Search Count: 291
![]() |
Akt1 Mutant In Complex With The 3,5-Dimethyl 1,4-Substituted Pyrazole Containing Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2026-09-16 Classification: TRANSFERASE Ligands: A1JWV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-09-16
Ligands: A1JWV
![]() |
Akt1 Mutant In Complex With The Trimethyl 1,4-Substituted Pyrazole Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2026-09-16 Classification: TRANSFERASE Ligands: A1JW3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-09-16
Ligands: A1JW3
![]() |
Akt1 Mutant In Complex With The 3-Ethyl 1-Methyl 1,4-Substituted Pyrazole Containing Compound And Eg
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2026-09-16 Classification: TRANSFERASE Ligands: EDO, A1JWX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-09-16
Ligands: EDO, A1JWX
![]() |
Akt1 Mutant In Complex With The 3-Ethyl 1-Methyl 1,4-Substituted Pyrazole Containing Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2026-09-16 Classification: TRANSFERASE Ligands: A1JWX |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-09-16
Ligands: A1JWX
![]() |
Akt1 Mutant In Complex With The 1-Ethyl 1,5-Substituted Pyrazole Containing Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2026-09-16 Classification: TRANSFERASE Ligands: A1JW0 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-09-16
Ligands: A1JW0
![]() |
Akt1 Mutant In Complex With The 1-Isopropyl 1,5-Substituted Pyrazole Containing Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2026-09-16 Classification: TRANSFERASE Ligands: A1JW2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-09-16
Ligands: A1JW2
![]() |
Akt1 Mutant In Complex With The 1-Propyl 1,5-Substituted Pyrazole Containing Compound And Eg
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2026-09-16 Classification: TRANSFERASE Ligands: A1JW1, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-09-16
Ligands: A1JW1, EDO
![]() |
Akt1 Mutant In Complex With 2-Methyl Pyridine Containing Compound And Eg
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2026-09-16 Classification: TRANSFERASE Ligands: EDO, A1JWY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-09-16
Ligands: EDO, A1JWY
![]() |
Akt1 Mutant In Complex With The 1-Cyclobutyl 1,5-Substituted Pyrazole Containing Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2026-09-16 Classification: TRANSFERASE Ligands: A1JWZ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-09-16
Ligands: A1JWZ
![]() |
Akt1 Mutant In Complex With 2-Methyl Pyridine Containing Compound
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2026-09-16 Classification: TRANSFERASE Ligands: A1JWY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-09-16
Ligands: A1JWY
![]() |
Akt1 Mutant In Complex With 2-Amino, 6-Methyl Pyridine Containing Compound And Eg
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2026-09-16 Classification: TRANSFERASE Ligands: A1JWW, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-09-16
Ligands: A1JWW, EDO
![]() |
Azetidine-1- Carboxylic Acid Synthase Azej From Saccharotrix Sp. Nrrl B-16348
Organism: Saccharothrix sp. nrrl b-16348
Method: X-RAY DIFFRACTION Resolution:2.67 Å Release Date: 2026-08-05 Classification: LYASE |
Organism: Saccharothrix sp. nrrl b-16348
Method: X-RAY DIFFRACTION
Release Date: 2026-08-05
![]() |
Pdgfra-G680R Mutant Kinase Domain In Complex With Avapritinib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: 9JI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: 9JI
![]() |
Pdgfra-G680R Mutant Kinase Domain In Complex With A 6,7-Dimethoxyquinazoline-Based Compound (43)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVO
![]() |
Pdgfra-G680R Mutant Kinase Domain In Complex With A 6,7-Bis(2-Methoxyethoxy)Quinazoline-Based Compound (44)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVS
![]() |
Pdgfra-G680R Mutant Kinase Domain In Complex With A 7-Methoxyquinazolin-6-Ol-Based Compound (45)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVR |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVR
![]() |
Kit Kinase Domain In Complex With A Pyrrolotriazine-Based Compound (11)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVQ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVQ
![]() |
Kit Kinase Domain In Complex With An Aminopyrimidine-Based Compound (15)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JV1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JV1
![]() |
Kit Kinase Domain In Complex With A Pyrrolopyrimidine-Based Compound (17)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVP |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVP
![]() |
Kit Kinase Domain In Complex With A 6-,7-Dimethoxyquinoline-Based Compound (19)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2026-07-15 Classification: TRANSFERASE Ligands: A1JVT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-07-15
Ligands: A1JVT
