Search Count: 37
![]() |
Retinoic Acid Receptor-Related Orphan Receptor (Ror) Gamma In Complex With Allosteric Compound 28
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.87 Å Release Date: 2020-03-04 Classification: TRANSCRIPTION Ligands: Q3Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-04
Ligands: Q3Y
![]() |
Nitric Oxide Reductase From Roseobacter Denitrificans (Rdnor)
Organism: Roseobacter denitrificans (strain atcc 33942 / och 114)
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2016-05-25 Classification: OXIDOREDUCTASE Ligands: HEM, UNL, CA, FE, HEC, CU |
Organism: Roseobacter denitrificans (strain atcc 33942 / och 114)
Method: X-RAY DIFFRACTION
Release Date: 2016-05-25
Ligands: HEM, UNL, CA, FE, HEC, CU
![]() |
Crystal Structure Of The Ror(Gamma)T Ligand Binding Domain In Complex With 4-(1-(2-Chloro-6-(Trifluoromethyl)Benzoyl)-1H-Indazol-3-Yl)Benzoic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.32 Å Release Date: 2015-12-23 Classification: TRANSCRIPTION Ligands: 4F1, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-23
Ligands: 4F1, MG
![]() |
Identification Of A Novel Allosteric Binding Site For Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2015-12-16 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 4F1, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: 4F1, GOL, SO4
![]() |
Identification Of A Novel Allosteric Binding Site For Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.23 Å Release Date: 2015-12-16 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 4Y5, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: 4Y5, GOL
![]() |
Identification Of A Novel Allosteric Binding Site For Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2015-12-16 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 4Y6, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: 4Y6, SO4, GOL
![]() |
Identification Of A Novel Allosteric Binding Site For Rorgt Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.08 Å Release Date: 2015-12-16 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 4Y7, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-12-16
Ligands: 4Y7, GOL
![]() |
Structural Basis For Kinase Selectivity Of Three Clinical P38Alpha Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2012-07-04 Classification: TRANSFERASE Ligands: SB2, BOG, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-04
Ligands: SB2, BOG, EDO
![]() |
X-Ray Structure Of P38Alpha Bound To Tak-715
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2012-06-13 Classification: TRANSFERASE Ligands: T75, BOG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-06-13
Ligands: T75, BOG
![]() |
X-Ray Structure Of P38Alpha Bound To Scio-469
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2012-06-13 Classification: TRANSFERASE Ligands: 469, BOG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-06-13
Ligands: 469, BOG
![]() |
X-Ray Structure Of P38Alpha Bound To Vx-745
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2012-06-13 Classification: TRANSFERASE Ligands: 52P, BOG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-06-13
Ligands: 52P, BOG
![]() |
Pr X-Ray Structures In Agonist Conformations Reveal Two Different Mechanisms For Partial Agonism In 11Beta-Substituted Steroids
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-04-25 Classification: TRANSCRIPTION Ligands: OR8, SO4, A2K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-25
Ligands: OR8, SO4, A2K
![]() |
Factor Xia In Complex With A Clorophenyl-Tetrazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-04-11 Classification: Hydrolase/Hydrolase inhibitor Ligands: CIT, O58 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-11
Ligands: CIT, O58
![]() |
Benzothiazinone Inhibitor In Complex With Fxia
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.58 Å Release Date: 2012-04-11 Classification: Hydrolase/Hydrolase Inhibitor Ligands: CIT, TRS, O61 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-11
Ligands: CIT, TRS, O61
![]() |
Pr X-Ray Structures In Agonist Conformations Reveal Two Different Mechanisms For Partial Agonism In 11Beta-Substituted Steroids
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-04-04 Classification: TRANSCRIPTION Ligands: AS0, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-04-04
Ligands: AS0, SO4
![]() |
Novel Atp-Competitive Mk2 Inhibitors With Potent Biochemical And Cell-Based Activity Throughout The Series
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2011-12-14 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: I85 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-12-14
Ligands: I85
![]() |
Structural Basis For Agonism And Antagonism For A Set Of Chemically Related Progesterone Receptor Modulators
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2011-08-17 Classification: RECEPTOR Ligands: OR8, GOL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-17
Ligands: OR8, GOL, SO4
![]() |
Structural Basis For Agonism And Antagonism For A Set Of Chemically Related Progesterone Receptor Modulators
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2011-08-17 Classification: HORMONE RECEPTOR Ligands: ORB, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-17
Ligands: ORB, SO4
![]() |
Structural Basis For Agonism And Antagonism For A Set Of Chemically Related Progesterone Receptor Modulators
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2011-08-17 Classification: RECEPTOR Ligands: OR8, SO4, GOL, ORC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-08-17
Ligands: OR8, SO4, GOL, ORC
![]() |
Mk3 Kinase Bound To Compound 5B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.09 Å Release Date: 2011-05-25 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 05B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: 05B
