Search Count: 51
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Akt1 Mutant In Complex With Miransertib (Arq 092)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2026-07-01 Classification: TRANSFERASE Ligands: 6S1, EDO, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-01
Ligands: 6S1, EDO, GOL
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Crystal Structure Of Egfr-Wt In Complex With Covalent Compound 10N
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2026-03-04 Classification: TRANSFERASE Ligands: A1ILN, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-03-04
Ligands: A1ILN, MES
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Crystal Structure Of Egfr-Wt In Complex With Covalent Compound 10A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2026-03-04 Classification: TRANSFERASE Ligands: A1ILJ, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-03-04
Ligands: A1ILJ, MES
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Crystal Structure Of Egfr-Wt In Complex With Bi-4020
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2026-03-04 Classification: TRANSFERASE Ligands: XA4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-03-04
Ligands: XA4
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Crystal Structure Of Egfr-Wt In Complex With Covalent Compound 10F
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2026-03-04 Classification: TRANSFERASE Ligands: A1ILK, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-03-04
Ligands: A1ILK, MES
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Crystal Structure Of Egfr-Wt In Complex With Covalent Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2026-03-04 Classification: TRANSFERASE Ligands: A1ILI, MES |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-03-04
Ligands: A1ILI, MES
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Crystal Structure Of Krasg13C In Complex With Nucleotide-Based Covalent Inhibitor 7B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2025-11-12 Classification: HYDROLASE Ligands: A1I08, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: A1I08, MG
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Apo C-Kit-Wt Kinase Domain
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: EDO
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C-Kit Kinase Domain In Complex With Sunitinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: B49, EDO, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: B49, EDO, CL
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C-Kit Kinase Domain In Complex With Nintedanib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: XIN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: XIN
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C-Kit Kinase Domain In Complex With Imatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: STI, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: STI, CL
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C-Kit Kinase Domain In Complex With Ponatinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: 0LI, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: 0LI, CL
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C-Kit Kinase Domain In Complex With S116836
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: A1H4U, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: A1H4U, CL
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C-Kit Kinase Domain In Complex With Staurosporine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: STU |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: STU
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C-Kit Kinase Domain In Complex With Crenolanib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: 6T2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: 6T2
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C-Kit Kinase Domain In Complex With Idrx-42 Via Soaking
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2025-09-03 Classification: TRANSFERASE Ligands: K3R, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-09-03
Ligands: K3R, CL
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Crystal Structure Of Tet2-Dna In Complex With Iox1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2025-04-09 Classification: OXIDOREDUCTASE Ligands: FE2, ZN, 8XQ, SO4, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-09
Ligands: FE2, ZN, 8XQ, SO4, CL
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C-Kit Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9JI, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9JI, SO4
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 98A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 98A
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 8
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9XO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9XO
