Search Count: 26
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Structure Of Human Vaccinia-Related Kinase 1 (Vrk1) Bound To Ach000400
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2024-09-04 Classification: TRANSFERASE Ligands: PEG, YD9, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2024-09-04
Ligands: PEG, YD9, SO4
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Structure Of Maternal Embryonic Leucine Zipper Kinase Bound To Ldsm276
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2020-07-29 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: F7D, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-07-29
Ligands: F7D, EDO
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Structure Of Human Vaccinia-Related Kinase 1 (Vrk1) Bound To Ldsm311
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2020-03-11 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, RYA, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-03-11
Ligands: SO4, RYA, EDO
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Human Prpf4B Bound To Benzothiophene Inhibitor 224
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-08-28 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: OCJ, EDO, PO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: OCJ, EDO, PO4
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Human Prpf4B Bound To Benzothiophene Inhibitor 329
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2019-08-28 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: SO4, OND |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: SO4, OND
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Human Pim1 Bound To Benzothiophene Inhibitor 213
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-07-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: O97, GOL |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2019-07-24
Ligands: O97, GOL
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Human Pim1 Bound To Benzothiophene Inhibitor 224
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-07-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: OCJ, GOL, EDO |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2019-07-24
Ligands: OCJ, GOL, EDO
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Human Pim1 Bound To Benzothiophene Inhibitor 292
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-07-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: OD4, GOL |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2019-07-24
Ligands: OD4, GOL
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Human Pim1 Bound To Benzothiophene Inhibitor 354
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2019-07-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: OD1 |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2019-07-24
Ligands: OD1
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Human Pim1 Bound To Benzothiophene Inhibitor 379
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-07-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: SO4, OBY |
Organism: Homo sapiens, Synthetic construct
Method: X-RAY DIFFRACTION
Release Date: 2019-07-24
Ligands: SO4, OBY
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A N,N-Dipropynyl-Dihydropteridine-3-Hydroxyindazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2019-02-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: KWJ, SO4, EDO, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-02-20
Ligands: KWJ, SO4, EDO, PEG
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Crystal Structure Of Human Vaccinia-Related Kinase 2 (Vrk-2) Bound To Pyridin-Benzenesulfonamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2019-01-16 Classification: TRANSFERASE Ligands: KJD, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-16
Ligands: KJD, SO4
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A N,N-Dipropyl-Dihydropteridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-05-23 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CL, ACT, G6J, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-05-23
Ligands: CL, ACT, G6J, SO4, GOL
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Crystal Structure Of The Human Vaccinia-Related Kinase 1 (Vrk1) Bound To An N-Propynyl-N-Isopentyl-Dihydropteridin Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2018-04-04 Classification: Transferase/Transferase Inhibitor Ligands: F87, SO4, ACT, GOL, FCS |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
Ligands: F87, SO4, ACT, GOL, FCS
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A N-Methyl-N-Propyl-Dihydropteridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2018-04-04 Classification: Transferase/Transferase Inhibitor Ligands: SO4, ACT, PG4, FBY, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-04-04
Ligands: SO4, ACT, PG4, FBY, GOL, CL
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A N-Propynyl-N-Ethyl-Dihydropteridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2018-03-28 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: F8Y, SO4, ACT, GOL, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-28
Ligands: F8Y, SO4, ACT, GOL, CL
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A N,N-Dipropynyl-Dihydropteridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-03-21 Classification: Transferase/Transferase Inhibitor Ligands: ACT, F7D, SO4, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-21
Ligands: ACT, F7D, SO4, PEG
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A Propynyl-Pteridinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.45 Å Release Date: 2018-03-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CL, EA7, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-03-07
Ligands: CL, EA7, GOL
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A Phenyl-Pteridinone Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-12-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: CL, E8D, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: CL, E8D, SO4, GOL
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Crystal Structure Of The Human Vaccinia-Related Kinase Bound To A Bis-Difluorophenol-Aminopyridine Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2017-12-20 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: E8V, GOL, CL, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-12-20
Ligands: E8V, GOL, CL, SO4
