Search Count: 21
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Crystal Structure Of Integrin-Linked Kinase (Ilk) In Complex With Alpha-Parvin And Dihydropelitinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2026-06-03 Classification: CELL ADHESION Ligands: A1JW8, EPE, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-03
Ligands: A1JW8, EPE, EDO
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Crystal Structure Of Integrin-Linked Kinase (Ilk) In Complex With Alpha-Parvin And A Cyano-Quinoline Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2026-06-03 Classification: CELL ADHESION Ligands: A1JW7, EDO, EPE, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-03
Ligands: A1JW7, EDO, EPE, NA
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Usp28 Usp Domain In Complex With T-10531
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2026-05-06 Classification: ONCOPROTEIN Ligands: CL, MES, A1JQP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-05-06
Ligands: CL, MES, A1JQP
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Structure Of The C-Terminal Half Of Lrrk2 Bound To Rn277 (Type-Ii Inhibitor)
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY Resolution:3.35 Å Release Date: 2025-06-18 Classification: PROTEIN BINDING Ligands: A1A7Q |
Organism: Homo sapiens, Synthetic construct
Method: ELECTRON MICROSCOPY
Release Date: 2025-06-18
Ligands: A1A7Q
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Human Trim21 Pryspry Domain In Complex With Al236
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2025-03-12 Classification: LIGASE Ligands: A1I41, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-12
Ligands: A1I41, EDO
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Crystal Structure Of Human Clk3 Bound To Rn129
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2024-09-11 Classification: TRANSFERASE Ligands: SO4, A1H74 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-11
Ligands: SO4, A1H74
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Dual Bet/Hdac Inhibitor Nb161
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2023-07-05 Classification: GENE REGULATION Ligands: X9O, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: X9O, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Dual Bet/Hdac Inhibitor Nb390
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2023-07-05 Classification: GENE REGULATION Ligands: X9K, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: X9K, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Dual Bet/Hdac Inhibitor Nb437
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.19 Å Release Date: 2023-07-05 Classification: GENE REGULATION Ligands: X9C, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: X9C, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Dual Bet/Hdac Inhibitor Nb462
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.23 Å Release Date: 2023-07-05 Classification: GENE REGULATION Ligands: X8T, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: X8T, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Dual Bet/Hdac Inhibitor Nb500
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2023-07-05 Classification: GENE REGULATION Ligands: X8O, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: X8O, EDO
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Dual Bet/Hdac Inhibitor Nb503
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2023-07-05 Classification: GENE REGULATION Ligands: EDO, X9U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: EDO, X9U
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Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With The Dual Bet/Hdac Inhibitor Nb512
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.29 Å Release Date: 2023-07-05 Classification: GENE REGULATION Ligands: XA3, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-07-05
Ligands: XA3, EDO
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Crystal Structure Of Pvhl:Elonginc:Elonginb Complex Bound To Protac Jw48
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2022-12-28 Classification: LIGASE Ligands: SYF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-28
Ligands: SYF
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Structure Of Human Wdr5 And Pvhl:Elonginc:Elonginb Bound To Protac With C3 Linker
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2022-11-09 Classification: LIGASE Ligands: Q3R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: Q3R
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Structure Of Human Wdr5 And Pvhl:Elonginc:Elonginb Bound To Protac With Aryl Linker
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2022-11-09 Classification: LIGASE Ligands: SCN, Q43, EDO, K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-11-09
Ligands: SCN, Q43, EDO, K
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Structure Of Human Mps1 (Ttk) Covalently Bound To Rms-07 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2022-02-16 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: YB4, GOL, TOE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-16
Ligands: YB4, GOL, TOE
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Apo Structure Of Bir2 Domain Of Birc2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2022-02-09 Classification: LIGASE Ligands: ZN, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-09
Ligands: ZN, EDO
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Quaternary Complex Of Human Wdr5 And Pvhl:Elonginc:Elonginb Bound To Protac Homer
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2021-11-24 Classification: STRUCTURAL PROTEIN Ligands: 8KH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-11-24
Ligands: 8KH
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Clk1 Bound With Caf052
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2020-11-11 Classification: TRANSFERASE Ligands: RH8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-11
Ligands: RH8
