Search Count: 54
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Trim21 Pryspry Domain Bound To An Enhanced Prlx-93936 Analog
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2025-08-27 Classification: IMMUNE SYSTEM Ligands: A1BLD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-08-27
Ligands: A1BLD
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Tricomplex Of Compound 1, Kras G12D, And Cypa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2025-07-23 Classification: HYDROLASE Ligands: GNP, MG, CL, A1AZV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-23
Ligands: GNP, MG, CL, A1AZV
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Tricomplex Of Compound 2, Kras G12D, And Cypa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.28 Å Release Date: 2025-07-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GNP, MG, A1AZX, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-23
Ligands: GNP, MG, A1AZX, CL
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Tricomplex Of Compound 3, Kras G12D, And Cypa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.35 Å Release Date: 2025-07-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GNP, MG, CL, A1AZY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-23
Ligands: GNP, MG, CL, A1AZY
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Tricomplex Of Rmc-9945, Kras G12D, And Cypa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.29 Å Release Date: 2025-07-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GNP, MG, A1AZW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-23
Ligands: GNP, MG, A1AZW
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Tri-Complex Of Zoldonrasib (Rmc-9805), Kras G12D, And Cypa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.29 Å Release Date: 2025-07-23 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: GNP, MG, CL, A1AZZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-23
Ligands: GNP, MG, CL, A1AZZ
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Tricomplex Of Rmc-9945, Kras G12N, And Cypa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.08 Å Release Date: 2025-07-23 Classification: SIGNALING PROTEIN Ligands: GNP, MG, CL, A1BEA, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-23
Ligands: GNP, MG, CL, A1BEA, GOL
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Amg 193, A Clinical Stage Mta-Cooperative Prmt5 Inhibitor, Drives Anti-Tumor Activity Preclinically And In Patients With Mtap-Deleted Cancers
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2024-10-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GOL, DMS, A1ATH, MTA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-02
Ligands: GOL, DMS, A1ATH, MTA
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Bromodomain Of Cbp Liganded With Inhibitor Icbp5
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2024-02-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: EDO, YVK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-28
Ligands: EDO, YVK
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Bromodomain Of Cbp Liganded With Inhibitor Icbp2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2024-02-21 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: YRI, NI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-21
Ligands: YRI, NI
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Structure Of Bovine Pka Bound To (R)-N-(4-(1H-Pyrrolo[2,3-B]Pyridin-4-Yl)Phenyl)-2-Amino-4-Methylpentanamide
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2024-02-21 Classification: CYTOSOLIC PROTEIN Ligands: ZWG |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2024-02-21
Ligands: ZWG
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Bromodomain Of Cbp Liganded With Ccs-1477
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2024-02-07 Classification: TRANSCRIPTION/INHIBITOR Ligands: PO4, JHL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: PO4, JHL, EDO
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Bromodomain Of Ep300 Liganded With Ccs-1477
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2024-02-07 Classification: TRANSCRIPTION/INHIBITOR Ligands: JHL, EDO, NI, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: JHL, EDO, NI, SO4
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First Bromodomain Of Brd4 Liganded With Ccs-1477
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.53 Å Release Date: 2024-02-07 Classification: TRANSCRIPTION/INHIBITOR Ligands: JHL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: JHL, EDO
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Bromodomain Of Cbp Liganded With Icbp4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2024-02-07 Classification: TRANSCRIPTION/INHIBITOR Ligands: EDO, YJY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: EDO, YJY
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Bromodomain Of Cbp Liganded With Icbp6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2024-02-07 Classification: TRANSCRIPTION/INHIBITOR Ligands: YID, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: YID, EDO
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Bromodomain Of Cbp Liganded With Icbp8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2024-02-07 Classification: TRANSCRIPTION/INHIBITOR Ligands: YN5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: YN5
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Tricomplex Of Rmc-7977, Kras Wt, And Cypa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2024-02-07 Classification: HYDROLASE/INHIBITOR Ligands: GNP, MG, EDO, ZNI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: GNP, MG, EDO, ZNI
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Tricomplex Of Rmc-7977, Hras Wt, And Cypa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2024-02-07 Classification: HYDROLASE/INHIBITOR Ligands: GNP, MG, GOL, ZNI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: GNP, MG, GOL, ZNI
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Tricomplex Of Rmc-7977, Kras G12R, And Cypa
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2024-02-07 Classification: HYDROLASE/INHIBITOR Ligands: GNP, MG, ZNI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-02-07
Ligands: GNP, MG, ZNI
