Search Count: 51
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Crystal Structure Of The Smarca2 Bromodomain Bound To A Fragment Screening Hit
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.07 Å Release Date: 2025-06-18 Classification: GENE REGULATION Ligands: A1I5P, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-18
Ligands: A1I5P, ZN
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Crystal Structure Of The Smarca2 Bromodomain Bound To A Tricyclic Pyrimidoindolone Inhibitor (Compound 17)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2025-05-14 Classification: GENE REGULATION Ligands: A1I45, ZN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-05-14
Ligands: A1I45, ZN
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Induced Myeloid Leukemia Cell Differentiation Protein Fabcomplex In Complex With Compound 1
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2023-05-24 Classification: APOPTOSIS Ligands: VF8 |
Organism: Homo sapiens, Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2023-05-24
Ligands: VF8
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Eed In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2021-12-08 Classification: PROTEIN BINDING Ligands: L9W, 51A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-08
Ligands: L9W, 51A
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Eed In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2021-12-08 Classification: PROTEIN BINDING Ligands: L9W, 52R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-08
Ligands: L9W, 52R
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Eed In Complex With Compound 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2021-12-08 Classification: PROTEIN BINDING Ligands: MG, L9W, 54N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-12-08
Ligands: MG, L9W, 54N
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Mertk Kinase Domain With Type 1.5 Inhibitor Containing A Di-Methyl Pyrazole Group
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VJZ, CL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VJZ, CL, DMS
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Mertk Kinase Domain With Type 1.5 Inhibitor Containing A Di-Methyl, Cyano Pyrazole Group
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VK2, CL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VK2, CL, DMS
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Mertk Kinase Domain With Type 1.5 Inhibitor Containing A Tri-Methyl Pyrazole Group
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2021-09-15 Classification: TRANSFERASE Ligands: VK5, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-15
Ligands: VK5, CL
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Eed In Complex With A Cyano-Benzofuran
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2021-05-12 Classification: PROTEIN BINDING Ligands: CA, L9W, PV5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: CA, L9W, PV5
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Eed In Complex With A Triazolopyrimidine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2021-05-12 Classification: PROTEIN BINDING Ligands: L9W, GOL, EJR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-12
Ligands: L9W, GOL, EJR
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Mertk Kinase Domain In Complex With Nps-1034
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.44 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4K
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Mertk Kinase Domain In Complex With Quinazoline-Based Inhbitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4E, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4E, SO4
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Mertk Kinase Domain In Complex With A Bisaminopyrimidine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4N
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Mertk Kinase Domain In Complex With Purine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4Q
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Mertk Kinase Domain In Complex With A Type 2 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4T
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Mertk Kinase Domain With Type 1.5 Inhibitor From A Dna-Encoded Library
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4W
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Mertk Kinase Domain With Type 1 Inhibitor From A Dna-Encoded Library
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S4Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S4Z
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Mertk Kinase Domain With Type 3 Inhibitor From A Dna-Encoded Library
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2021-03-03 Classification: SIGNALING PROTEIN Ligands: S5E, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-03
Ligands: S5E, CL, EDO
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Crystal Structure Of The Catalytic Domain Of Human Parp1 (Apo)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2021-01-13 Classification: TRANSFERASE Ligands: SO4, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-13
Ligands: SO4, DMS, EDO