Search Count: 33
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Structure Of Khk In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2020-09-23 Classification: TRANSFERASE Ligands: RYS, SO4, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: RYS, SO4, CIT
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Structure Of Khk In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2020-09-23 Classification: TRANSFERASE Ligands: RZA, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: RZA, SO4
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Structure Of Khk In Complex With Compound 4 (6-[(1~{S},5~{R})-6-(Hydroxymethyl)-3-Azabicyclo[3.1.0]Hexan-3-Yl]-2-[(2~{S},3~{R})-2-Methyl-3-Oxidanyl-Azetidin-1-Yl]-4-(Trifluoromethyl)Pyridine-3-Carbonitrile)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2020-09-23 Classification: TRANSFERASE Ligands: S6J, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: S6J, SO4
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Structure Of Khk In Complex With Compound 6 (2-[(1~{R},5~{S})-3-[5-Cyano-6-[(2~{S},3~{R})-2-Methyl-3-Oxidanyl-Azetidin-1-Yl]-4-(Trifluoromethyl)Pyridin-2-Yl]-3-Azabicyclo[3.1.0]Hexan-6-Yl]Ethanoic Acid)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.54 Å Release Date: 2020-09-23 Classification: TRANSFERASE Ligands: S6S, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: S6S, SO4
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Structure Of Khk In Complex With Compound 8 (2-[(1~{S},5~{R})-3-[2-[(2~{S})-2-Methylazetidin-1-Yl]-6-(Trifluoromethyl)Pyrimidin-4-Yl]-3-Azabicyclo[3.1.0]Hexan-6-Yl]Ethanoic Acid)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2020-09-23 Classification: TRANSFERASE Ligands: S6D, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-09-23
Ligands: S6D, SO4
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Structure Of Human Ketohexokinase Complexed With Hits From Fragment Screening
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.16 Å Release Date: 2017-09-13 Classification: TRANSFERASE Ligands: A4G, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-13
Ligands: A4G, SO4
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Structure Of Human Ketohexokinase Complexed With Hits From Fragment Screening
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2017-09-13 Classification: TRANSFERASE Ligands: A1Y, SO4, CIT, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-13
Ligands: A1Y, SO4, CIT, GOL
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Structure Of Human Ketohexokinase Complexed With Hits From Fragment Screening
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.74 Å Release Date: 2017-09-13 Classification: TRANSFERASE Ligands: A2J, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-13
Ligands: A2J, SO4, GOL
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Structure Of Human Ketohexokinase Complexed With Hits From Fragment Screening
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-09-13 Classification: TRANSFERASE Ligands: A3J, SO4, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-13
Ligands: A3J, SO4, CL
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Structure Of Human Ketohexokinase Complexed With Hits From Fragment Screening
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2017-09-13 Classification: TRANSFERASE Ligands: A3Y, SO4, CIT, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-13
Ligands: A3Y, SO4, CIT, GOL
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Structure Of Human Ketohexokinase Complexed With Hits From Fragment Screening
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2017-09-13 Classification: TRANSFERASE Ligands: A4J, SO4, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-09-13
Ligands: A4J, SO4, CIT
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Covalent Inhibitor Of Lyplal1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2016-07-20 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: 6WG, NO3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-07-20
Ligands: 6WG, NO3
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Crystal Structure Of Glucokinase-Activator Complex
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2013-07-24 Classification: Transferase/transferase activator Ligands: GLC, 926 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-07-24
Ligands: GLC, 926
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Glucokinase In Complex With An Activator And Glucose
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-02-08 Classification: TRANSFERASE/TRANSFERASE ACTIVATOR Ligands: GLC, 0H4, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-08
Ligands: GLC, 0H4, NA
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Glucokinase In Complex With Glucose And Atpgs
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2012-02-08 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GLC, NA, AGS, 0H5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-08
Ligands: GLC, NA, AGS, 0H5
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Glucokinase In Complex With Glucose And Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2012-02-08 Classification: TRANSFERASE/TRANSFERASE ACTIVATOR Ligands: GLC, 0H6, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-08
Ligands: GLC, 0H6, NA
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Insights Into Glucokinase Activation Mechanism: Observation Of Multiple Distinct Protein Conformations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2012-02-08 Classification: TRANSFERASE Ligands: GLC, 4DC, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-08
Ligands: GLC, 4DC, IOD
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Crystal Structure Of Human Glucokinase In Complex With Glucose And Activator
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2012-02-08 Classification: TRANSFERASE/TRANSFERASE ACTIVATOR Ligands: GLC, S41, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-08
Ligands: GLC, S41, NA
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Glucokinase In Complex With Activator And Glucose
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2011-09-14 Classification: TRANSFERASE Ligands: GLC, NA, S41 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-09-14
Ligands: GLC, NA, S41
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Thermodynamic And Structure Guided Design Of Statin Hmg-Coa Reductase Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2008-06-17 Classification: OXIDOREDUCTASE Ligands: 3HI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-06-17
Ligands: 3HI