Search Count: 24
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Human Pif + Z48847594 (Occupancy 0.7)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2024-10-02 Classification: DNA BINDING PROTEIN Ligands: ANP, MG, O0J, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: ANP, MG, O0J, NA
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Xchem Refined Pif1-X0076 Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2024-09-18 Classification: DNA BINDING PROTEIN Ligands: ANP, MG, O0J, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-18
Ligands: ANP, MG, O0J, DMS
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Crystal Structure Of Human Clk1 In Complex With Leucettinib-92
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2023-05-17 Classification: TRANSFERASE Ligands: WAK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-17
Ligands: WAK
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Crystal Structure Of Human Casein Kinase Ii Subunit Alpha (Ck2A1) In Complex With Leucettinib-92
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2023-05-17 Classification: TRANSFERASE Ligands: SO4, WAK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-17
Ligands: SO4, WAK
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Crystal Structure Of Human Clk1 In Complex With Leucettinib-21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2023-05-17 Classification: TRANSFERASE Ligands: WAZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-17
Ligands: WAZ
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Human Cyclophilin D In Complex With 1-((1S,9S,10S)-10-Hydroxy-12-Oxa-8-Aza-Tricyclo[7.3.1.02,7]Trideca-2,4,6-Trien-4-Ylmethyl)-3- {2-[(R)-2-(2-Methylsulfanyl-Phenyl)-Pyrrolidin-1-Yl]-2-Oxo-Ethyl}-Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.64 Å Release Date: 2019-11-27 Classification: ISOMERASE Ligands: JUZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: JUZ
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Human Cyclophilin D In Complex With 1-(((2R,3S,6R)-3-Hydroxy-2,3,4,6-Tetrahydro-1H-2,6-Methanobenzo[C][1,5]Oxazocin-8-Yl)Methyl)-3-(2-((R)-2-(2-(Methylthio)Phenyl)Pyrrolidin-1-Yl)-2-Oxoethyl)Urea
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.36 Å Release Date: 2019-11-27 Classification: ISOMERASE Ligands: PG4, SO4, PO4, JV2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: PG4, SO4, PO4, JV2
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Human Cyclophilin D In Complex With 2-(Exo-3,5-Dioxo-4-Aza-Tricyclo[5.2.1.02,6]Dec-4-Yl)-N-((1R,9R,10S)-10-Hydroxy-12-Oxa-8-Aza-Tricyclo[7.3.1.02,7]Trideca-2(7),3,5-Trien-4-Ylmethyl)-Acetamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2019-11-27 Classification: ISOMERASE Ligands: O4B, P6G, JVH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: O4B, P6G, JVH
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Human Cyclophilin D In Complex With Bicyclic Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-11-27 Classification: ISOMERASE Ligands: JVN, 1PE, PG4, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: JVN, 1PE, PG4, SO4
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Human Cyclophilin D In Complex With Fragment
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.26 Å Release Date: 2019-11-27 Classification: ISOMERASE Ligands: JVQ, SO4, PGE, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: JVQ, SO4, PGE, PG4
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Human Cyclophilin D In Complex With N-Cyclopentyl-N'-Pyridin-2-Ylmethyl-Oxalamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2019-11-27 Classification: ISOMERASE Ligands: JW2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: JW2
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Human Cyclophilin D In Complex With Norbornane Fragment Derivative
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-11-27 Classification: ISOMERASE Ligands: JWB, JVQ, PEG, PG4, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-27
Ligands: JWB, JVQ, PEG, PG4, SO4
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Crystal Structure Of Human Caspase-1 With N-{3-[1-((S)-2-Hydroxy-5-Oxo-Tetrahydro-Furan-3-Ylcarbamoyl)-Ethyl]-1-Methyl-2,4-Dioxo-1,2,3,4-Tetrahydro-Pyrimidin-5-Yl}-4-(Quinoxalin-2-Ylamino)-Benzamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2018-05-02 Classification: HYDROLASE Ligands: CVE, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: CVE, SO4
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Crystal Structure Of Human Caspase-1 With (3S,6S,10As)-N-((2S,3S)-2-Hydroxy-5-Oxotetrahydrofuran-3-Yl)-6-(Isoquinoline-1-Carboxamido)-5-Oxodecahydropyrrolo[1,2-A]Azocine-3-Carboxamide (Pge-3935199)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2018-02-28 Classification: HYDROLASE Ligands: N7N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-28
Ligands: N7N
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Crystal Structure Of Human Caspase-1 With 2-((2-Naphthoyl)-L-Valyl)-4-Hydroxy-N-((3S)-2-Hydroxy-5-Oxotetrahydrofuran-3-Yl)-2-Azabicyclo[2.2.2]Octane-3-Carboxamide (Compound 1)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2017-12-20 Classification: HYDROLASE Ligands: WE0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: WE0
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Structure-Based Design Of 7-Azaindole-Pyrrolidines As Inhibitors Of 11Beta-Hydroxysteroid-Dehydrogenase Type I
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2010-11-17 Classification: OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR Ligands: NDP, 2M3, SO4 |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2010-11-17
Ligands: NDP, 2M3, SO4
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Structure Of The Dnag Catalytic Core
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2000-04-07 Classification: TRANSFERASE Ligands: SR |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2000-04-07
Ligands: SR
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Structure Of The Dnag Catalytic Core
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2000-04-07 Classification: TRANSFERASE Ligands: Y1 |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2000-04-07
Ligands: Y1
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Peptide Deformylase As Zn2+ Containing Form (Native) In Complex With Inhibitor Polyethylene Glycol
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 1999-08-27 Classification: HYDROLASE Ligands: ZN, 2PE, SO4 |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 1999-08-27
Ligands: ZN, 2PE, SO4
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Peptide Deformylase As Zn2+ Containing Form
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 1999-08-27 Classification: HYDROLASE Ligands: ZN, SO4 |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 1999-08-27
Ligands: ZN, SO4
