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11GY image
Crystal Structure Of Selective Inhibitor 16 Bound At The Active Site Of Cdk1

10YS image
Structure Of Cbl-B Bound To Compound 33
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2026-07-01
Classification: LIGASE
Ligands: GOL, IOD, EDO, MG, ZN, A1DCD, DMS

10ZF image
Structure Of C-Cbl Bound To Compound 33

9Y9B image
Plk4 In Complex With Compound 6 (3-Hydroxy-N-(3-(Pyridin-2-Yl)-1H-Pyrazol-4-Yl)-8-Azabicyclo[3.2.1]Octane-8-Carboxamide)

9Y9N image
Plk4 In Complex With Compound 25 ((R)-7-Hydroxy-N-(3-(1-(2,2,2-Trifluoroethyl)-1H-Pyrazolo[4,3-C]Pyridin-6-Yl)-1H-Pyrazol-4-Yl)-7-(Trifluoromethyl)-4-Azaspiro[2.5]Octane-4-Carboxamide)

8ERD image
Cyclin-Free Cdk2 In Complex With Cpd17
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.33 Å Release Date: 2023-10-18
Classification: TRANSFERASE
Ligands: WQ6

8ERN image
Cyclin-Free Cdk2 In Complex With Cpd21
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.64 Å Release Date: 2023-10-18
Classification: TRANSFERASE
Ligands: GOL, WQK

7SIY image
Ccbl Tkb Domain In Complex With Pzap70 Peptide

7QCD image
Cryoem Structure Of The Smc5/6-Holocomplex (Composite Structure)

7KHH image
Ternary Complex Of Vhl/Brd4-Bd1/Compound9 (4-(3,5-Difluoropyridin-2-Yl)-N-(11-(((S)-1-((2S,4R)-4-Hydroxy-2-((4-(4-Methylthiazol-5-Yl)Benzyl)Carbamoyl)Pyrrolidin-1-Yl)-3,3-Dimethyl-1-Oxobutan-2-Yl)Amino)-11-Oxoundecyl)-10-Methyl-7-((Methylsulfonyl)Methyl)-11-Oxo-3,4,10,11-Tetrahydro-1H-1,4,10-Triazadibenzo[Cd,F]Azulene-6-Carboxamide)

7KHL image
Brd4-Bd1 Compound6 (Methyl 4-(3,5-Difluoropyridin-2-Yl)-10-Methyl-7-((Methylsulfonyl)Methyl)-11-Oxo-3,4,10,11-Tetrahydro-1H-1,4,10-Triazadibenzo[Cd,F]Azulene-6-Carboxylate)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.29 Å Release Date: 2021-02-24
Classification: CELL CYCLE
Ligands: WEM, GOL

6NO8 image
Pim1 In Complex With Cpd9 ((R)-5-Amino-N-(3-(4-Aminoazepan-1-Yl)-1H-Pyrazol-4-Yl)-2-(2,6-Difluorophenyl)Thiazole-4-Carboxamide)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.38 Å Release Date: 2019-11-27
Classification: TRANSFERASE
Ligands: KUY, PO4

6ALB image
Crebbp Bromodomain In Complex With Cpd 30 (1-(3-(3-(1-Methyl-1H-Pyrazol-4-Yl)Isoquinolin-8-Yl)-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridin-5-Yl)Ethan-1-One)

5VZS image
Brd4-Bd1 In Complex With Cpd19 (3-(7-(Difluoromethyl)-6-(1-Methyl-1H-Pyrazol-4-Yl)-3,4-Dihydroquinolin-1(2H)-Yl)-N-Methyl-1-(Tetrahydro-2H-Pyran-4-Yl)-1,4,6,7-Tetrahydro-5H-Pyrazolo[4,3-C]Pyridine-5-Carboxamide)

5WHC image
Usp7 In Complex With Cpd2 (4-(3-(1-Methylpiperidin-4-Yl)-1,2,4-Oxadiazol-5-Yl)Phenol)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.55 Å Release Date: 2017-12-13
Classification: HYDROLASE
Ligands: AJJ, GOL

6AUD image
Pi3K-Gamma K802T In Complex With Cpd 8 10-((1-(Tert-Butyl)Piperidin-4-Yl)Sulfinyl)-2-(1-Isopropyl-1H-1,2,4-Triazol-5-Yl)-5,6-Dihydrobenzo[F]Imidazo[1,2-D][1,4]Oxazepine

6B4A image
Crystal Structure Of The C-Terminal Domain Of Doublecortin (Tgdcx) From Toxoplasma Gondii Me49

5VRG image
Structural Insights Into Lipoprotein N-Acylation By Escherichia Coli Apolipoprotein N-Acyltransferase

5VRH image
Apolipoprotein N-Acyltransferase C387S Active Site Mutant

5MG8 image
Crystal Structure Of The S.Pombe Smc5/6 Hinge Domain
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