Search Count: 24
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Crystal Structure Of Chk1 In Complex With Prexasertib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2026-08-05 Classification: CELL CYCLE Ligands: A1DNH, PEG, GOL, EOH, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: A1DNH, PEG, GOL, EOH, EDO
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Crystal Structure Of Chk1 In Complex With Bbi-355
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.97 Å Release Date: 2026-08-05 Classification: CELL CYCLE Ligands: A1DNI, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
Ligands: A1DNI, EDO
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Crystal Structures Of Flap Bound To Dg-031
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2020-12-02 Classification: MEMBRANE PROTEIN Ligands: QY1, CA, BOG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-02
Ligands: QY1, CA, BOG
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Crystal Structures Of Flap Bound To Mk-866
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.61 Å Release Date: 2020-12-02 Classification: MEMBRANE PROTEIN Ligands: QY7, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-02
Ligands: QY7, SO4
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Crystal Structure Of Mpges-1 Bound To Dg-031
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2020-12-02 Classification: ISOMERASE, MEMBRANE PROTEIN Ligands: QY1, BOG, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-02
Ligands: QY1, BOG, PG4
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Crystal Structure Of Mpges-1 Bound To Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2017-03-01 Classification: MEMBRANE PROTEIN Ligands: 755, GSH, BOG, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-01
Ligands: 755, GSH, BOG, PG4
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Crystal Structure Of Mpges-1 Bound To Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.76 Å Release Date: 2017-03-01 Classification: MEMBRANE PROTEIN Ligands: 758, GSH, BOG, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-01
Ligands: 758, GSH, BOG, PG4
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Crystal Structure Of Mpges-1 Bound To Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.20 Å Release Date: 2017-03-01 Classification: Membrane Protein, Transferase Ligands: 7DN, GSH, JZR, BOG, PG4, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-03-01
Ligands: 7DN, GSH, JZR, BOG, PG4, PEG
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Mpges1 Bound To An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.30 Å Release Date: 2016-09-14 Classification: Isomerase/Isomerase Inhibitor Ligands: 6PW, GSH, BOG, PG4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-14
Ligands: 6PW, GSH, BOG, PG4
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Crystal Structure Of Autotaxin And Compound 1
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.41 Å Release Date: 2016-08-10 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 6ZM, ZN, CL |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2016-08-10
Ligands: NAG, 6ZM, ZN, CL
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Crystal Structure Of Autotaxin And Compound 1
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:3.06 Å Release Date: 2016-08-10 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: NAG, 6ZN, CL, ZN |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2016-08-10
Ligands: NAG, 6ZN, CL, ZN
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Crystal Structure Of Autotaxin And Compound Pf-8380
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION Resolution:2.73 Å Release Date: 2016-08-10 Classification: HYDROLASE/HYDROLASE inhibitor Ligands: ZN, CA, 6ZO, EPE, CL |
Organism: Rattus norvegicus
Method: X-RAY DIFFRACTION
Release Date: 2016-08-10
Ligands: ZN, CA, 6ZO, EPE, CL
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Crystal Structure Of The Rar Alpha Ligand-Binding Domain In Complex With An Antagonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2016-06-22 Classification: TRANSCRIPTION Ligands: 6Q7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-06-22
Ligands: 6Q7
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Crystal Structure Of Mpges-1 Bound To An Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.44 Å Release Date: 2016-04-13 Classification: Isomerase/Isomerase inhibitor Ligands: 4UJ, GSH, JZR, BOG, PGE, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-13
Ligands: 4UJ, GSH, JZR, BOG, PGE, PEG
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Discovery Of A Potent And Selective Mpges-1 Inhibitor For The Treatment Of Pain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2016-04-13 Classification: Isomerase/isomerase inhibitor Ligands: 4UK, GSH, BOG, PG4, 1KA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-13
Ligands: 4UK, GSH, BOG, PG4, 1KA
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Discovery Of A Potent And Selective Mpges-1 Inhibitor For The Treatment Of Pain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2016-04-13 Classification: Isomerase/isomerase inhibitor Ligands: 4UL, GSH, BOG, PG4, 1KA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-13
Ligands: 4UL, GSH, BOG, PG4, 1KA
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Estrogen Receptor Beta Ligand-Binding Domain Complexed To A Benzopyran Ligand
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.53 Å Release Date: 2007-10-30 Classification: transcription regulator Ligands: 3AS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-10-30
Ligands: 3AS
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Benzopyrans As Selective Estrogen Receptor B Agonists (Serbas). Part 2: Structure Activity Relationship Studies On The Benzopyran Scaffold.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2007-09-11 Classification: LIPID BINDING PROTEIN Ligands: WST |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-11
Ligands: WST
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Estrogen Receptor Alpha Ligand-Binding Domain In Complex With A Benzopyran Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2007-09-04 Classification: TRANSCRIPTION Ligands: JJ3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-09-04
Ligands: JJ3
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Estrogen Receptor Beta Ligand Binding Domain In Complex With A Benzopyran Agonist
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.28 Å Release Date: 2007-08-07 Classification: TRANSCRIPTION Ligands: JJ3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2007-08-07
Ligands: JJ3
