Search Count: 41
 |
First Bromodomain Of Brdt Liganded With Inhibitor Gxh-Iv-076 (Compound 33)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2026-07-29 Classification: TRANSCRIPTION/INHIBITOR Ligands: ZNJ, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-29
Ligands: ZNJ, EDO, CL
 |
Brd4 Bd1 Liganded With Macrocyclic Compound 2B (Jj-Ii-352A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2025-03-19 Classification: TRANSCRIPTION Ligands: A1AAL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-03-19
Ligands: A1AAL, EDO
 |
Brd4 Bd1 Liganded With Macrocyclic Compound 2D (Jj-Ii-363A)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.22 Å Release Date: 2024-12-18 Classification: TRANSCRIPTION Ligands: YPB, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-12-18
Ligands: YPB, EDO
 |
Crystal Structure Of The Brd2-Bd2 In Complex With A Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2023-05-03 Classification: TRANSCRIPTION Ligands: EDO, QJ1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-05-03
Ligands: EDO, QJ1
 |
Crystal Structure Of Bptf Bromodomain In Complex With 4-Chloro-5-{4-[(Dimethylamino)Methyl]Anilino}-2-Methylpyridazin-3(2H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2022-08-24 Classification: GENE REGULATION/INHIBITOR Ligands: 7WE, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: 7WE, EDO
 |
Crystal Structure Of Bptf Bromodomain In Complex With 4-Chloro-2-Methyl-5-[(1,2,3,4-Tetrahydroisoquinolin-7-Yl)Amino]Pyridazin-3(2H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.58 Å Release Date: 2022-08-24 Classification: GENE REGULATION/INHIBITOR Ligands: 7WN, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: 7WN, EDO
 |
Crystal Structure Of Bptf Bromodomain In Complex With 5-[4-(Aminomethyl)Anilino]-4-Chloro-2-Methylpyridazin-3(2H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.73 Å Release Date: 2022-08-24 Classification: GENE REGULATION/INHIBITOR Ligands: 7WZ, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: 7WZ, CA
 |
Crystal Structure Of Bptf Bromodomain In Complex With 4-Chloro-2-Methyl-5-[(1,2,3,4-Tetrahydroisoquinolin-6-Yl)Amino]Pyridazin-3(2H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2022-08-24 Classification: GENE REGULATION/INHIBITOR Ligands: 7XE, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-24
Ligands: 7XE, CA
 |
Crystal Structure Of Bptf Bromodomain In Complex With Inhibitor Pdy-3-077
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.66 Å Release Date: 2022-08-10 Classification: GENE REGULATION/INHIBITOR Ligands: P2L, DMS, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-10
Ligands: P2L, DMS, EDO
 |
Crystal Structure Of Bptf Bromodomain In Complex With Inhibitor Hz-03-112
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.39 Å Release Date: 2022-08-10 Classification: GENE REGULATION/INHIBITOR Ligands: Y9P, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-10
Ligands: Y9P, EDO
 |
Crystal Structure Of Bptf Bromodomain In Complex With Inhibitor Pdy-3-093
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.44 Å Release Date: 2022-08-10 Classification: GENE REGULATION/INHIBITOR Ligands: YC4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-10
Ligands: YC4, EDO
 |
Crystal Structure Of Bptf Bromodomain In Complex With Inhibitor Hz-01-105
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2022-08-10 Classification: GENE REGULATION/INHIBITOR Ligands: DMS, YBV, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-10
Ligands: DMS, YBV, EDO
 |
Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With Sj001011461-1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.18 Å Release Date: 2022-08-03 Classification: CELL CYCLE Ligands: EDO, 5Z0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: EDO, 5Z0
 |
Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With Sj001010551-2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.05 Å Release Date: 2022-08-03 Classification: CELL CYCLE Ligands: EDO, 5ZQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-08-03
Ligands: EDO, 5ZQ
 |
Crystal Structure Of The First Bromodomain Of Human Brd4 In Complex With Inhibitor Jj-Ii-131
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2022-07-06 Classification: TRANSCRIPTION/INHIBITOR Ligands: XZG, EDO, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-06
Ligands: XZG, EDO, NA
 |
Crystal Structure Of The First Bromodomain (Bd1) Of Human Brd4 Bound To Gxh-Ii-076
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2022-05-11 Classification: GENE REGULATION Ligands: ZNJ, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-05-11
Ligands: ZNJ, EDO
 |
Crystal Structure Of Bptf Bromodomain In Complex With Cb02-092
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2022-02-16 Classification: GENE REGULATION Ligands: YOV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-02-16
Ligands: YOV
 |
Cocrystal Of Brd4(D1) With N,N-Dimethyl-2-[(3R)-3-(5-{2-[2-Methyl-5-(Propan-2-Yl)Phenoxy]Pyrimidin-4-Yl}-4-[4-(Trifluoromethyl)Phenyl]-1H-Imidazol-1-Yl)Pyrrolidin-1-Yl]Ethan-1-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2022-01-19 Classification: GENE REGULATION/INHIBITOR Ligands: EDO, 2IR, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: EDO, 2IR, CL
 |
Crystal Structure Of Brd4(D1) With 4-[4-(4-Bromophenyl)-1-(Piperidin-4-Yl)-1H-Imidazol-5-Yl]-N-(3,5-Dimethylphenyl)Pyrimidin-2-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.41 Å Release Date: 2022-01-19 Classification: GENE REGULATION/INHIBITOR Ligands: EDO, 7ZB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: EDO, 7ZB
 |
Crystal Of Brd4(D1) With 2-[(3S)-3-{5-[2-(3,5-Dimethylphenoxy)Pyrimidin-4-Yl]-4-(4-Iodophenyl)-1H-Imidazol-1-Yl}Pyrrolidin-1-Yl]Ethan-1-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.43 Å Release Date: 2022-01-19 Classification: GENE REGULATION/INHIBITOR Ligands: EDO, 7ZT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-01-19
Ligands: EDO, 7ZT