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Search Count: 29

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8S16 image
C-Kit Kinase Domain In Complex With Imatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: STI, CL

7N9G image
Crystal Structure Of The Abl 1B Kinase Domain In Complex With Dasatinib And Imatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2022-04-27
Classification: CELL CYCLE
Ligands: STI, 1N1, PO4


6JOL image
Crystal Structure Of Pdgfra In Complex With Imatinib By Co-Crystallization
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.90 Å Release Date: 2020-03-25
Classification: ONCOPROTEIN
Ligands: STI

6KTN image
Human Ppargamma Ligand-Binding Domain R288A Mutant In Complex With Imatinib

6NPE image
C-Abl Kinase Domain With The Activator(Cmpd6), 2-Cyano-N-(4-(3,4-Dichlorophenyl)Thiazol-2-Yl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.15 Å Release Date: 2019-03-13
Classification: TRANSFERASE
Ligands: SO4, STI, KWD, 2PE

6NPU image
C-Abl Kinase Domain With The Activator(Cmpd29), N-(1-(3,4-Dichlorophenyl)-4,5-Dihydro-1H-Pyrazol-3-Yl)Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.33 Å Release Date: 2019-03-13
Classification: TRANSFERASE
Ligands: STI, KWV, SO4, GOL, 2PE

6NPV image
C-Abl Kinase Domain With The Activator(Cmpd51), N-(1-(3,4-Dichlorophenyl)-4-(2-Hydroxyethyl)-4,5-Dihydro-1H-Pyrazol-3-Yl)Isonicotinamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.86 Å Release Date: 2019-03-13
Classification: TRANSFERASE
Ligands: SO4, STI, KWP, GOL, 2PE

6HD4 image
Abl1 In Complex With Compound 7 And Imatinib (Sti-571)
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Resolution:2.03 Å Release Date: 2018-10-24
Classification: TRANSFERASE
Ligands: GOL, CL, FYW, STI

6HD6 image
Abl1 In Complex With Compound6 And Imatinib (Sti-571)
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2018-09-12
Classification: TRANSFERASE
Ligands: CL, FYH, STI

5MQT image
Crystal Structure Of Dck Mutant C3S In Complex With Imatinib And Udp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.20 Å Release Date: 2017-11-22
Classification: TRANSFERASE
Ligands: UDP, STI, MG, DCM

4R7I image
Crystal Structure Of Fms Kinase Domain With A Small Molecular Inhibitor, Gleevec

4CSV image
Tyrosine Kinase As - A Common Ancestor Of Src And Abl Bound To Gleevec

4BKJ image
Crystal Structure Of The Human Ddr1 Kinase Domain In Complex With Imatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.70 Å Release Date: 2013-05-22
Classification: TRANSFERASE
Ligands: STI, EDO

3OEZ image
Crystal Structure Of The L317I Mutant Of The Chicken C-Src Tyrosine Kinase Domain Complexed With Imatinib

3PYY image
Discovery And Characterization Of A Cell-Permeable, Small-Molecule C-Abl Kinase Activator That Binds To The Myristoyl Binding Site
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2011-03-09
Classification: TRANSFERASE
Ligands: SO4, STI, 3YY, 2PE, GOL

3MS9 image
Abl Kinase In Complex With Imatinib And A Fragment (Frag1) In The Myristate Pocket

3MSS image
Abl Kinase In Complex With Imatinib And Fragment (Frag2) In The Myristate Site

3K5V image
Structure Of Abl Kinase In Complex With Imatinib And Gnf-2
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Resolution:1.74 Å Release Date: 2010-01-19
Classification: TRANSFERASE
Ligands: STJ, STI, CL

3HEC image
P38 In Complex With Imatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.50 Å Release Date: 2009-11-10
Classification: TRANSFERASE
Ligands: STI, BOG
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