Search Count: 22
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Discovery And Clinical Validation Of Rly-4008, The First Highly Selective Fgfr2 Inhibitor With Activity Across Fgfr2 Alterations And Resistance Mutations
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.79 Å Release Date: 2023-06-07 Classification: TRANSFERASE/INHIBITOR Ligands: WCJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-07
Ligands: WCJ
 |
Crystal Structure Of Abnu: An Exo-Specific Intermolecular Diels-Alderase
Organism: Frankia sp. cc1.17
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2021-08-18 Classification: ISOMERASE Ligands: EDO, DMS |
Organism: Frankia sp. cc1.17
Method: X-RAY DIFFRACTION
Release Date: 2021-08-18
Ligands: EDO, DMS
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Pyri4 In Complex With Intermolecular Diels-Alder Product
Organism: Streptomyces rugosporus
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2021-08-18 Classification: ISOMERASE Ligands: HOF, GOL |
Organism: Streptomyces rugosporus
Method: X-RAY DIFFRACTION
Release Date: 2021-08-18
Ligands: HOF, GOL
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Prmt5 Bound To Pbm Peptide From Riok1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.11 Å Release Date: 2020-08-26 Classification: TRANSFERASE/SPLICING Ligands: SFG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-26
Ligands: SFG
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Prmt5 Bound To The Pbm Peptide From Picln
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.86 Å Release Date: 2020-08-26 Classification: Transferase/Splicing Ligands: SFG, ACE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-26
Ligands: SFG, ACE
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Brd4 Bromodomain 1 In Complex With Triple Cdk4/6-Pi3K-Bet Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2020-08-26 Classification: TRANSCRIPTION Ligands: YR0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-26
Ligands: YR0
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Brd4 Bromodomain 1 In Complex With Multi-Action Inhibitor Srx3212P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2020-08-05 Classification: TRANSCRIPTION Ligands: ZVP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-05
Ligands: ZVP
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Brd4 Bromodomain 1 In Complex With Multi-Action Inhibitor Srx3212
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2020-08-05 Classification: TRANSCRIPTION Ligands: KV9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-05
Ligands: KV9
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Brd4 Bromodomain 1 In Complex With Multi-Action Inhibitor Sf2523P
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2020-08-05 Classification: TRANSCRIPTION Ligands: UT4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-08-05
Ligands: UT4
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Structure Of Ubiquitin Activating Enzyme (Uba1) In Complex With Ubiquitin And Tak-243
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Bos taurus
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2017-11-01 Classification: LIGASE/LIGASE INHIBITOR Ligands: 61T |
Organism: Saccharomyces cerevisiae (strain atcc 204508 / s288c), Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2017-11-01
Ligands: 61T
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Structure Of Yeast 20S Open-Gate Proteasome With Compound 20
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.65 Å Release Date: 2012-06-13 Classification: Hydrolase/Hydrolase Inhibitor Ligands: MG, 3SD, MES |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2012-06-13
Ligands: MG, 3SD, MES
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Structure Of Yeast 20S Open-Gate Proteasome With Compound 34
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2012-06-13 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: MG, P3N, MES |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2012-06-13
Ligands: MG, P3N, MES
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Structure Of S. Pombe Nuclear Import Adaptor Nro1 (Space Group P21)
Organism: Schizosaccharomyces pombe
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2011-09-21 Classification: TRANSLATION Ligands: SO4, CL, EDO |
Organism: Schizosaccharomyces pombe
Method: X-RAY DIFFRACTION
Release Date: 2011-09-21
Ligands: SO4, CL, EDO
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Structure Of S. Pombe Nuclear Import Adaptor Nro1 (Space Group P6522)
Organism: Schizosaccharomyces pombe
Method: X-RAY DIFFRACTION Resolution:3.50 Å Release Date: 2011-09-21 Classification: TRANSLATION |
Organism: Schizosaccharomyces pombe
Method: X-RAY DIFFRACTION
Release Date: 2011-09-21
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Structure Of Yeast 20S Open-Gate Proteasome With Compound 24
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-07-20 Classification: Hydrolase/Hydrolase Inhibitor Ligands: MG, OEU, MES |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2011-07-20
Ligands: MG, OEU, MES
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Structure Of Yeast 20S Open-Gate Proteasome With Compound 25
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2011-07-20 Classification: Hydrolase/Hydrolase Inhibitor Ligands: MG, 3OE, MES |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2011-07-20
Ligands: MG, 3OE, MES
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Structure Of Yeast 20S Proteasome With Bortezomib
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.68 Å Release Date: 2011-05-18 Classification: HYDROLASE Ligands: BO2 |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2011-05-18
Ligands: BO2
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Structure Of Yeast 20S Open-Gate Proteasome With Compound 6
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2011-05-18 Classification: HYDROLASE Ligands: MG, LZT, MES |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2011-05-18
Ligands: MG, LZT, MES
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Structure Of Yeast 20S Open-Gate Proteasome With Compound 8
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.78 Å Release Date: 2011-05-18 Classification: HYDROLASE Ligands: MG, L2T, MES |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2011-05-18
Ligands: MG, L2T, MES
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Structure Of Yeast 20S Open-Gate Proteasome With Compound 16
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2011-05-18 Classification: HYDROLASE Ligands: MG, L3T, MES |
Organism: Saccharomyces cerevisiae
Method: X-RAY DIFFRACTION
Release Date: 2011-05-18
Ligands: MG, L3T, MES