Search Count: 88
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Human Tlr8 Bound To The Potent Agonist, Gs-9688 (Selgantolimod)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2021-02-03 Classification: IMMUNE SYSTEM Ligands: MAN, NAG, U57 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-03
Ligands: MAN, NAG, U57
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Discovery Of A Potent Cyclophilin Inhibitor (Compound 3) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 7HG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 7HG
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Discovery Of A Potent Cyclophilin Inhibitor (Compound 5) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 78E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 78E
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Discovery Of A Potent Cyclophilin Inhibitor (Compound 6) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 78R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 78R
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Discovery Of A Potent Cyclophilin Inhibitor (Compound 7) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 78X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 78X
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Discovery Of A Potent Cyclophilin Inhibitor (Compound 8) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 838, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 838, SO4
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Hiv-1 Reverse Transcriptase In Complex With Dna
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2010-03-23 Classification: TRANSFERASE/DNA Ligands: SO4, MG |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2010-03-23
Ligands: SO4, MG
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Hiv-1 Reverse Transcriptase-Dna Complex With Nuceotide Inhibitor Gs-9148-Diphosphate Bound In Nucleotide Site
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2010-03-23 Classification: TRANSFERASE/DNA Ligands: SO4, MG, 914 |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2010-03-23
Ligands: SO4, MG, 914
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Hiv-1 Reverse Transcriptase-Dna Complex With Datp Bound In The Nucleotide Binding Site
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2010-03-23 Classification: TRANSFERASE/DNA Ligands: SO4, MG, DTP |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2010-03-23
Ligands: SO4, MG, DTP
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Hiv-1 Reverse Transcriptase-Dna Complex With Gs-9148 Terminated Primer
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2010-03-23 Classification: TRANSFERASE/DNA Ligands: MG, SO4 |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2010-03-23
Ligands: MG, SO4
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Dissecting And Designing Inhibitor Selectivity Determinants At The S1 Site Using An Artificial Ala190 Protease (Ala190 Upa)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2004-09-21 Classification: BLOOD CLOTTING, hydrolase Ligands: 696, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-09-21
Ligands: 696, CIT
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Dissecting And Designing Inhibitor Selectivity Determinants At The S1 Site Using An Artificial Ala190 Protease (Ala190 Upa)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2004-09-21 Classification: BLOOD CLOTTING, hydrolase Ligands: ESI, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-09-21
Ligands: ESI, CIT
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Dissecting And Designing Inhibitor Selectivity Determinants At The S1 Site Using An Artificial Ala190 Protease (Ala190 Upa)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2004-09-21 Classification: BLOOD CLOTTING, hydrolase Ligands: CR9, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-09-21
Ligands: CR9, CIT
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Dissecting And Designing Inhibitor Selectivity Determinants At The S1 Site Using An Artificial Ala190 Protease (Ala190 Upa)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2004-09-21 Classification: BLOOD CLOTTING, hydrolase Ligands: CR9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-09-21
Ligands: CR9
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Dissecting And Designing Inhibitor Selectivity Determinants At The S1 Site Using An Artificial Ala190 Protease (Ala190 Upa)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2004-09-21 Classification: serine protease, hydrolase Ligands: 132 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-09-21
Ligands: 132
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Dissecting And Designing Inhibitor Selectivity Determinants At The S1 Site Using An Artificial Ala190 Protease (Ala190 Upa)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2004-09-21 Classification: serine protease, hydrolase Ligands: CR9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-09-21
Ligands: CR9
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Dissecting And Designing Inhibitor Selectivity Determinants At The S1 Site Using An Artificial Ala190 Protease (Ala190 Upa)
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2004-09-21 Classification: BLOOD CLOTTING,HYDROLASE/INHIBITOR |
Organism: Hirudo medicinalis, Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-09-21
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Elaborate Manifold Of Short Hydrogen Bond Arrays Mediating Binding Of Active Site-Directed Serine Protease Inhibitors
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2003-09-02 Classification: HYDROLASE Ligands: CA, SO4, 991 |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2003-09-02
Ligands: CA, SO4, 991
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Elaborate Manifold Of Short Hydrogen Bond Arrays Mediating Binding Of Active Site-Directed Serine Protease Inhibitors
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.45 Å Release Date: 2003-09-02 Classification: HYDROLASE Ligands: CA, CL, SO4, CR9 |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2003-09-02
Ligands: CA, CL, SO4, CR9
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Elaborate Manifold Of Short Hydrogen Bond Arrays Mediating Binding Of Active Site-Directed Serine Protease Inhibitors
Organism: Bos taurus
Method: X-RAY DIFFRACTION Resolution:1.65 Å Release Date: 2003-09-02 Classification: HYDROLASE Ligands: CA, CL, CR4 |
Organism: Bos taurus
Method: X-RAY DIFFRACTION
Release Date: 2003-09-02
Ligands: CA, CL, CR4