Search Count: 10
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Covalent Inhibitor Vvd-442 Bound To The Ras Binding Domain (Rbd) Of Pi3Ka
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.83 Å Release Date: 2025-01-01 Classification: PROTEIN BINDING Ligands: A1BF9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-01-01
Ligands: A1BF9
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Keap1 Btb Domain In Complex With The Covalent Activator Vvd-065
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2024-10-23 Classification: PROTEIN BINDING Ligands: A1BCT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-10-23
Ligands: A1BCT
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Crystal Structure Of Werner Helicase Fragment 517-945 In Complex With Adp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.57 Å Release Date: 2024-05-01 Classification: HYDROLASE Ligands: ADP, CD, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-01
Ligands: ADP, CD, EDO, CL
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Crystal Structure Of Werner Helicase Fragment 517-945 In Complex With Atp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2024-05-01 Classification: HYDROLASE Ligands: ZN, ATP, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-01
Ligands: ZN, ATP, MG
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Crystal Structure Of Werner Helicase Fragment 517-945 In Covalent Complex With N-[(E,1S)-1-Cyclopropyl-3-Methylsulfonylprop-2-Enyl]-2-(1,1-Difluoroethyl)-4-Phenoxypyrimidine-5-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2024-05-01 Classification: HYDROLASE Ligands: ZN, ADP, X1L, GOL, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-01
Ligands: ZN, ADP, X1L, GOL, NA
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Crystal Structure Of Small Molecule Ars-1620 Covalently Bound To K-Ras G12C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2018-02-07 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: CA, 91S, GOL, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-02-07
Ligands: CA, 91S, GOL, GDP
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Crystal Structure Of Small Molecule Ars-853 Covalently Bound To K-Ras G12C
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2016-01-13 Classification: HYDROLASE Ligands: MG, GOL, 5UT, GLY, GDP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-01-13
Ligands: MG, GOL, 5UT, GLY, GDP
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Crystal Structure Of Type Ii Inhibitor Ng25 Bound To Tak1-Tab1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2014-07-30 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: NG2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-07-30
Ligands: NG2
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Discovery Of Potent And Selective Covalent Inhibitors Of Jnk
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2012-02-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CQQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-01
Ligands: CQQ
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Discovery Of Potent And Selective Covalent Inhibitors Of Jnk
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.97 Å Release Date: 2012-02-01 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0F0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-02-01
Ligands: 0F0
