Search Count: 17
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E. Coli Fabh With Small Molecule Inhibitor 1
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:1.70 Å Release Date: 2016-05-18 Classification: Transferase/Transferase Inhibitor Ligands: SO4, 4VK, PG4 |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: SO4, 4VK, PG4
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E. Coli Fabh With Small Molecule Inhibitor 2
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:1.89 Å Release Date: 2016-05-18 Classification: Transferase/Transferase Inhibitor Ligands: 4VL |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: 4VL
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E. Coli Fabh With Small Molecule Inhibitor 2
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2016-05-18 Classification: Transferase/Transferase Inhibitor Ligands: 4VM |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
Ligands: 4VM
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S. Pneumoniae Fabh With Small Molecule Inhibitor 4
Organism: Streptococcus pneumoniae
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2016-05-18 Classification: Transferase/Transferase Inhibitor |
Organism: Streptococcus pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2016-05-18
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Antibacterial Fabh Inhibitors With Validated Mode Of Action In Haemophilus Influenzae By In Vitro Resistance Mutation Mapping
Organism: Escherichia coli o157:h7
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2016-05-04 Classification: Transferase/Transferase inhibitor Ligands: 4LB, SO4 |
Organism: Escherichia coli o157:h7
Method: X-RAY DIFFRACTION
Release Date: 2016-05-04
Ligands: 4LB, SO4
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S.Aureus Tmk In Complex With A Potent Inhibitor Compound 18, 2-(3-Chlorophenoxy)-3-Methoxy-4-{[(3S)-3-(5-Methyl-2,4-Dioxo-3,4-Dihydropyrimidin-1(2H)-Yl)Piperidin-1-Yl]Methyl}Benzoic Acid
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:1.67 Å Release Date: 2014-06-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 32K |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: 32K
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S.Aureus Tmk In Complex With Potent Inhibitor Compound 19, 2-(3-Chlorophenoxy)-3-Fluoro-4-{[(3S)-3-(5-Methyl-2,4-Dioxo-3,4-Dihydropyrimidin-1(2H)-Yl)Piperidin-1-Yl]Methyl}Benzoic Acid
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:1.94 Å Release Date: 2014-06-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 31Z |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: 31Z
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S.Aureus Tmk In Complex With The Potent Inhibitor Compound 38, 2-(3-Chlorophenoxy)-3-Methoxy-4-{(1R)-1-[(3S)-3-(5-Methyl-2,4-Dioxo-3,4-Dihydropyrimidin-1(2H)-Yl)Piperidin-1-Yl]Propyl}Benzoic Acid
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:1.83 Å Release Date: 2014-06-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 32B |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: 32B
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Tmk In Complex With Compound 46, 2-(3-Chlorophenoxy)-3-Fluoro-4-{(1R)-3-Methyl-1-[(3S)-3-(5-Methyl-2,4-Dioxo-3,4-Dihydropyrimidin-1(2H)-Yl)Piperidin-1-Yl]Butyl}Benzoic Acid
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:1.62 Å Release Date: 2014-06-11 Classification: Transferase/transferase inhibitor Ligands: 32C |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: 32C
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S.Aureus Tmk In Complex With Potent Inhibitor Compound 47
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2014-06-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 32E |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2014-06-11
Ligands: 32E
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Thymidylate Kinase (Tmk) From S. Aureus In Complex With Tk-666
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-10-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 0YB |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2012-10-24
Ligands: 0YB
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Crystal Structure Of Thymidylate Kinase From Staphylococcus Aureus Bound To Inhibitor.
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2012-10-24 Classification: Transferase/Transferase inhibitor Ligands: 0Y5 |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2012-10-24
Ligands: 0Y5
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Discovery Of Selective And Potent Inhibitors Of Gram-Positive Bacterial Thymidylate Kinase (Tmk: Compound 41)
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2012-10-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 13Y |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2012-10-24
Ligands: 13Y
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Discovery Of Selective And Potent Inhibitors Of Gram-Positive Bacterial Thymidylate Kinase (Tmk): Compund 16
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-10-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: 14D |
Organism: Staphylococcus aureus subsp. aureus
Method: X-RAY DIFFRACTION
Release Date: 2012-10-24
Ligands: 14D
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E.Coli Glmu In Complex With An Antibacterial Inhibitor
Organism: Escherichia coli
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2012-08-15 Classification: TRANSFERASE Ligands: R82, SO4 |
Organism: Escherichia coli
Method: X-RAY DIFFRACTION
Release Date: 2012-08-15
Ligands: R82, SO4
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S.Pneumoniae Glmu In Complex With An Antibacterial Inhibitor
Organism: Streptococcus pneumoniae
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2012-02-15 Classification: TRANSFERASE Ligands: R84, SO4 |
Organism: Streptococcus pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2012-02-15
Ligands: R84, SO4
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S.Pneumoniae Glmu In Complex With An Antibacterial Inhibitor
Organism: Streptococcus pneumoniae
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2012-02-15 Classification: TRANSFERASE Ligands: R83, SO4 |
Organism: Streptococcus pneumoniae
Method: X-RAY DIFFRACTION
Release Date: 2012-02-15
Ligands: R83, SO4
