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9TDA image
Erap1 In Complex With 1-[2-(5-Bromo-7-Fluoro-2-Oxo-2,3-Dihydro-1,3-Benzothiazol-3-Yl)Acetamido]-4,4-Difluorocyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.55 Å Release Date: 2026-05-06
Classification: PEPTIDE BINDING PROTEIN
Ligands: ZN, SIN, PO4, EDO, A1JVE

9TD3 image
Erap1 In Complex With 1-[2-(6-Bromo-2,2-Difluoro-3-Oxo-3,4-Dihydro-2H-1,4-Benzoxazin-4-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.57 Å Release Date: 2026-04-22
Classification: PEPTIDE BINDING PROTEIN
Ligands: ZN, PO4, EDO, A1JVD

9TD4 image
Erap1 In Complex With 1-[2-(2-Oxo-5-Phenyl-2,3-Dihydro-1,3-Benzoxazol-3-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.73 Å Release Date: 2026-04-22
Classification: PEPTIDE BINDING PROTEIN
Ligands: ZN, MLT, EDO, A1JVG

9TD5 image
Erap1 In Complex With 1-[2-(5-Chloro-2-Oxo-2,3-Dihydro-1,3-Benzothiazol-3-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.45 Å Release Date: 2026-04-22
Classification: PEPTIDE BINDING PROTEIN
Ligands: ZN, PO4, EDO, A1JVH

9TD7 image
Erap1 In Complex With 1-[2-(3-Oxo-6-Phenyl-3,4-Dihydro-2H-1,4-Benzoxazin-4-Yl)Acetamido]Cyclohexane-1-Carboxylic Acid
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.37 Å Release Date: 2026-04-22
Classification: PEPTIDE BINDING PROTEIN
Ligands: ZN, PO4, EDO, A1JVF

9H2X image
Crystal Structure Of Stabilized A2A Adenosine Receptor A2Ar-Star2-Bril In Complex With Compound 7, A Novel Nanomolar A2A Receptor Antagonist From Modern Hit-Finding With Structure-Guided De Novo Design
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Resolution:1.75 Å Release Date: 2025-06-18
Classification: MEMBRANE PROTEIN

9H37 image
Crystal Structure Of Stabilized A2A Adenosine Receptor A2Ar-Star2-Bril In Complex With Compound 9, A Novel Nanomolar A2A Receptor Antagonist From Modern Hit-Finding With Structure-Guided De Novo Design
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Resolution:1.72 Å Release Date: 2025-06-18
Classification: MEMBRANE PROTEIN

8OL8 image
Solution Nmr Structure Of Lactamised Alpha-Synuclein 2-12 Peptide In 50% Tfe.
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2024-07-10
Classification: LIPID BINDING PROTEIN

8EWV image
Dna-Encoded Library (Del)-Enabled Discovery Of Proximity Inducing Small Molecules
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:3.40 Å Release Date: 2023-10-04
Classification: APOPTOSIS
Ligands: X5K

8OJR image
Solution Nmr Structure Of Alpha-Synuclein 1-25 Peptide In 50% Tfe.
Organism: Homo sapiens
Method: SOLUTION NMR
Release Date: 2023-08-09
Classification: LIPID BINDING PROTEIN

7P0F image
Crystal Structure Of A Cgrp Receptor Ectodomain Heterodimer Bound To Macrocyclic Inhibitor Htl0028125
Organism: Escherichia coli (strain k12), Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.85 Å Release Date: 2022-06-15
Classification: MEMBRANE PROTEIN
Ligands: 7IR, PG4

7P0I image
Crystal Structure Of A Cgrp Receptor Ectodomain Heterodimer Bound To Macrocyclic Inhibitor Compound 13
Organism: Escherichia coli (strain k12), Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.30 Å Release Date: 2022-06-15
Classification: MEMBRANE PROTEIN
Ligands: PG4, 7IU

7RQ8 image
Crystal Structure Of The Wild-Type Thermus Thermophilus 70S Ribosome In Complex With Iboxamycin, Mrna, Deacylated A- And E-Site Trnas, And Aminoacylated P-Site Trna At 2.50A Resolution

7RQ9 image
Crystal Structure Of The A2058-Dimethylated Thermus Thermophilus 70S Ribosome In Complex With Iboxamycin, Mrna, Deacylated A- And E-Site Trnas, And Aminoacylated P-Site Trna At 2.60A Resolution

6ZDR image
Crystal Structure Of Stabilized A2A Adenosine Receptor A2Ar-Star2-Bril In Complex With Chromone 4D
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Resolution:1.92 Å Release Date: 2020-09-16
Classification: PROTEIN BINDING
Ligands: QGE, NA, CLR, OLA, OLC

6ZDV image
Crystal Structure Of Stabilized A2A Adenosine Receptor A2Ar-Star2-Bril In Complex With Chromone 5D
Organism: Homo sapiens, Escherichia coli
Method: X-RAY DIFFRACTION
Resolution:2.13 Å Release Date: 2020-09-16
Classification: PROTEIN BINDING
Ligands: QGW, NA, CLR, OLB, OLA, OLC

6ZHO image
Crystal Structure Of A Cgrp Receptor Ectodomain Heterodimer With Bound High Affinity Inhibitor
Organism: Escherichia coli (strain k12), Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.60 Å Release Date: 2020-07-15
Classification: MEMBRANE PROTEIN
Ligands: QLQ, PG4

6ZIS image
Crystal Structure Of A Cgrp Receptor Ectodomain Heterodimer With Bound High Affinity Inhibitor
Organism: Escherichia coli (strain k12), Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:1.73 Å Release Date: 2020-07-15
Classification: MEMBRANE PROTEIN
Ligands: PG4, 3N6

6ODA image
Crystal Structure Of Hdac8 In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.88 Å Release Date: 2020-04-01
Classification: HYDROLASE
Ligands: C7, ZN, K

6ODB image
Crystal Structure Of Hdac8 In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Resolution:2.70 Å Release Date: 2020-04-01
Classification: HYDROLASE
Ligands: M8G, ZN, K, GOL
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