Search Count: 44
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Crystal Structure Of The Schistosoma Mansoni Vkr2 Kinase Domain In An Active-Like State (Adp-Bound)
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION Resolution:3.07 Å Release Date: 2022-10-12 Classification: TRANSFERASE Ligands: ADP |
Organism: Schistosoma mansoni
Method: X-RAY DIFFRACTION
Release Date: 2022-10-12
Ligands: ADP
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L1 Metallo-B-Lactamase With Compound Ebl-1306
Organism: Stenotrophomonas maltophilia
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2021-10-06 Classification: ANTIMICROBIAL PROTEIN Ligands: ZN, RBW, SO4 |
Organism: Stenotrophomonas maltophilia
Method: X-RAY DIFFRACTION
Release Date: 2021-10-06
Ligands: ZN, RBW, SO4
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Focal Adhesion Kinase Catalytic Domain In Complex With 6-[4-(3-Methanesulfonyl-Benzylamino)-5-Trifluoromethyl-Pyrimidin-2-Ylamino]-3,4-Dihydro-1H-Quinolin-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.36 Å Release Date: 2021-02-10 Classification: TRANSFERASE Ligands: P4N |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: P4N
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Focal Adhesion Kinase Catalytic Domain In Complex With N-Methyl-N-(3-{[2-(2-Oxo-1,2,3,4-Tetrahydro-Quinolin-6-Ylamino)-5-Trifluoromethyl-Pyrimidin-4-Ylamino]-Methyl}-Pyridin-2-Yl)-Methanesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2021-02-10 Classification: TRANSFERASE Ligands: P7N, NA, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: P7N, NA, SO4
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Focal Adhesion Kinase Catalytic Domain In Complex With N-Methyl-N-(2-{[2-(2-Oxo-2,3-Dihydro-1H-Indol-5-Ylamino)-5-Trifluoromethyl-Pyrimidin-4-Ylamino]-Methyl}-Phenyl)-Methanesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2021-02-10 Classification: TRANSFERASE Ligands: P9K |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: P9K
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Focal Adhesion Kinase Catalytic Domain In Complex With N-Methyl-N-(3-{[2-(2-Oxo-2,3-Dihydro-1H-Indol-5-Ylamino)-Pyrimidin-4-Ylamino]-Methyl}-Pyridin-2-Yl)-Methanesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2021-02-10 Classification: TRANSFERASE Ligands: PKE, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: PKE, SO4
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Focal Adhesion Kinase Catalytic Domain In Complex With 5-{4-[(Pyridin-3-Ylmethyl)-Amino]-5-Trifluoromethyl-Pyrimidin-2-Ylamino}-1,3-Dihydro-Indol-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.81 Å Release Date: 2021-02-10 Classification: TRANSFERASE Ligands: PVT, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: PVT, SO4
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Focal Adhesion Kinase Catalytic Domain In Complex With 4-{[4-{[(1R,2R)-2-(Dimethylamino)Cyclopentyl]Amino}-5-(Trifluoromethyl)Pyrimidin-2-Yl]Amino}-N-Methylbenzenesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2021-02-10 Classification: TRANSFERASE Ligands: P1E, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: P1E, SO4
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Focal Adhesion Kinase Catalytic Domain In Complex With N-Methyl-N-{3-[(2-Phenylamino-5-Trifluoromethyl-Pyrimidin-4-Ylamino)-Methyl]-Pyridin-2-Yl}-Methanesulfonamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2021-02-10 Classification: TRANSFERASE Ligands: Q2H, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-10
Ligands: Q2H, SO4
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Crystal Structure Of Dyrk1A With Small Molecule Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.38 Å Release Date: 2019-06-26 Classification: TRANSFERASE Ligands: SO4, PG4, KR8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-06-26
Ligands: SO4, PG4, KR8
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Crystal Structure Of The Ampc From Pseudomonas Aeruginosa With 1C
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION Resolution:2.21 Å Release Date: 2019-02-20 Classification: HYDROLASE Ligands: C6S |
Organism: Pseudomonas aeruginosa
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: C6S
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P.Vivax Nmt With An Aminomethylindazole Inhibitor Bound
Organism: Plasmodium vivax
Method: X-RAY DIFFRACTION Resolution:1.69 Å Release Date: 2018-05-16 Classification: TRANSFERASE Ligands: NHW, 9K2, DMS, MG, CL, SO4 |
Organism: Plasmodium vivax
Method: X-RAY DIFFRACTION
Release Date: 2018-05-16
Ligands: NHW, 9K2, DMS, MG, CL, SO4
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P.Vivax Nmt With Aminomethylindazole And Quinoline Inhibitors Bound
Organism: Plasmodium vivax
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2018-05-16 Classification: TRANSFERASE Ligands: NHW, 9K2, DMS, MG, CL, SO4, 9KZ |
Organism: Plasmodium vivax
Method: X-RAY DIFFRACTION
Release Date: 2018-05-16
Ligands: NHW, 9K2, DMS, MG, CL, SO4, 9KZ
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Human Nmt1 In Complex With Myristoyl-Coa And Inhibitor Imp-917
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.29 Å Release Date: 2018-05-16 Classification: TRANSFERASE Ligands: MYA, PO4, 9M2, MG, GOL, DMS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-16
Ligands: MYA, PO4, 9M2, MG, GOL, DMS
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Human Nmt1 In Complex With Myristoyl-Coa And Inhibitor Imp-1031
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2018-05-16 Classification: TRANSFERASE Ligands: MYA, PO4, MG, 9M8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-16
Ligands: MYA, PO4, MG, 9M8
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Complex Of A C. Perfringens O-Glcnacase With A Fragment Hit
Organism: Clostridium perfringens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2018-05-16 Classification: HYDROLASE Ligands: CD, B2W |
Organism: Clostridium perfringens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-16
Ligands: CD, B2W
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Crystal Structure Of Scgas2 In Complex With Compound 7.
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2018-05-02 Classification: TRANSFERASE Ligands: 9PB, EDO |
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: 9PB, EDO
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Crystal Structure Of Gas2 In Complex With Compound 10
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2018-05-02 Classification: TRANSFERASE Ligands: 9P8, EDO |
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: 9P8, EDO
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Crystal Structure Of Scgas2 In Complex With Compound 6
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2018-05-02 Classification: TRANSFERASE Ligands: 9PH |
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: 9PH
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Crystal Structure Of Scgas2 In Complex With Compound 9
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2018-05-02 Classification: TRANSFERASE Ligands: 9PK, EDO, SO4 |
Organism: Saccharomyces cerevisiae s288c
Method: X-RAY DIFFRACTION
Release Date: 2018-05-02
Ligands: 9PK, EDO, SO4
