Search Count: 21
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Structure Of The Diels Alderase Tedj, In Complex With Cofactor Fad
Organism: Streptomyces
Method: X-RAY DIFFRACTION Resolution:1.59 Å Release Date: 2024-11-13 Classification: OXIDOREDUCTASE Ligands: FAD |
Organism: Streptomyces
Method: X-RAY DIFFRACTION
Release Date: 2024-11-13
Ligands: FAD
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Structure Of The Diels Alderase Enzyme Abyu, From Micromonospora Maris, Co-Crystallised With A Non Transformable Substrate Analogue
Organism: Micromonospora maris ab-18-032
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2022-11-16 Classification: LIGASE Ligands: 8IF, EPE |
Organism: Micromonospora maris ab-18-032
Method: X-RAY DIFFRACTION
Release Date: 2022-11-16
Ligands: 8IF, EPE
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Estrogen Receptor Mutant L536S
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2019-11-27 Classification: TRANSCRIPTION Ligands: L5B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: L5B
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Crystal Structure Of C-Met Mutant Y1230H In Complex With Compound 14
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2016-11-23 Classification: TRANSFERASE Ligands: CL, 62E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-23
Ligands: CL, 62E
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Crystal Structure Of Cmet Wt With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2016-11-23 Classification: TRANSFERASE Ligands: 63B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-23
Ligands: 63B
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Crystal Structure Of Cmet In Complex With Cmpd.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2016-11-23 Classification: TRANSFERASE Ligands: 63K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-23
Ligands: 63K
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Crystal Structure Of C-Met L1195V In Complex With Sar125844
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2016-11-23 Classification: TRANSFERASE Ligands: 63K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-23
Ligands: 63K
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Crystal Structure Of C-Met-M1250T In Complex With Sar125844.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-11-23 Classification: TRANSFERASE Ligands: 63K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-23
Ligands: 63K
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Water Network Determines Selectivity For A Series Of Pyrimidone Indoline Amide Pi3Kbeta Inhibitors Over Pi3K-Delta
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2015-09-30 Classification: TRANSFERASE Ligands: J82 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2015-09-30
Ligands: J82
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Discovery Of (2S)-8-((3R)-3-Methylmorpholin-4-Yl)-1-(3-Methyl-2-Oxo- Butyl)-2-(Trifluoromethyl)-3,4-Dihydro-2H-Pyrimido(1,2-A)Pyrimidin-6- One: A Novel Potent And Selective Inhibitor Of Vps34 For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.99 Å Release Date: 2014-11-26 Classification: TRANSFERASE Ligands: EUT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-26
Ligands: EUT
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Discovery Of (2S)-8-((3R)-3-Methylmorpholin-4-Yl)-1-(3-Methyl-2-Oxo- Butyl)-2-(Trifluoromethyl)-3,4-Dihydro-2H-Pyrimido(1,2-A)Pyrimidin-6- One: A Novel Potent And Selective Inhibitor Of Vps34 For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2014-11-26 Classification: TRANSFERASE Ligands: SO4, RBQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-26
Ligands: SO4, RBQ
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Discovery Of (2S)-8-((3R)-3-Methylmorpholin-4-Yl)-1-(3-Methyl-2-Oxo- Butyl)-2-(Trifluoromethyl)-3,4-Dihydro-2H-Pyrimido(1,2-A)Pyrimidin-6- One: A Novel Potent And Selective Inhibitor Of Vps34 For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2014-11-26 Classification: TRANSFERASE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-26
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Discovery Of (2S)-8-((3R)-3-Methylmorpholin-4-Yl)-1-(3-Methyl-2-Oxo- Butyl)-2-(Trifluoromethyl)-3,4-Dihydro-2H-Pyrimido(1,2-A)Pyrimidin-6- One: A Novel Potent And Selective Inhibitor Of Vps34 For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.83 Å Release Date: 2014-11-26 Classification: TRANSFERASE Ligands: SO4, GOL, UJB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-26
Ligands: SO4, GOL, UJB
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Discovery Of (2S)-8-((3R)-3-Methylmorpholin-4-Yl)-1-(3-Methyl-2-Oxo- Butyl)-2-(Trifluoromethyl)-3,4-Dihydro-2H-Pyrimido(1,2-A)Pyrimidin-6- One: A Novel Potent And Selective Inhibitor Of Vps34 For The Treatment Of Solid Tumors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-11-26 Classification: TRANSFERASE Ligands: SO4, 7A5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-26
Ligands: SO4, 7A5
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Sar156497 An Exquisitely Selective Inhibitor Of Aurora Kinases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2014-11-19 Classification: TRANSFERASE Ligands: Y3M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-19
Ligands: Y3M
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Sar156497 An Exquisitely Selective Inhibitor Of Aurora Kinases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.20 Å Release Date: 2014-11-19 Classification: TRANSFERASE Ligands: QMN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-19
Ligands: QMN
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Sar156497 An Exquisitely Selective Inhibitor Of Aurora Kinases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-11-19 Classification: TRANSFERASE Ligands: JVE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-11-19
Ligands: JVE
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Crystal Structure Of Vps34 In Complex With Sar405.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2014-10-22 Classification: LIPID KINASE Ligands: SO4, 1TT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-22
Ligands: SO4, 1TT
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Discovery And Optimization Of Pyrimidone Indoline Amide Pi3Kbeta Inhibitors For The Treatment Of Phosphatase And Tensin Homologue (Pten)-Deficient Cancers
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2014-01-15 Classification: TRANSFERASE Ligands: J82 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2014-01-15
Ligands: J82
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X-Ray Structure Of Pi3K-Gamma Bound To A 4-(Morpholin-4-Yl)- (6-Oxo-1,6-Dihydropyrimidin-2-Yl)Amide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.40 Å Release Date: 2012-11-14 Classification: Transferase/Transferase Inhibitor Ligands: 0W7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-11-14
Ligands: 0W7