Search Count: 102
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Pdgfra-G680R Mutant Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: 9JI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: 9JI
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Pdgfra-G680R Mutant Kinase Domain In Complex With A 6,7-Dimethoxyquinazoline-Based Compound (43)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVO
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Pdgfra-G680R Mutant Kinase Domain In Complex With A 6,7-Bis(2-Methoxyethoxy)Quinazoline-Based Compound (44)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVS
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Pdgfra-G680R Mutant Kinase Domain In Complex With A 7-Methoxyquinazolin-6-Ol-Based Compound (45)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVR
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Kit Kinase Domain In Complex With A Pyrrolotriazine-Based Compound (11)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVQ
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Kit Kinase Domain In Complex With An Aminopyrimidine-Based Compound (15)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JV1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JV1
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Kit Kinase Domain In Complex With A Pyrrolopyrimidine-Based Compound (17)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVP
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Kit Kinase Domain In Complex With A 6-,7-Dimethoxyquinoline-Based Compound (19)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVT
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Kit Kinase Domain In Complex With A 7-Methylquinazoline-Based Compound (25)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVW |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVW
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Kit Kinase Domain In Complex With A 6,7-Bis(2-Methoxyethoxy)Quinazoline-Based Compound (33)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVV
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Kit Kinase Domain In Complex With A 6,7-Dimethoxyquinazoline-Based Compound (34)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVZ
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Kit Kinase Domain In Complex With A Quinoline-3-Carbonitrile-Based Compound (38)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVY
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Kit Kinase Domain In Complex With A Methyl Quinazoline-7-Carboxylate-Based Compound (41)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JV0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JV0
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Kit Kinase Domain In Complex With A 7-Methoxyquinazolin-6-Ol-Based Compound (45)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVR
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Crystal Structure Of Krasg13C In Complex With Nucleotide-Based Covalent Inhibitor 7B
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2025-11-12 Classification: HYDROLASE Ligands: A1I08, MG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-11-12
Ligands: A1I08, MG
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Protein Kinase Mkk7 In Complex With K221 Targeting Compound 1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2025-06-04 Classification: TRANSFERASE Ligands: A1IY7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-06-04
Ligands: A1IY7
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Crystal Structure Of Tet2-Dna In Complex With Iox1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2025-04-09 Classification: OXIDOREDUCTASE Ligands: FE2, ZN, 8XQ, SO4, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-04-09
Ligands: FE2, ZN, 8XQ, SO4, CL
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Pdgfra-T674I In Complex With Covalent Ponatinib Derivative 19
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2025-02-12 Classification: TRANSFERASE Ligands: A1IRC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2025-02-12
Ligands: A1IRC
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C-Kit Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 9JI, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 9JI, SO4
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C-Kit Kinase Domain In Complex With Avapritinib Derivative 4
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2023-12-27 Classification: TRANSFERASE Ligands: 98A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-12-27
Ligands: 98A
