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Search Count: 44

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7ZVS image
Crystal Structure Of The Schistosoma Mansoni Vkr2 Kinase Domain In An Active-Like State (Adp-Bound)

7AFZ image
L1 Metallo-B-Lactamase With Compound Ebl-1306

6YOJ image
Focal Adhesion Kinase Catalytic Domain In Complex With 6-[4-(3-Methanesulfonyl-Benzylamino)-5-Trifluoromethyl-Pyrimidin-2-Ylamino]-3,4-Dihydro-1H-Quinolin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.36 Å Release Date: 2021-02-10
Classification: TRANSFERASE
Ligands: P4N

6YQ1 image
Focal Adhesion Kinase Catalytic Domain In Complex With N-Methyl-N-(3-{[2-(2-Oxo-1,2,3,4-Tetrahydro-Quinolin-6-Ylamino)-5-Trifluoromethyl-Pyrimidin-4-Ylamino]-Methyl}-Pyridin-2-Yl)-Methanesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.78 Å Release Date: 2021-02-10
Classification: TRANSFERASE
Ligands: P7N, NA, SO4

6YR9 image
Focal Adhesion Kinase Catalytic Domain In Complex With N-Methyl-N-(2-{[2-(2-Oxo-2,3-Dihydro-1H-Indol-5-Ylamino)-5-Trifluoromethyl-Pyrimidin-4-Ylamino]-Methyl}-Phenyl)-Methanesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.93 Å Release Date: 2021-02-10
Classification: TRANSFERASE
Ligands: P9K

6YT6 image
Focal Adhesion Kinase Catalytic Domain In Complex With N-Methyl-N-(3-{[2-(2-Oxo-2,3-Dihydro-1H-Indol-5-Ylamino)-Pyrimidin-4-Ylamino]-Methyl}-Pyridin-2-Yl)-Methanesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.54 Å Release Date: 2021-02-10
Classification: TRANSFERASE
Ligands: PKE, SO4

6YVS image
Focal Adhesion Kinase Catalytic Domain In Complex With 5-{4-[(Pyridin-3-Ylmethyl)-Amino]-5-Trifluoromethyl-Pyrimidin-2-Ylamino}-1,3-Dihydro-Indol-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.81 Å Release Date: 2021-02-10
Classification: TRANSFERASE
Ligands: PVT, SO4

6YVY image
Focal Adhesion Kinase Catalytic Domain In Complex With 4-{[4-{[(1R,2R)-2-(Dimethylamino)Cyclopentyl]Amino}-5-(Trifluoromethyl)Pyrimidin-2-Yl]Amino}-N-Methylbenzenesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.92 Å Release Date: 2021-02-10
Classification: TRANSFERASE
Ligands: P1E, SO4

6YXV image
Focal Adhesion Kinase Catalytic Domain In Complex With N-Methyl-N-{3-[(2-Phenylamino-5-Trifluoromethyl-Pyrimidin-4-Ylamino)-Methyl]-Pyridin-2-Yl}-Methanesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2021-02-10
Classification: TRANSFERASE
Ligands: Q2H, SO4

6S1I image
Crystal Structure Of Dyrk1A With Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.38 Å Release Date: 2019-06-26
Classification: TRANSFERASE
Ligands: SO4, PG4, KR8

6I30 image
Crystal Structure Of The Ampc From Pseudomonas Aeruginosa With 1C

5O48 image
P.Vivax Nmt With An Aminomethylindazole Inhibitor Bound

5O4V image
P.Vivax Nmt With Aminomethylindazole And Quinoline Inhibitors Bound

5O6H image
Human Nmt1 In Complex With Myristoyl-Coa And Inhibitor Imp-917
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.29 Å Release Date: 2018-05-16
Classification: TRANSFERASE
Ligands: MYA, PO4, 9M2, MG, GOL, DMS

5O6J image
Human Nmt1 In Complex With Myristoyl-Coa And Inhibitor Imp-1031
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.45 Å Release Date: 2018-05-16
Classification: TRANSFERASE
Ligands: MYA, PO4, MG, 9M8

5OXD image
Complex Of A C. Perfringens O-Glcnacase With A Fragment Hit

5O9O image
Crystal Structure Of Scgas2 In Complex With Compound 7.

5O9P image
Crystal Structure Of Gas2 In Complex With Compound 10

5O9Q image
Crystal Structure Of Scgas2 In Complex With Compound 6

5O9R image
Crystal Structure Of Scgas2 In Complex With Compound 9
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