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Search Count: 51

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29MJ image
Akt1 Mutant In Complex With Miransertib (Arq 092)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.50 Å Release Date: 2026-07-01
Classification: TRANSFERASE
Ligands: 6S1, EDO, GOL

9GHR image
Crystal Structure Of Egfr-Wt In Complex With Covalent Compound 10N

9GHS image
Crystal Structure Of Egfr-Wt In Complex With Covalent Compound 10A

9GHT image
Crystal Structure Of Egfr-Wt In Complex With Bi-4020
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.60 Å Release Date: 2026-03-04
Classification: TRANSFERASE
Ligands: XA4

9GHU image
Crystal Structure Of Egfr-Wt In Complex With Covalent Compound 10F

9GHV image
Crystal Structure Of Egfr-Wt In Complex With Covalent Compound 13

9I7Y image
Crystal Structure Of Krasg13C In Complex With Nucleotide-Based Covalent Inhibitor 7B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2025-11-12
Classification: HYDROLASE
Ligands: A1I08, MG

8S13 image
Apo C-Kit-Wt Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: EDO

8S14 image
C-Kit Kinase Domain In Complex With Sunitinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.50 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: B49, EDO, CL

8S15 image
C-Kit Kinase Domain In Complex With Nintedanib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.40 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: XIN

8S16 image
C-Kit Kinase Domain In Complex With Imatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: STI, CL

8S17 image
C-Kit Kinase Domain In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: 0LI, CL

8S18 image
C-Kit Kinase Domain In Complex With S116836

8S19 image
C-Kit Kinase Domain In Complex With Staurosporine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: STU

8S1A image
C-Kit Kinase Domain In Complex With Crenolanib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: 6T2

8S1B image
C-Kit Kinase Domain In Complex With Idrx-42 Via Soaking
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.00 Å Release Date: 2025-09-03
Classification: TRANSFERASE
Ligands: K3R, CL

9HXV image
Crystal Structure Of Tet2-Dna In Complex With Iox1

8PQ9 image
C-Kit Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.70 Å Release Date: 2023-12-27
Classification: TRANSFERASE
Ligands: 9JI, SO4

8PQA image
C-Kit Kinase Domain In Complex With Avapritinib Derivative 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.65 Å Release Date: 2023-12-27
Classification: TRANSFERASE
Ligands: 98A

8PQB image
C-Kit Kinase Domain In Complex With Avapritinib Derivative 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.87 Å Release Date: 2023-12-27
Classification: TRANSFERASE
Ligands: 9XO
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