Search Count: 35
![]() |
Crystal Structure Of Human Kras G12C Covalently Bound To Thiazol-2-Yl Piperidine Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2026-08-12 Classification: SIGNALING PROTEIN Ligands: MG, GDP, A1DI3, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-12
Ligands: MG, GDP, A1DI3, EDO
![]() |
Crystal Structure Of Human Kras G12C Covalently Bound To 4-Methyl-Thiazol-5-Yl Piperidine Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.10 Å Release Date: 2026-08-12 Classification: SIGNALING PROTEIN Ligands: MG, GDP, A1DI5, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-12
Ligands: MG, GDP, A1DI5, EDO
![]() |
Crystal Structure Of Human Kras G12C Covalently Bound To 1,4-Dimethyl-Pyrazol-5-Yl Piperidine Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.26 Å Release Date: 2026-08-12 Classification: SIGNALING PROTEIN Ligands: MG, GDP, A1DI6, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-12
Ligands: MG, GDP, A1DI6, EDO
![]() |
Crystal Structure Of Human Kras G12C Covalently Bound To Am-8719
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2026-08-12 Classification: SIGNALING PROTEIN Ligands: MG, GDP, A1DI7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-12
Ligands: MG, GDP, A1DI7
![]() |
Crystal Structure Of Human Kras G12D In Complex With Gdp And Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2026-07-22 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: MG, GDP, A1CZE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-22
Ligands: MG, GDP, A1CZE
![]() |
Crystal Structure Of Human Kras G12D In Complex With Gdp And Am-2383
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.25 Å Release Date: 2026-07-22 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: MG, GDP, A1AG3, EDO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-22
Ligands: MG, GDP, A1AG3, EDO, SO4
![]() |
Crystal Structure Of Human Kras G12D In Complex With Gmppcp And Am-2383
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.12 Å Release Date: 2026-07-22 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: MG, GCP, A1AG3, EDO, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-22
Ligands: MG, GCP, A1AG3, EDO, SO4
![]() |
Crystal Structure Of Human Kras G12V In Complex With Gdp And Am-2383
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2026-07-22 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: MG, GDP, A1AG3, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-22
Ligands: MG, GDP, A1AG3, EDO
![]() |
Crystal Structure Of Human Kras G12V In Complex With Gmppcp And Am-2383
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2026-07-22 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: MG, GCP, A1AG3, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-22
Ligands: MG, GCP, A1AG3, EDO
![]() |
Crystal Structure Of Human Kras G12C Covalently Bound To Del Triazine Compound 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2025-02-26 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: CA, GDP, A1BH6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-26
Ligands: CA, GDP, A1BH6
![]() |
Crystal Structure Of Human Kras G12C Covalently Bound To Nopinone-Derived Naphthol Compound 21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.18 Å Release Date: 2025-02-26 Classification: SIGNALING PROTEIN,ONCOPROTEIN/INHIBITOR Ligands: MG, GDP, A1BH5, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-26
Ligands: MG, GDP, A1BH5, EDO
![]() |
Crystal Structure Of Human Kras G12C Covalently Bound To A Phthalazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: MG, GDP, OJ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: MG, GDP, OJ1
![]() |
Crystal Structure Of Human Kras G12C Covalently Bound To A Quinazolinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2019-12-25 Classification: SIGNALING PROTEIN/Inhibitor Ligands: GDP, CA, OHY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-12-25
Ligands: GDP, CA, OHY
![]() |
Crystal Structure Of Human Kras G12C Covalently Bound To Amg 510
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2019-11-06 Classification: SIGNALING PROTEIN Ligands: MG, GDP, MOV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-11-06
Ligands: MG, GDP, MOV
![]() |
Crystal Structure Of Human Pim-1 Kinase In Complex With A Quinazolinone-Pyrrolodihydropyrrolone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-01-16 Classification: TRANSFERASE Ligands: JYG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-16
Ligands: JYG, GOL
![]() |
Crystal Structure Of Human Pim-1 Kinase In Complex With A Quinazolinone-Pyrrolopyrrolone Inhibitor.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-06-22 Classification: transferase/transferase inhibitor Ligands: 6CD, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-22
Ligands: 6CD, GOL
![]() |
Crystal Structure Of Human Pim-1 Kinase In Complex With A Macrocyclic Quinoxaline-Pyrrolodihydropiperidinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-05-04 Classification: transferase/transferase inhibitor Ligands: 5QO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 5QO, GOL
![]() |
Crystal Structure Of C-Met In Complex With Naphthyridinone Inhibitor 5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2016-02-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5SZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: 5SZ
![]() |
Crystal Structure Of C-Met In Complex With Amg 337
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2016-02-10 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 5T1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-10
Ligands: 5T1
![]() |
Crystal Structure Of C-Met In Complex With (R)-5-(8-Fluoro-3-(1-Fluoro-1-(3-Methoxyquinolin-6-Yl)Ethyl)-[1,2,4]Triazolo[4,3-A]Pyridin-6-Yl)-3-Methylisoxazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2015-03-11 Classification: Transferase/transferase inhibitor Ligands: 46G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-03-11
Ligands: 46G
