Search Count: 51
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Crystal Structure Of A Cgrp Receptor Ectodomain Heterodimer Bound To Macrocyclic Inhibitor Htl0029881
Organism: Escherichia coli k-12, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2022-12-07 Classification: MEMBRANE PROTEIN Ligands: OKU, PG4 |
Organism: Escherichia coli k-12, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-07
Ligands: OKU, PG4
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Crystal Structure Of A Cgrp Receptor Ectodomain Heterodimer Bound To Macrocyclic Inhibitor Htl0029882
Organism: Escherichia coli k-12, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2022-12-07 Classification: MEMBRANE PROTEIN Ligands: OP9, PG4 |
Organism: Escherichia coli k-12, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-07
Ligands: OP9, PG4
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Crystal Structure Of A Cgrp Receptor Ectodomain Heterodimer Bound To Macrocyclic Inhibitor Htl0031448
Organism: Escherichia coli k-12, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2022-12-07 Classification: MEMBRANE PROTEIN Ligands: PG4, OL0, ACT |
Organism: Escherichia coli k-12, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-12-07
Ligands: PG4, OL0, ACT
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Crystal Structure Of A Cgrp Receptor Ectodomain Heterodimer Bound To Macrocyclic Inhibitor Htl0028125
Organism: Escherichia coli (strain k12), Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2022-06-15 Classification: MEMBRANE PROTEIN Ligands: 7IR, PG4 |
Organism: Escherichia coli (strain k12), Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-15
Ligands: 7IR, PG4
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Crystal Structure Of A Cgrp Receptor Ectodomain Heterodimer Bound To Macrocyclic Inhibitor Compound 13
Organism: Escherichia coli (strain k12), Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2022-06-15 Classification: MEMBRANE PROTEIN Ligands: PG4, 7IU |
Organism: Escherichia coli (strain k12), Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-06-15
Ligands: PG4, 7IU
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Crystal Structure Of Prostaglandin D2 Synthase In Complex With Fragment 1A At 1.84A Resolution.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2021-07-28 Classification: ISOMERASE Ligands: GSH, MG, QPN, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-28
Ligands: GSH, MG, QPN, GOL
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H-Pdgs Complexed With A 2-Phenylimidazo[1,2-A]Pyridine-6-Carboxamide Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2021-05-26 Classification: Isomerase, Transferase/Inhibitor Ligands: GSH, VH4, MG, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-26
Ligands: GSH, VH4, MG, NA
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H-Pdgs Complexed With A 2-Phenylimidazo[1,2-A]Pyridine-6-Carboxamide Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.13 Å Release Date: 2021-05-26 Classification: Isomerase, Transferase/Inhibitor Ligands: CL, EDO, GSH, VH7, MG, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-26
Ligands: CL, EDO, GSH, VH7, MG, NA
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Hpgds Complexed With An Aza-Quinoline
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2020-11-04 Classification: HYDROLASE Ligands: GSH, SWS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-04
Ligands: GSH, SWS
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H-Pgds Complexed With Inhibitor 1Y
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2020-11-04 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GSH, EDO, TJG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-11-04
Ligands: GSH, EDO, TJG
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Small Molecule Inhibitor Of The Keap1-Nrf2 Protein-Protein Interaction
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2019-04-24 Classification: PROTEIN BINDING Ligands: J6H |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: J6H
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Small Molecule Inhibitor Of The Keap1-Nrf2 Protein-Protein Interaction
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2019-04-24 Classification: PROTEIN BINDING Ligands: DMS, J6N |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: DMS, J6N
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Small Molecule Inhibitor Of The Keap1-Nrf2 Protein-Protein Interaction
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2019-04-24 Classification: PROTEIN BINDING Ligands: SO4, J6Q |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: SO4, J6Q
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Small Molecule Inhibitor Of The Keap1-Nrf2 Protein-Protein Interaction
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2019-04-24 Classification: PROTEIN BINDING Ligands: SO4, CL, J6K |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: SO4, CL, J6K
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Small Molecule Inhibitor Of The Keap1-Nrf2 Protein-Protein Interaction
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.72 Å Release Date: 2019-04-24 Classification: PROTEIN BINDING Ligands: CL, J8H |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-04-24
Ligands: CL, J8H
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Hpgds Complexed With A Quinoline-3-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-03-27 Classification: HYDROLASE Ligands: GSH, KCD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-27
Ligands: GSH, KCD
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Rat Hpgds Complexed With A Quinoline
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-03-27 Classification: HYDROLASE Ligands: GSH, KDV |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2019-03-27
Ligands: GSH, KDV
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Fragment Derived Xiap Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.63 Å Release Date: 2018-08-22 Classification: APOPTOSIS Ligands: ZN, FUK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-22
Ligands: ZN, FUK
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Fragment Derived Xiap Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2018-08-22 Classification: APOPTOSIS Ligands: ZN, NA, FUE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-08-22
Ligands: ZN, NA, FUE
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Structure Of The Keap1 Kelch Domain In Complex With A Small Molecule Inhibitor.
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.91 Å Release Date: 2016-04-13 Classification: TRANSCRIPTION Ligands: S0W |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2016-04-13
Ligands: S0W
