Search Count: 15
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Phosphoinositide 3-Kinase Gamma Bound To An Pyrrolopyridinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.31 Å Release Date: 2018-06-27 Classification: Transferase/Transferase Inhibitor Ligands: EFV, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-06-27
Ligands: EFV, SO4
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Crystal Structure Of Rock1 Bound To An Aminopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2018-03-07 Classification: Transferase/Transferase Inhibitor Ligands: 8UV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 8UV
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Crystal Structure Of Pka Bound To An Pyrrolo Pyridine Inhibitor
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2018-03-07 Classification: Transferase/Transferase Inhibitor Ligands: 504 |
Organism: Homo sapiens, Oryctolagus cuniculus
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: 504
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Rock 1 Bound To Azaindole Thiazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6U1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 6U1
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Rock 1 Bound To Azaindole Thiazole Piperazine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2017-06-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 6U2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-06-28
Ligands: 6U2
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The X-Ray Structure Of Jcv Helicase
Organism: Jc polyomavirus
Method: X-RAY DIFFRACTION Resolution:2.17 Å Release Date: 2016-07-20 Classification: HYDROLASE/INHIBITOR Ligands: ZN, MES, SO4 |
Organism: Jc polyomavirus
Method: X-RAY DIFFRACTION
Release Date: 2016-07-20
Ligands: ZN, MES, SO4
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The X-Ray Structure Of Inhibitor Bound To Jcv Helicase
Organism: Jc polyomavirus
Method: X-RAY DIFFRACTION Resolution:1.99 Å Release Date: 2016-07-20 Classification: HYDROLASE/INHIBITOR Ligands: ZN, MES, 6JJ |
Organism: Jc polyomavirus
Method: X-RAY DIFFRACTION
Release Date: 2016-07-20
Ligands: ZN, MES, 6JJ
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The Crystal Structure Of Inhibitor Bound To Jcv Helicase
Organism: Jc polyomavirus
Method: X-RAY DIFFRACTION Resolution:2.94 Å Release Date: 2016-07-20 Classification: HYDROLASE/INHIBITOR Ligands: ZN, MES, SO4, 6JH |
Organism: Jc polyomavirus
Method: X-RAY DIFFRACTION
Release Date: 2016-07-20
Ligands: ZN, MES, SO4, 6JH
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The Crystal Structure Of N-(4-(2-(Thiazolo[5,4-C]Pyridin-2-Yl)Phenoxy)Phenyl)Acetamide Bound To Jcv Helicase
Organism: Jc polyomavirus
Method: X-RAY DIFFRACTION Resolution:2.59 Å Release Date: 2016-07-20 Classification: HYDROLASE/INHIBITOR Ligands: ZN, MES, SO4, 6JG |
Organism: Jc polyomavirus
Method: X-RAY DIFFRACTION
Release Date: 2016-07-20
Ligands: ZN, MES, SO4, 6JG
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Crystal Structure Of Gsk3B In Complex With A Pyrimidylpyrrole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2010-01-12 Classification: TRANSFERASE Ligands: Z48 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-01-12
Ligands: Z48
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Crystal Structure Of Erk2 Bound To (S)-N-(2-Hydroxy-1-Phenylethyl)-4-(5-Methyl-2-(Phenylamino)Pyrimidin-4-Yl)-1H-Pyrrole-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2010-01-12 Classification: TRANSFERASE Ligands: SO4, Z48 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-01-12
Ligands: SO4, Z48
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Crystal Structure Of Erk2 Bound To (S)-4-(2-(2-Chlorophenylamino)-5-Methylpyrimidin-4-Yl)-N-(2-Hydroxy-1-Phenylethyl)-1H-Pyrrole-2-Carboxamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-01-12 Classification: TRANSFERASE Ligands: SO4, E86 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-01-12
Ligands: SO4, E86
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2-Aminopyrazolo[1,5-A]Pyrimidines As Potent And Selective Inhibitors Of Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: 1P5 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-10
Ligands: 1P5
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2-Aminopyrazolo[1,5-A]Pyrimidines As Potent And Selective Inhibitors Of Jak2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2009-11-10 Classification: TRANSFERASE Ligands: 1P6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2009-11-10
Ligands: 1P6
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Discovery And Sar Of Novel 4-Thiazolyl-2-Phenylaminopyrimidines As Potent Inhibitors Of Spleen Tyrosine Kinase (Syk)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2008-12-02 Classification: TRANSFERASE Ligands: 685 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-12-02
Ligands: 685
