Search Count: 36
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Cdk2/Cycline Bound To Compound 11 With P-Loop In The Ee And Cc Conformations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2025-04-30 Classification: CELL CYCLE Ligands: A1CAE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-30
Ligands: A1CAE
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Cdk2/Cycline Bound To Compound 16 With P-Loop In The Ee Conformation
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.98 Å Release Date: 2025-04-30 Classification: CELL CYCLE Ligands: A1CAH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-30
Ligands: A1CAH
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Cdk2/Cycline Bound To Compound 19 With P-Loop In The Ee And Ec Conformations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2025-04-30 Classification: CELL CYCLE Ligands: A1CAF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-30
Ligands: A1CAF
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Cdk2/Cycline Bound To Compound 20 With P-Loop In The Ee And Cc Conformations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2025-04-30 Classification: CELL CYCLE Ligands: A1CAG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-30
Ligands: A1CAG
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Cdk2/Cycline Bound To Compound 21 With P-Loop In The Ee And Cc Conformations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2025-04-30 Classification: CELL CYCLE Ligands: A1CAI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-30
Ligands: A1CAI
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Crystal Structure Of Hdac8 In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.88 Å Release Date: 2020-04-01 Classification: HYDROLASE Ligands: C7, ZN, K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: C7, ZN, K
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Crystal Structure Of Hdac8 In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2020-04-01 Classification: HYDROLASE Ligands: M8G, ZN, K, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: M8G, ZN, K, GOL
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Crystal Structure Of Hdac8 In Complex With Compound 30
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2020-04-01 Classification: HYDROLASE Ligands: ZN, K, M7Y, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-04-01
Ligands: ZN, K, M7Y, EDO
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Taf1-Bd2 In Complex With Cpd27 (6-(But-3-En-1-Yl)-4-(1-Methyl-6-(Morpholine-4-Carbonyl)-1H-Benzo[D]Imidazol-4-Yl)-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-11-14 Classification: Transcription/Inhibitor Ligands: G9V |
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2018-11-14
Ligands: G9V
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Taf1-Bd2 In Complex With Cpd8 (6-(But-3-En-1-Yl)-4-(3-(Morpholine-4-Carbonyl)Phenyl)-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2018-10-31 Classification: Transcription/Inhibitor Ligands: G9Y |
Organism: Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2018-10-31
Ligands: G9Y
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Cecr2 In Complex With Cpd6 (6-Allyl-N,2-Dimethyl-7-Oxo-N-(1-(1-Phenylethyl)Piperidin-4-Yl)-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridine-4-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2017-06-14 Classification: Transcription/Inhibitor Ligands: SO4, 96V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-14
Ligands: SO4, 96V
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Crystal Structure Of The Bromodomain Of Human Crebbp Bound To Pyrazolopiperidine Scaffold
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.38 Å Release Date: 2016-11-02 Classification: TRANSFERASE Ligands: 6XB, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: 6XB, DMS
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Crebbp Bromodomain In Complex With Cpd 44 (3-((5-Acetyl-1-(Cyclopropylmethyl)-4,5,6,7-Tetrahydro-1H-Pyrazolo[4,3-C]Pyridin-3-Yl)Amino)-N-Isopropylbenzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.09 Å Release Date: 2016-11-02 Classification: TRANSFERASE Ligands: 6XG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: 6XG, EDO
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Crebbp Bromodomain In Complex With Cpd59 ((S)-1-(3-((2-Fluoro-4-(1-Methyl-1H-Pyrazol-4-Yl)Phenyl)Amino)-1-(Tetrahydrofuran-3-Yl)-6,7-Dihydro-1H-Pyrazolo[4,3-C]Pyridin-5(4H)-Yl)Ethanone)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2016-11-02 Classification: TRANSFERASE Ligands: 6XH, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: 6XH, EDO, DMS
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Brd4 Bromodomain In Complex With Cpd59 ((S)-1-(3-((2-Fluoro-4-(1-Methyl-1H-Pyrazol-4-Yl)Phenyl)Amino)-1-(Tetrahydrofuran-3-Yl)-6,7-Dihydro-1H-Pyrazolo[4,3-C]Pyridin-5(4H)-Yl)Ethanone)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.14 Å Release Date: 2016-11-02 Classification: TRANSFERASE Ligands: EDO, DMS, GOL, PEG, 6XH |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-11-02
Ligands: EDO, DMS, GOL, PEG, 6XH
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Brd9 In Complex With Cpd1 (6-Methyl-1,6-Dihydro-7H-Pyrrolo[2,3-C]Pyridin-7-One)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.04 Å Release Date: 2016-10-12 Classification: RNA BINDING PROTEIN Ligands: EDO, PEG, 67N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: EDO, PEG, 67N
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Brd9 In Complex With Cpd2 (N,N-Dimethyl-3-(6-Methyl-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)Benzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.18 Å Release Date: 2016-10-12 Classification: RNA BINDING PROTEIN Ligands: 67B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: 67B
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Brd9 In Complex With Cpd4 ((E)-3-(6-(But-2-En-1-Yl)-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)-N,N-Dimethylbenzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2016-10-12 Classification: TRANSCRIPTION Ligands: 69G |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: 69G
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Brd4 In Complex With Cpd2 (N,N-Dimethyl-3-(6-Methyl-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)Benzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2016-10-12 Classification: TRANSCRIPTION Ligands: 67B, EDO, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: 67B, EDO, DMS
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Brd4 In Complex With Cpd4 ((E)-3-(6-(But-2-En-1-Yl)-7-Oxo-6,7-Dihydro-1H-Pyrrolo[2,3-C]Pyridin-4-Yl)-N,N-Dimethylbenzamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2016-10-12 Classification: TRANSCRIPTION Ligands: PGE, EDO, DMS, 69G, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-10-12
Ligands: PGE, EDO, DMS, 69G, GOL
