)Azetidin-3-Yl]Oxy-3-Pyridyl]Isoindolin-1-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.77 Å Release Date: 2020-06-24 Classification: OXIDOREDUCTASE Ligands: HEC, O4W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-24
Ligands: HEC, O4W
