Search Count: 14
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Akt1 Mutant In Complex With Miransertib (Arq 092)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2026-07-01 Classification: TRANSFERASE Ligands: 6S1, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-01
Ligands: 6S1, EDO, GOL
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Structure Of Mature Activin A From Dmso Solvent Optimisation Of Xchem Fragment Screen
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2025-02-12 Classification: SIGNALING PROTEIN Ligands: DMS, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: DMS, SO4
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Co-Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-09-08 Classification: TRANSFERASE Ligands: UCE, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: UCE, ACT
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Co-Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 6
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2021-09-08 Classification: TRANSFERASE Ligands: ACT, UC8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-09-08
Ligands: ACT, UC8
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Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 16A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-10-16 Classification: TRANSFERASE Ligands: L1Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-16
Ligands: L1Z
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Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 15C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2019-10-16 Classification: TRANSFERASE Ligands: L1W |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-10-16
Ligands: L1W
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Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor Borussertib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2019-03-20 Classification: TRANSFERASE Ligands: G4K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-03-20
Ligands: G4K
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Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 27
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-02-20 Classification: TRANSFERASE Ligands: G4T |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: G4T
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Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 31
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2019-02-20 Classification: TRANSFERASE Ligands: G4Q |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: G4Q
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Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 30B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2019-02-20 Classification: TRANSFERASE Ligands: G4N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: G4N
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Crystal Structure Of Akt1 In Complex With Covalent-Allosteric Akt Inhibitor 24B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2019-02-20 Classification: TRANSFERASE Ligands: G4H |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: G4H
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Crystal Structure Of Glycogen Synthase Kinase-3 Beta (Gsk3B) In Complex With Pik-75
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2018-06-20 Classification: TRANSFERASE Ligands: CL, F4N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-20
Ligands: CL, F4N
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Covalent Inhibitor 4B Bound To The Lipid Pocket Of P38Alpha Mutant S252C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-09-06 Classification: TRANSFERASE Ligands: 9O5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-06
Ligands: 9O5
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Covalent Inhibitor 4A Bound To The Lipid Pocket Of P38Alpha Mutant S251C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-09-06 Classification: TRANSFERASE Ligands: 9O2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-06
Ligands: 9O2
