Search Count: 79
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Tgfb1 In Complex With Nis793 Fab
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.75 Å Release Date: 2026-06-17 Classification: CYTOKINE Ligands: SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-06-17
Ligands: SO4
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Crystal Structure Of Htead2 Bound To A Methoxypyridine Lipid Pocket Binder
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2023-08-16 Classification: TRANSCRIPTION/INHIBITOR Ligands: TRS, Y2S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2023-08-16
Ligands: TRS, Y2S
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Crystal Structure Of Braf In Complex With Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.49 Å Release Date: 2021-05-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: V5J, IOD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-26
Ligands: V5J, IOD
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Crystal Structure Of Braf In Complex With Inhibitor Gne-0749
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.93 Å Release Date: 2021-05-26 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: VQP, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-05-26
Ligands: VQP, CL
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Crystal Structure Of Braf Kinase Domain Bound To Belvarafenib
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2021-03-10 Classification: SIGNALING PROTEIN Ligands: V1Y, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-10
Ligands: V1Y, CL
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Apo Braf Dimer Bound To 14-3-3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.30 Å Release Date: 2020-10-07 Classification: SIGNALING PROTEIN/Transferase Ligands: EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-07
Ligands: EDO
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Braf-Mek Complex With Amp-Pcp Bound To Braf
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.89 Å Release Date: 2019-08-28 Classification: TRANSFERASE Ligands: ACP, MG, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: ACP, MG, SO4
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Braf Dimer Bound To 14-3-3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2019-08-28 Classification: SIGNALING PROTEIN/Transferase Ligands: 29L |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-08-28
Ligands: 29L
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Lactate Dehydrogenase In Complex With Inhibitor 6-(3-Aminophenyl)-3-((2-Chlorophenyl)Thio)-4-Hydroxy-6-(Thiophen-3-Yl)-5,6-Dihydro-2H-Pyran-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE/Inhibitor Ligands: NAD, EPE, SO4, D4S |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: NAD, EPE, SO4, D4S
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Lactate Dehydrogenase In Complex With Inhibitor (S)-5-((2-Chlorophenyl)Thio)-6'-((4-Fluorophenyl)Amino)-4-Hydroxy-2-(Thiophen-3-Yl)-2,3-Dihydro-[2,2'-Bipyridin]-6(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE/Inhibitor Ligands: EPE, NAD, LAC, SO4, D47 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: EPE, NAD, LAC, SO4, D47
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Lactate Dehydrogenase In Complex With Inhibitor (R)-3-((2-Chlorophenyl)Thio)-6-(3-((4-Fluorophenyl)Amino)Phenyl)-4-Hydroxy-6-(Thiophen-3-Yl)-5,6-Dihydro-2H-Pyran-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE Ligands: NAD, EPE, SO4, D3S, LAC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: NAD, EPE, SO4, D3S, LAC
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Lactate Dehydrogenase In Complex With Inhibitor (R)-5-((2-Chlorophenyl)Thio)-6'-(4-Fluorophenoxy)-4-Hydroxy-2-(Thiophen-3-Yl)-2,3-Dihydro-[2,2'-Bipyridin]-6(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE/Inhibitor Ligands: NAD, SO4, D3J, LAC |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: NAD, SO4, D3J, LAC
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Lactate Dehydrogenase In Complex With Inhibitor (S)-5-((2-Chlorophenyl)Thio)-6'-(4-Fluorophenoxy)-4-Hydroxy-2-(Thiophen-3-Yl)-2,3-Dihydro-[2,2'-Bipyridin]-6(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.47 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE/Inhibitor Ligands: NAD, SO4, LAC, D4J |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: NAD, SO4, LAC, D4J
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Lactate Dehydrogenase In Complex With Inhibitor 3-((2-Chlorophenyl)Thio)-6-(6-((4-Fluorophenyl)Amino)Pyridin-2-Yl)-4-Hydroxy-6-(Thiophen-3-Yl)-5,6-Dihydro-2H-Pyran-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2018-10-24 Classification: OXIDOREDUCTASE/Inhibitor Ligands: NAD, SO4, D4A |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-24
Ligands: NAD, SO4, D4A
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Lactate Dehydrogenase In Complex With Inhibitor (R)-3-((2-Chlorophenyl)Thio)-6-(3-((4-Fluorophenyl)Amino)Phenyl)-4-Hydroxy-6-(Thiophen-3-Yl)-5,6-Dihydro-2H-Pyran-2-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2018-10-17 Classification: OXIDOREDUCTASE/Inhibitor Ligands: NAD, EPE, SO4, D0Y |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: NAD, EPE, SO4, D0Y
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Lactate Dehydrogenase In Complex With Inhibitor (R)-5-((2-Chlorophenyl)Thio)-6'-((4-Fluorophenyl)Amino)-4-Hydroxy-2-(Thiophen-3-Yl)-2,3-Dihydro-[2,2'-Bipyridin]-6(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2018-10-17 Classification: OXIDOREDUCTASE/Inhibitor Ligands: EPE, NAD, SO4, D0V |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2018-10-17
Ligands: EPE, NAD, SO4, D0V
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Lactate Dehydrogenase In Complex With Hydroxylactam Inhibitor Compound 9: (6R)-3-[(2-Chlorophenyl)Sulfanyl]-4-Hydroxy-6-(3-Hydroxyphenyl)-6-(Thiophen-3-Yl)-5,6-Dihydropyridin-2(1H)-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2016-09-14 Classification: OXIREDUCTASE/OXIREDUCTASE INHIBITOR Ligands: EPE, TXD, 6EY, SO4, NAI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-14
Ligands: EPE, TXD, 6EY, SO4, NAI
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Lactate Dehydrogenase In Complex With Hydroxylactam Inhibitor Compound 31: (2~{S})-5-(2-Chlorophenyl)Sulfanyl-2-(4-Morpholin-4-Ylphenyl)-4-Oxidanyl-2-Thiophen-3-Yl-1,3-Dihydropyridin-6-One
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.00 Å Release Date: 2016-09-14 Classification: OXIREDUCTASE/OXIREDUCTASE INHIBITOR Ligands: NAD, SO4, GN2 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-14
Ligands: NAD, SO4, GN2
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Egfr Kinase Domain Mutant "Tmlr" With Azabenzimidazole Compound 7
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60B |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60B
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Egfr Kinase Domain Mutant "Tmlr" With 3-Carboxamide Azaindole Compound 13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.46 Å Release Date: 2016-09-07 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SO4, 60D |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-09-07
Ligands: SO4, 60D
