Search Count: 30
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A Potent And Selective Ror Gamma Inhibitor For The Treatment Of Autoimmune Diseases
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.18 Å Release Date: 2026-04-29 Classification: DNA BINDING PROTEIN Ligands: A1MCM |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-04-29
Ligands: A1MCM
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Crystal Structure Of The Mutant Ror Gamma Lbd With Compound 28
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2025-07-30 Classification: NUCLEAR PROTEIN Ligands: A1MAM, EDO, ACT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-07-30
Ligands: A1MAM, EDO, ACT
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Optimization Efforts For Identification Of Novel Highly Potent Keap1-Nrf2 Protein-Protein Interaction Ihhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.32 Å Release Date: 2024-05-22 Classification: PEPTIDE BINDING PROTEIN Ligands: A1LVB, ACT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-22
Ligands: A1LVB, ACT, SO4
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Optimization Efforts For Identification Of Novel Highly Potent Keap1-Nrf2 Protein-Protein Interaction (Ppi) Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.42 Å Release Date: 2024-05-22 Classification: PEPTIDE BINDING PROTEIN Ligands: A1LVC, ACT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-05-22
Ligands: A1LVC, ACT, SO4
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Methyl And Fluorine Effects In Novel Orally Bioavailable Keap1/Nrf2 Ppi Inhibitor For Treatment Of Chronic Kidney Disease
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2023-06-14 Classification: PEPTIDE BINDING PROTEIN Ligands: SGO, DTT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: SGO, DTT, SO4
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Methyl And Fluorine Effects In Novel Orally Bioavailable Keap1/Nrf2 Ppi Inhibitor For Treatment Of Chronic Kidney Disease
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2023-06-14 Classification: PEPTIDE BINDING PROTEIN Ligands: SIU, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: SIU, SO4
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Methyl And Fluorine Effects In Novel Orally Bioavailable Keap1/Nrf2 Ppi Inhibitor For Treatment Of Chronic Kidney Disease
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2023-06-14 Classification: PEPTIDE BINDING PROTEIN Ligands: T6I, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-06-14
Ligands: T6I, SO4
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Discovery Of Functionally Selective Transforming Growth Factor Beta Type Ii Receptor (Tgf-Beta Rii) Inhibitors As Anti-Fibrosis Agents
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2021-06-16 Classification: IMMUNE SYSTEM Ligands: HJF |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-06-16
Ligands: HJF
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Crystal Structure Of Full-Length Cbnr Complexed With The Target Dna Complex
Organism: Cupriavidus necator
Method: X-RAY DIFFRACTION Resolution:3.60 Å Release Date: 2021-03-10 Classification: DNA BINDING PROTEIN/DNA |
Organism: Cupriavidus necator
Method: X-RAY DIFFRACTION
Release Date: 2021-03-10
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X-Ray Structure Of The Ligand-Free Human Trpv1 Ankyrin Repeat Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:4.47 Å Release Date: 2020-03-18 Classification: TRANSPORT PROTEIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-18
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Crystal Structure Of The Modified Fructosyl Peptide Oxidase From Aspergillus Nidulans, Seleno-Methionine Derivative
Organism: Aspergillus nidulans
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2019-05-15 Classification: OXIDOREDUCTASE Ligands: FAD, D1D, SO4 |
Organism: Aspergillus nidulans
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: FAD, D1D, SO4
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Crystal Structure Of The Modified Fructosyl Peptide Oxidase From Aspergillus Nidulans In Complex With Fsa, Seleno-Methionine Derivative
Organism: Aspergillus nidulans
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-05-15 Classification: OXIDOREDUCTASE Ligands: FAD, FSA, D1D, SO4 |
Organism: Aspergillus nidulans
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: FAD, FSA, D1D, SO4
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Crystal Structure Of The Modified Fructosyl Peptide Oxidase From Aspergillus Nidulans With R61G Mutation
Organism: Aspergillus nidulans
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2019-05-15 Classification: OXIDOREDUCTASE Ligands: FAD, SO4, D1D |
Organism: Aspergillus nidulans
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: FAD, SO4, D1D
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Crystal Structure Of The Modified Fructosyl Peptide Oxidase From Aspergillus Nidulans With R61G Mutation, In Complex With Fsa
Organism: Aspergillus nidulans
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2019-05-15 Classification: OXIDOREDUCTASE Ligands: FAD, FSA, D1D, SO4 |
Organism: Aspergillus nidulans
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: FAD, FSA, D1D, SO4
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Crystal Structure Of The Modified Fructosyl Peptide Oxidase From Aspergillus Nidulans With 7 Additional Mutations, In Complex With Fsa
Organism: Aspergillus nidulans
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2019-05-15 Classification: OXIDOREDUCTASE Ligands: FAD, FSA |
Organism: Aspergillus nidulans
Method: X-RAY DIFFRACTION
Release Date: 2019-05-15
Ligands: FAD, FSA
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Crystal Structure Of Hematopoietic Prostaglandin D Synthase In Complex With F092
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.74 Å Release Date: 2018-09-05 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: GSH, 93C, GOL, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-09-05
Ligands: GSH, 93C, GOL, MG
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Crystal Structure Of Cbnr_Dbd-Dna Complex
Organism: Cupriavidus necator
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2018-01-17 Classification: DNA BINDING PROTEIN |
Organism: Cupriavidus necator
Method: X-RAY DIFFRACTION
Release Date: 2018-01-17
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Crystal Structure Of Pim-1 In Complex With The Fluorescent Compound Skf86002
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2014-02-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SK8, GOL, CA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: SK8, GOL, CA
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Crystal Structure Of Pim1 In Complex With 2-{4-[(3-Aminopropyl)Amino]Quinazolin-2-Yl}Phenol (Resulting From Displacement Of Skf86002)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2014-02-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: Q17, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: Q17, GOL
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Crystal Structure Of Pim1 In Complex With The Inhibitor Quercetin (Resulting From Displacement Of Skf86002)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2014-02-12 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: QUE, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-02-12
Ligands: QUE, GOL