Search Count: 16
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Crystal Structure Of Sars Cov-2 3Cl Protease In Complex With Gsk4365096A
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2024-03-13 Classification: HYDROLASE Ligands: WTE |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-03-13
Ligands: WTE
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Crystal Structure Of Sars Cov-2 3Cl Protease In Complex With Gsk4365097A
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2024-02-14 Classification: HYDROLASE Ligands: WTV, GOL, CL |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: WTV, GOL, CL
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Crystal Structure Of Sars Cov-2 3Cl Protease In Complex With Gsk4365096A
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION Resolution:2.02 Å Release Date: 2024-02-14 Classification: HYDROLASE Ligands: A1ADS |
Organism: Severe acute respiratory syndrome coronavirus 2
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: A1ADS
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Sara Cov-2 3C-Like Protease In Complex With Gsk3487016A
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2024-02-14 Classification: HYDROLASE Ligands: WYR, EDO |
Organism: Severe acute respiratory syndrome coronavirus
Method: X-RAY DIFFRACTION
Release Date: 2024-02-14
Ligands: WYR, EDO
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Optimization Of Tead P-Site Binding Fragment Hit Into In Vivo Active Lead Msc-4106
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.19 Å Release Date: 2022-07-13 Classification: TRANSCRIPTION Ligands: JJU, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-13
Ligands: JJU, SO4
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Human Tead3 In Complex With 1-Cyclopentyl-1H-Pyrazolo[3,4-B]Pyridine-5-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2022-07-13 Classification: TRANSCRIPTION Ligands: JIK |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2022-07-13
Ligands: JIK
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1.98A Structure Of Gsk945237 With S.Aureus Dna Gyrase And Singly Nicked Dna
Organism: Staphylococcus aureus, Staphylococcus aureus (strain n315), Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2016-05-25 Classification: ISOMERASE Ligands: MN, GOL, CL, 6EJ |
Organism: Staphylococcus aureus, Staphylococcus aureus (strain n315), Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: MN, GOL, CL, 6EJ
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2.5A Structure Of Gsk945237 With S.Aureus Dna Gyrase And Dna.
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2016-05-25 Classification: ISOMERASE Ligands: MN, GOL, 6EJ |
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: MN, GOL, 6EJ
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Novel Hydroxyl Tricyclics (E.G. Gsk966587) As Potent Inhibitors Of Bacterial Type Iia Topoisomerases
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2013-08-07 Classification: ISOMERASE Ligands: MN, AE8 |
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2013-08-07
Ligands: MN, AE8
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Crystal Structure Of Catalytic Core Of A. Baumannii Topo Iv (Pare- Parc Fusion Truncate)
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2010-09-01 Classification: ISOMERASE Ligands: SO4, GOL |
Organism: Acinetobacter baumannii
Method: X-RAY DIFFRACTION
Release Date: 2010-09-01
Ligands: SO4, GOL
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Crystal Structure Of Moxifloxacin, Dna, And A. Baumannii Topo Iv (Pare-Parc Fusion Truncate)
Organism: Acinetobacter baumannii, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:3.25 Å Release Date: 2010-09-01 Classification: ISOMERASE/DNA/ANTIBIOTIC Ligands: MG, MFX |
Organism: Acinetobacter baumannii, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2010-09-01
Ligands: MG, MFX
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The Twinned 3.35A Structure Of S. Aureus Gyrase Complex With Ciprofloxacin And Dna
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:3.35 Å Release Date: 2010-08-25 Classification: ISOMERASE/DNA/ANTIBIOTIC Ligands: MN, CPF |
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2010-08-25
Ligands: MN, CPF
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The 3.1A Crystal Structure Of The Catalytic Core (B'A' Region) Of Staphylococcus Aureus Dna Gyrase
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2010-08-04 Classification: ISOMERASE Ligands: CA |
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION
Release Date: 2010-08-04
Ligands: CA
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The 2.98A Crystal Structure Of The Catalytic Core (B'A' Region) Of Staphylococcus Aureus Dna Gyrase
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION Resolution:2.98 Å Release Date: 2010-08-04 Classification: ISOMERASE Ligands: HOH |
Organism: Staphylococcus aureus
Method: X-RAY DIFFRACTION
Release Date: 2010-08-04
Ligands: HOH
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The 3.5A Crystal Structure Of The Catalytic Core (B'A' Region) Of Staphylococcus Aureus Dna Gyrase Complexed With Gsk299423 And Dna
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2010-08-04 Classification: ISOMERASE Ligands: RXV |
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2010-08-04
Ligands: RXV
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The 2.1A Crystal Structure Of S. Aureus Gyrase Complex With Gsk299423 And Dna
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2010-08-04 Classification: ISOMERASE Ligands: MN, RXV |
Organism: Staphylococcus aureus, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2010-08-04
Ligands: MN, RXV
