Search Count: 37
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The Virulence-Associated Protein Hsva From The Fire Blight Pathogen Erwinia Amylovora Is A Polyamine Amidinotransferase
Organism: Erwinia amylovora
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2017-11-15 Classification: TRANSFERASE Ligands: EDO |
Organism: Erwinia amylovora
Method: X-RAY DIFFRACTION
Release Date: 2017-11-15
Ligands: EDO
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Egfr Kinase Domain Mutant "Tmlr" With Azabenzimidazole Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60B
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Egfr Kinase Domain Mutant "Tmlr" With 3-Carboxamide Azaindole Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60D
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Egfr Kinase Domain Mutant "Tmlr" With 3-Azetidinyl Azaindazole Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.62 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60E
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Braf Kinase Domain B3Ac Loop Deletion Mutant In Complex With Sorafenib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.51 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: BAX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: BAX
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Egfr Kinase Domain Mutant "Tmlr" With A Pyrazolopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 63M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: 63M
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Egfr Kinase Domain Mutant "Tmlr" With A Imidazopyridinyl-Aminopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 63N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: SO4, 63N
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Braf Kinase Domain B3Ac Loop Deletion Mutant In Complex With Az628
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: B1E, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: B1E, PEG
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Braf Kinase Domain B3Ac Loop Deletion Mutant In Complex With Dabrafenib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2016-04-06 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: P06 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: P06
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Egfr Kinase Domain Mutant "Tmlr" With Pyridone Compound 2: 4-[2-(4-Chlorophenyl)Ethylamino]-~{N}-[4-(4-Methylpiperazin-1-Yl)Phenyl]-2-Oxidanylidene-1~{H}-Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2015-12-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5Q2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-30
Ligands: 5Q2
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Egfr Kinase Domain Mutant "Tmlr" With Pyridone Compound 19: 4-[(2-Azanylpyrimidin-4-Yl)Amino]-~{N}-[4-(4-Methylpiperazin-1-Yl)Phenyl]-2-Oxidanylidene-1~{H}-Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.78 Å Release Date: 2015-12-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 5Q3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-30
Ligands: SO4, 5Q3
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Egfr Kinase Domain Mutant "Tmlr" With Pyridone Compound 13: 4-[(2-Methoxyphenyl)Amino]-~{N}-[4-(4-Methylpiperazin-1-Yl)Phenyl]-2-Oxidanylidene-1~{H}-Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.81 Å Release Date: 2015-12-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 5Q4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-30
Ligands: SO4, 5Q4
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Egfr Kinase Domain With Pyridone Compound 13: 4-[(2-Methoxyphenyl)Amino]-~{N}-[4-(4-Methylpiperazin-1-Yl)Phenyl]-2-Oxidanylidene-1~{H}-Pyridine-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-12-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5Q4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-30
Ligands: 5Q4
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Egfr Kinase (T790M/L858R) Apo
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2015-12-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-02
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Egfr Kinase (T790M/L858R) With Inhibitor Compound 15: ~{N}-(7-Chloranyl-1~{H}-Indazol-3-Yl)-7,7-Dimethyl-2-(1~{H}-Pyrazol-4-Yl)-5~{H}-Furo[3,4-D]Pyrimidin-4-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2015-12-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5N3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-02
Ligands: 5N3
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Egfr Kinase (T790M/L858R) With Inhibitor Compound 27: ~{N}-(1~{H}-Indazol-3-Yl)-7,7-Dimethyl-2-(2-Methylpyrazol-3-Yl)-5~{H}-Furo[3,4-D]Pyrimidin-4-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2015-12-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5N4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-02
Ligands: 5N4
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Egfr Kinase Domain Mutant "Tmlr" With Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: 4YV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 4YV
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Egfr Kinase Domain Mutant "Tmlr" With Compound 17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: 4YW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 4YW
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Egfr Kinase Domain Mutant "Tmlr" With Compound 23
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: SO4, 4YX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: SO4, 4YX
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Egfr Kinase Domain Mutant "Tmlr" With Compound 24
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2015-10-28 Classification: Transferase/transferase inhibitor Ligands: 4Z8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-10-28
Ligands: 4Z8
