Search Count: 50
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Crystal Structure Of The Lsd1/Corest Histone Demethylase In Complex With The Cofactor Fad And The Inhibitor Gsk690
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.66 Å Release Date: 2025-09-17 Classification: GENE REGULATION Ligands: FAD, GOL, A1A5U |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-17
Ligands: FAD, GOL, A1A5U
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Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7G
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Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.42 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7H
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Crystal Structure Of Rar-Related Orphan Receptor C (Nhis-Rorgt(244-487)-L6-Src1(678-692)) In Complex With {3,5-Dichloro-4-[4-Methoxy-3-(Propan-2-Yl)Phenoxy]Phenyl}Methanol
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.14 Å Release Date: 2021-01-20 Classification: TRANSFERASE/Agonist Ligands: Z7I |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-01-20
Ligands: Z7I
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Cryo-Em Structure Of Irp2-Fbxl5-Skp1 Complex
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Release Date: 2020-08-05 Classification: LIGASE Ligands: FES |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2020-08-05
Ligands: FES
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Substituted Benzyloxytricyclic Compounds As Retinoic Acid-Related Orphan Receptor Gamma T Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2020-06-17 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: Z7F |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-06-17
Ligands: Z7F
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Substituted Benzyloxytricyclic Compounds As Retinoic Acid-Related Orphan Receptor Gamma T Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2020-04-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: TKJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: TKJ
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Substituted Benzyloxytricyclic Compounds As Retinoic Acid-Related Orphan Receptor Gamma T Agonists
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2020-04-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: Z7D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-29
Ligands: Z7D
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Human Dyrk1A In Complex With Ldn-211898
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2015-02-25 Classification: TRANSFERASE Ligands: AWR, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-02-25
Ligands: AWR, PO4
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Glycogen Synthase Kinase 3 Beta Complexed With Axin Peptide And Leucettine L4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.77 Å Release Date: 2013-01-30 Classification: TRANSFERASE/PEPTIDE Ligands: CWT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-01-30
Ligands: CWT
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Human Proto-Oncogene Serine Threonine Kinase (Pim1) In Complex With A Consensus Peptide And Leucettine L41
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-10-03 Classification: TRANSFERASE Ligands: 3RA, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-03
Ligands: 3RA, EDO
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Human Dyrk1A In Complex With Leucettine L41
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.15 Å Release Date: 2012-09-05 Classification: TRANSFERASE Ligands: 3RA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-09-05
Ligands: 3RA
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Human Dyrk2 In Complex With Leucettine L41
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2012-09-05 Classification: TRANSFERASE Ligands: 3RA, EDO, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-09-05
Ligands: 3RA, EDO, PO4
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Crystal Structure Of Dual-Specificity Tyrosine Phosphorylation Regulated Kinase 2 (Dyrk2) In Complex With An Indirubin Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2010-01-05 Classification: TRANSFERASE Ligands: IRB, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-01-05
Ligands: IRB, CL
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Crystal Structure Of Dual-Specificity Tyrosine Phosphorylation Regulated Kinase 2 (Dyrk2)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2009-10-13 Classification: TRANSFERASE Ligands: SO4, NA, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-13
Ligands: SO4, NA, CL
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Human Dual-Specificity Tyrosine-Phosphorylation-Regulated Kinase 1A In Complex With A Consensus Substrate Peptide
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2009-08-18 Classification: TRANSFERASE/PEPTIDE Ligands: D15, CL |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2009-08-18
Ligands: D15, CL
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Crystal Structure Of Human Dual Specificity Protein Kinase (Ttk) In Complex With A Pyrimido-Diazepin Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2009-05-19 Classification: TRANSFERASE Ligands: MG, 92M |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-05-19
Ligands: MG, 92M
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Crystal Structure Of Human Mitogen Activated Protein Kinase 11 (P38 Beta) In Complex With Nilotinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2009-04-07 Classification: Transferase/Transferase Inhibitor Ligands: NIL, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-04-07
Ligands: NIL, EDO, CL
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Crystal Structure Of Human Dual Specificity Protein Kinase (Ttk) In Complex With A Pyrolo-Pyridin Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2009-03-17 Classification: TRANSFERASE Ligands: S22, 7PE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-03-17
Ligands: S22, 7PE
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Crystal Structure Of Human Mitogen-Activated Protein Kinase Kinase 6 (Mek6) Activated Mutant (S207D, T211D)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.26 Å Release Date: 2009-01-06 Classification: TRANSFERASE Ligands: STU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-01-06
Ligands: STU
