Search Count: 19
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Human Parp14 (Artd8), Catalytic Fragment In Complex With Rbn012042
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.25 Å Release Date: 2021-04-21 Classification: TRANSFERASE/Inhibitor Ligands: XRM, CL, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: XRM, CL, EDO
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Human Parp14 (Artd8), Catalytic Fragment In Complex With Rbn011980
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.57 Å Release Date: 2021-04-21 Classification: TRANSFERASE/Inhibitor Ligands: YFG, CL, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-04-21
Ligands: YFG, CL, GOL
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Human Parp14 (Artd8), Catalytic Fragment In Complex With Rbn012759
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.66 Å Release Date: 2021-03-24 Classification: TRANSFERASE/Inhibitor Ligands: XBA, EDO |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: XBA, EDO
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Human Parp14 (Artd8), Catalytic Fragment In Complex With Compound 3
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.95 Å Release Date: 2021-03-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: TZ7, EDO, PEG, GOL, SO4, PGE |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: TZ7, EDO, PEG, GOL, SO4, PGE
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Human Parp14 (Artd8), Catalytic Fragment In Complex With Compound 2
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2021-03-24 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: FDR, EDO, TYG, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-03-24
Ligands: FDR, EDO, TYG, GOL
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Human Poly(Adp-Ribose) Polymerase 12, Catalytic Fragment With Four Point Mutations In Complex With Rbn-2397
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.04 Å Release Date: 2020-12-16 Classification: TRANSFERASE Ligands: QO4, CL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-12-16
Ligands: QO4, CL
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Human Parp16 In Complex With Rbn010860
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.13 Å Release Date: 2020-10-07 Classification: TRANSFERASE Ligands: T9D, CIT, GOL, EDO, PEG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2020-10-07
Ligands: T9D, CIT, GOL, EDO, PEG
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Crystal Structure Of Prmt5:Mep50 With Compound 8 And Sinefungin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.27 Å Release Date: 2016-02-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SFG, 5QJ, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: SFG, 5QJ, GOL
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Crystal Structure Of Prmt5:Mep50 With Compound 9 And Sinefungin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.52 Å Release Date: 2016-02-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SFG, 5QH, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: SFG, 5QH, GOL
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Crystal Structure Of Prmt5:Mep50 With Compound 10 And Sam
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.39 Å Release Date: 2016-02-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAM, 5QK, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: SAM, 5QK, GOL
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Crystal Structure Of Prmt5:Mep50 With Compound 15 And Sinefungin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.37 Å Release Date: 2016-02-24 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SFG, 5QL, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-02-24
Ligands: SFG, 5QL, GOL
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Crystal Structure Of Prmt5:Mep50 With Epz015666 And Sinefungin
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.35 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SFG, 3XV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SFG, 3XV, GOL
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Crystal Structure Of Prmt5:Mep50 With Epz015666 And Sam
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAM, 3XV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SAM, 3XV, GOL
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Crystal Structure Of Prmt5:Mep50 With Epz015666 And Sah
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:3.05 Å Release Date: 2015-04-22 Classification: TRANSFERASE/TRANSFERASE INHIBITOR Ligands: SAH, 3XV |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-04-22
Ligands: SAH, 3XV
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Crystal Structure Of Dot1L In Complex With Epz000004
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2012-10-17 Classification: transferase/transferase inhibitor Ligands: EP4, SO4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-17
Ligands: EP4, SO4, GOL
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Crystal Structure Of Dot1L In Complex With Epz003696
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.80 Å Release Date: 2012-10-17 Classification: transferase/transferase inhibitor Ligands: 0QJ |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-17
Ligands: 0QJ
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Crystal Structure Of Dot1L In Complex With Epz004777
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.85 Å Release Date: 2012-10-17 Classification: transferase/transferase inhibitor Ligands: 0QK, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-17
Ligands: 0QK, SO4
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Dot1L Structure In Complex With Sam
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2011-05-25 Classification: TRANSFERASE Ligands: SAM, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: SAM, SO4
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Dot1L Structure In Complex With Sah
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2011-05-25 Classification: TRANSFERASE Ligands: SAH, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2011-05-25
Ligands: SAH, SO4
