Search Count: 49
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Translation Initiation Factor Eif-2B Complex With The Isohexide Diamine Gsk735
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2026-03-04 Classification: TRANSLATION Ligands: PRO, SO4, EDO, A1C32 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-03-04
Ligands: PRO, SO4, EDO, A1C32
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Potent Long-Acting Inhibitors Targeting Hiv-1 Capsid Based On A Versatile Quinazolin-4-One Scaffold
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.56 Å Release Date: 2023-02-15 Classification: ANTIVIRAL-PROTEIN/INHIBITOR Ligands: EDO, Y05 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2023-02-15
Ligands: EDO, Y05
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Crystal Structure Of Prostaglandin D2 Synthase In Complex With Fragment 1A At 1.84A Resolution.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.84 Å Release Date: 2021-07-28 Classification: ISOMERASE Ligands: GSH, MG, QPN, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-07-28
Ligands: GSH, MG, QPN, GOL
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H-Pdgs Complexed With A 2-Phenylimidazo[1,2-A]Pyridine-6-Carboxamide Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2021-05-26 Classification: Isomerase, Transferase/Inhibitor Ligands: GSH, VH4, MG, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-26
Ligands: GSH, VH4, MG, NA
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H-Pdgs Complexed With A 2-Phenylimidazo[1,2-A]Pyridine-6-Carboxamide Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.13 Å Release Date: 2021-05-26 Classification: Isomerase, Transferase/Inhibitor Ligands: CL, EDO, GSH, VH7, MG, NA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-26
Ligands: CL, EDO, GSH, VH7, MG, NA
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Structure Of Hiv-1 Integrase With Potent 5,6,7,8-Tetrahydro-1,6-Naphthyridine Derivatives Allosteric Site Inhibitors
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2019-01-16 Classification: VIRAL PROTEIN Ligands: EDO, KJJ, SO4 |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2019-01-16
Ligands: EDO, KJJ, SO4
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Hiv Integrase Catalytic Domain Containing F185K Mutation Complexed With Gsk0002
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2016-12-14 Classification: TRANSFERASE/INHIBITOR Ligands: CAC, SO4, EDO, 65P |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-12-14
Ligands: CAC, SO4, EDO, 65P
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Hiv Integrase Catalytic Domain Containing F185K + A124T Mutations Complexed With Gsk0002
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2016-12-14 Classification: TRANSFERASE/INHIBITOR Ligands: CAC, SO4, EDO, 65P |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-12-14
Ligands: CAC, SO4, EDO, 65P
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Hiv Integrase Catalytic Domain Containing F185K + A124N + T125S Mutations Complexed With Gsk0002
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.88 Å Release Date: 2016-12-14 Classification: TRANSFERASE/INHIBITOR Ligands: CAC, SO4, EDO, 65P |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-12-14
Ligands: CAC, SO4, EDO, 65P
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Hiv Integrase Catalytic Domain Containing F185K + A124N + T125A Mutations Complexed With Gsk0002
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION Resolution:1.86 Å Release Date: 2016-12-14 Classification: TRANSFERASE/INHIBITOR Ligands: CAC, SO4, EDO, 65P |
Organism: Human immunodeficiency virus 1
Method: X-RAY DIFFRACTION
Release Date: 2016-12-14
Ligands: CAC, SO4, EDO, 65P
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Crystal Structure Of Unglycosylated Apo Human Furin @1.89A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2016-05-04 Classification: HYDROLASE Ligands: CA, PO4, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: CA, PO4, EDO
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The Structure Of Human Pde12 Residues 161-609
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2015-06-17 Classification: HYDROLASE Ligands: MG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-17
Ligands: MG, GOL
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The Structure Of Human Pde12 Residues 161-609 In Complex With Gsk3036342A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2015-06-17 Classification: Hydrolase/Hydrolase Inhibitor Ligands: SO4, EDO, TRS, 4LC, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-06-17
Ligands: SO4, EDO, TRS, 4LC, MG
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Crystal Structure Of The Hiv-1 Integrase Catalytic Domain With Gsk1264
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2014-06-11 Classification: VIRAL PROTEIN Ligands: 2SQ, CAC, SO4 |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: 2SQ, CAC, SO4
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X-Ray Structure Of Receptor Interacting Protein 1 (Rip1)Kinase Domain With A 1-Aminoisoquinoline Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2013-11-20 Classification: TRANSFERASE Ligands: MG, Q1A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-11-20
Ligands: MG, Q1A
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Hiv-1 Reverse Transcriptase Y188L Mutant In Complex With Inhibitor Gsk560
Organism: Hiv-1 m\:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.36 Å Release Date: 2013-01-09 Classification: HYDROLASE Ligands: MG, TAR, WHU |
Organism: Hiv-1 m\:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2013-01-09
Ligands: MG, TAR, WHU
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Hiv-1 Reverse Transcriptase In Complex With Inhibitor Gsk560
Organism: Hiv-1 m\:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2013-01-09 Classification: HYDROLASE Ligands: MG, SRT, WHU |
Organism: Hiv-1 m\:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2013-01-09
Ligands: MG, SRT, WHU
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Hiv-1 Reverse Transcriptase In Complex With Inhibitor Gsk500
Organism: Hiv-1 m\:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2013-01-09 Classification: HYDROLASE Ligands: TAR, EUR |
Organism: Hiv-1 m\:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2013-01-09
Ligands: TAR, EUR
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Hiv-1 Reverse Transcriptase In Complex With Inhibitor Gsk952
Organism: Hiv-1 m\:b_hxb2r
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2013-01-09 Classification: HYDROLASE Ligands: MG, TAR, CXD |
Organism: Hiv-1 m\:b_hxb2r
Method: X-RAY DIFFRACTION
Release Date: 2013-01-09
Ligands: MG, TAR, CXD
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Crystal Structure Of A Deletion Mutant Of Human Reverba Ligand Binding Domain Bound With An Ncor Id1 Peptide Determined To 2.60A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2010-06-30 Classification: Transcription regulator |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-06-30
