Search Count: 23
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Crystal Structure Of Mouse Btk Kinase Domain In Complex With Compound 9A
Organism: Mus musculus
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2019-01-30 Classification: TRANSFERASE Ligands: JVP |
Organism: Mus musculus
Method: X-RAY DIFFRACTION
Release Date: 2019-01-30
Ligands: JVP
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Crystal Structure Of Itk In Complex With Compound 1 [4-(Carbamoylamino)-1-(Naphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: M0Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: M0Y
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Crystal Structure Of Itk In Complex With Compound 5 {4-(Carbamoylamino)-1-(7-Methoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide}
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: M0Z |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: M0Z
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Crystal Structure Of Itk In Complex With Compound 7 [4-(Carbamoylamino)-1-(7-Ethoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1YZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 1YZ
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Crystal Structure Of Itk In Complex With Compound 8 [4-(Carbamoylamino)-1-(7-Propoxynaphthalen-1-Yl)-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 1E0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: 1E0
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Crystal Structure Of Itk In Complex With Compound 9 [4-(Carbamoylamino)-1-[7-(Propan-2-Yloxy)Naphthalen-1-Yl]-1H-Pyrazole-3-Carboxamide]
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.55 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QWS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: QWS
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Crystal Structure Of Itk In Complex With Compound 9 [4-(Carbamoylamino)-1-[7-(Propan-2-Yloxy)Naphthalen-1-Yl]-1H-Pyrazole-3-Carboxamide] And Adp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.52 Å Release Date: 2014-04-02 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QWS, ADP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-04-02
Ligands: QWS, ADP
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Crystal Structure Of Ppargamma In Complex With Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2013-08-21 Classification: TRANSCRIPTION/TRANSCRIPTION INHIBITOR Ligands: 14R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-08-21
Ligands: 14R
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X-Ray Crystal Structure Of The Nuclear Hormone Receptor Ppar-Gamma In A Complex With A Compound With Dual Ppar Gamma Agonism And Angiotensin Ii Type I Receptor Antagonism Activity
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2012-03-14 Classification: NUCLEAR PROTEIN Ligands: HIG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-03-14
Ligands: HIG
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X-Ray Crystal Structure Of The Nuclear Hormone Receptor Ppar-Gamma In A Complex With A Ppar Gamma/Alpha Dual Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2009-10-13 Classification: TRANSCRIPTION Ligands: UNT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-10-13
Ligands: UNT
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X-Ray Crystal Structure Of The Nuclear Hormone Receptor Ppar-Gamma In A Complex With A Ppar Gamma/Alpha Dual Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-10-14 Classification: hormone receptor Ligands: L92 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-10-14
Ligands: L92
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Crystal Structure Of Aspartate Semialdehyde Dehydrogenase Ii From Vibrio Cholerae
Organism: Vibrio cholerae
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2008-04-08 Classification: OXIDOREDUCTASE |
Organism: Vibrio cholerae
Method: X-RAY DIFFRACTION
Release Date: 2008-04-08
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Crystal Structure Of Aspartate Semialdehyde Dehydrogenase Ii Complexed With Asa From Vibrio Cholerae
Organism: Vibrio cholerae
Method: X-RAY DIFFRACTION Resolution:2.03 Å Release Date: 2008-04-08 Classification: OXIDOREDUCTASE Ligands: OEG |
Organism: Vibrio cholerae
Method: X-RAY DIFFRACTION
Release Date: 2008-04-08
Ligands: OEG
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Characterization Of Substrate Binding And Catalysis Of The Potential Antibacterial Target N-Acetylglucosamine-1-Phosphate Uridyltransferase (Glmu)
Organism: Haemophilus influenzae
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2008-01-15 Classification: TRANSFERASE Ligands: PEG, SO4, CO |
Organism: Haemophilus influenzae
Method: X-RAY DIFFRACTION
Release Date: 2008-01-15
Ligands: PEG, SO4, CO
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Characterization Of Substrate Binding And Catalysis Of The Potential Antibacterial Target N-Acetylglucosamine-1-Phosphate Uridyltransferase (Glmu)
Organism: Haemophilus influenzae
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2008-01-15 Classification: TRANSFERASE Ligands: UD1, PG4, PEG, SO4 |
Organism: Haemophilus influenzae
Method: X-RAY DIFFRACTION
Release Date: 2008-01-15
Ligands: UD1, PG4, PEG, SO4
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Characterization Of Substrate Binding And Catalysis Of The Potential Antibacterial Target N-Acetylglucosamine-1-Phosphate Uridyltransferase (Glmu)
Organism: Haemophilus influenzae
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2008-01-15 Classification: TRANSFERASE Ligands: H2U, MG, PG4, PGE, SO4 |
Organism: Haemophilus influenzae
Method: X-RAY DIFFRACTION
Release Date: 2008-01-15
Ligands: H2U, MG, PG4, PGE, SO4
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Characterization Of Substrate Binding And Catalysis Of The Potential Antibacterial Target N-Acetylglucosamine-1-Phosphate Uridyltransferase (Glmu)
Organism: Haemophilus influenzae
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2008-01-15 Classification: TRANSFERASE Ligands: UDP, PG4, PGE, SO4 |
Organism: Haemophilus influenzae
Method: X-RAY DIFFRACTION
Release Date: 2008-01-15
Ligands: UDP, PG4, PGE, SO4
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Characterization Of Substrate Binding And Catalysis Of The Potential Antibacterial Target N-Acetylglucosamine-1-Phosphate Uridyltransferase (Glmu)
Organism: Haemophilus influenzae
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2008-01-15 Classification: TRANSFERASE Ligands: URI, PG4, PGE, SO4 |
Organism: Haemophilus influenzae
Method: X-RAY DIFFRACTION
Release Date: 2008-01-15
Ligands: URI, PG4, PGE, SO4
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X-Ray Structure Of The Human Mitogen-Activated Protein Kinase Kinase 1 (Mek1) In A Complex With Ligand And Mgatp
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2007-10-02 Classification: TRANSFERASE Ligands: MG, MRA, ATP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-10-02
Ligands: MG, MRA, ATP
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Structure Of Aspartate-Semialdehyde Dehydrogenase From Methanococcus Jannaschii
Organism: Methanocaldococcus jannaschii
Method: X-RAY DIFFRACTION Resolution:2.29 Å Release Date: 2005-11-01 Classification: OXIDOREDUCTASE Ligands: NAP, MLA |
Organism: Methanocaldococcus jannaschii
Method: X-RAY DIFFRACTION
Release Date: 2005-11-01
Ligands: NAP, MLA
