Structural Entry Filters:

Search Count: 102

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9TF9 image
Pdgfra-G680R Mutant Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.20 Å Release Date: 2026-07-15
Classification: TRANSFERASE
Ligands: 9JI

9TFA image
Pdgfra-G680R Mutant Kinase Domain In Complex With A 6,7-Dimethoxyquinazoline-Based Compound (43)

9TFB image
Pdgfra-G680R Mutant Kinase Domain In Complex With A 6,7-Bis(2-Methoxyethoxy)Quinazoline-Based Compound (44)

9TFC image
Pdgfra-G680R Mutant Kinase Domain In Complex With A 7-Methoxyquinazolin-6-Ol-Based Compound (45)

9TFD image
Kit Kinase Domain In Complex With A Pyrrolotriazine-Based Compound (11)

9TFE image
Kit Kinase Domain In Complex With An Aminopyrimidine-Based Compound (15)

9TFF image
Kit Kinase Domain In Complex With A Pyrrolopyrimidine-Based Compound (17)

9TFG image
Kit Kinase Domain In Complex With A 6-,7-Dimethoxyquinoline-Based Compound (19)

9TFH image
Kit Kinase Domain In Complex With A 7-Methylquinazoline-Based Compound (25)

9TFI image
Kit Kinase Domain In Complex With A 6,7-Bis(2-Methoxyethoxy)Quinazoline-Based Compound (33)

9TFJ image
Kit Kinase Domain In Complex With A 6,7-Dimethoxyquinazoline-Based Compound (34)

9TFK image
Kit Kinase Domain In Complex With A Quinoline-3-Carbonitrile-Based Compound (38)

9TFL image
Kit Kinase Domain In Complex With A Methyl Quinazoline-7-Carboxylate-Based Compound (41)

9TFM image
Kit Kinase Domain In Complex With A 7-Methoxyquinazolin-6-Ol-Based Compound (45)

9I7Y image
Crystal Structure Of Krasg13C In Complex With Nucleotide-Based Covalent Inhibitor 7B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2025-11-12
Classification: HYDROLASE
Ligands: A1I08, MG

9HZ0 image
Protein Kinase Mkk7 In Complex With K221 Targeting Compound 1

9HXV image
Crystal Structure Of Tet2-Dna In Complex With Iox1

9GZH image
Pdgfra-T674I In Complex With Covalent Ponatinib Derivative 19

8PQ9 image
C-Kit Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.70 Å Release Date: 2023-12-27
Classification: TRANSFERASE
Ligands: 9JI, SO4

8PQA image
C-Kit Kinase Domain In Complex With Avapritinib Derivative 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.65 Å Release Date: 2023-12-27
Classification: TRANSFERASE
Ligands: 98A
Protein Functional Filters:
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