Search Count: 107
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Human Tlr8 Bound To The Potent Agonist, Gs-9688 (Selgantolimod)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2021-02-03 Classification: IMMUNE SYSTEM Ligands: MAN, NAG, U57 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2021-02-03
Ligands: MAN, NAG, U57
 |
N-Terminal Bromodomain Of Human Brd2 With N-((4-(3-(N-Cyclopentylsulfamoyl)-4-Methylphenyl)-3-Methylisoxazol-5-Yl)Methyl)Acetamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2019-01-23 Classification: transcription/transcription inhibitor Ligands: JWA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-23
Ligands: JWA
 |
N-Terminal Bromodomain Of Human Brd2 In Complex With 4,4'-(Quinoline-5,7-Diyl)Bis(3,5-Dimethylisoxazole) Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-01-23 Classification: transcription/transcription inhibitor Ligands: JWD, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-23
Ligands: JWD, SO4
 |
N-Terminal Bromodomain Of Human Brd2 In Complex With N-Cyclopentyl-7-(3,5-Dimethylisoxazol-4-Yl)Quinoline-5-Sulfonamide Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-01-23 Classification: transcription/transcription inhibitor Ligands: JVY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-23
Ligands: JVY
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C-Terminal Bromodomain Of Human Brd2 In Complex With 4-(2-Cyclopropyl-7-(6-Methylquinolin-5-Yl)-1H-Benzo[D]Imidazol-5-Yl)-3,5-Dimethylisoxazole Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.27 Å Release Date: 2019-01-23 Classification: transcription/transcription inhibitor Ligands: JW4, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-23
Ligands: JW4, GOL
 |
Discovery Of A Potent Cyclophilin Inhibitor (Compound 3) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.30 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 7HG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 7HG
 |
Discovery Of A Potent Cyclophilin Inhibitor (Compound 5) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 78E |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 78E
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Discovery Of A Potent Cyclophilin Inhibitor (Compound 6) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.40 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 78R |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 78R
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Discovery Of A Potent Cyclophilin Inhibitor (Compound 7) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.48 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 78X |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 78X
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Discovery Of A Potent Cyclophilin Inhibitor (Compound 8) Based On Structural Simplification Of Sanglifehrin A
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.50 Å Release Date: 2017-01-25 Classification: isomerase/isomerase inhibitor Ligands: 838, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-25
Ligands: 838, SO4
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Hiv-1 Reverse Transcriptase In Complex With Dna
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:3.10 Å Release Date: 2010-03-23 Classification: TRANSFERASE/DNA Ligands: SO4, MG |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2010-03-23
Ligands: SO4, MG
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Hiv-1 Reverse Transcriptase-Dna Complex With Nuceotide Inhibitor Gs-9148-Diphosphate Bound In Nucleotide Site
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2010-03-23 Classification: TRANSFERASE/DNA Ligands: SO4, MG, 914 |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2010-03-23
Ligands: SO4, MG, 914
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Hiv-1 Reverse Transcriptase-Dna Complex With Datp Bound In The Nucleotide Binding Site
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2010-03-23 Classification: TRANSFERASE/DNA Ligands: SO4, MG, DTP |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2010-03-23
Ligands: SO4, MG, DTP
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Hiv-1 Reverse Transcriptase-Dna Complex With Gs-9148 Terminated Primer
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2010-03-23 Classification: TRANSFERASE/DNA Ligands: MG, SO4 |
Organism: Human immunodeficiency virus type 1
Method: X-RAY DIFFRACTION
Release Date: 2010-03-23
Ligands: MG, SO4
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Dissecting And Designing Inhibitor Selectivity Determinants At The S1 Site Using An Artificial Ala190 Protease (Ala190 Upa)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.68 Å Release Date: 2004-09-21 Classification: BLOOD CLOTTING, hydrolase Ligands: 696, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-09-21
Ligands: 696, CIT
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Dissecting And Designing Inhibitor Selectivity Determinants At The S1 Site Using An Artificial Ala190 Protease (Ala190 Upa)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2004-09-21 Classification: BLOOD CLOTTING, hydrolase Ligands: ESI, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-09-21
Ligands: ESI, CIT
 |
Dissecting And Designing Inhibitor Selectivity Determinants At The S1 Site Using An Artificial Ala190 Protease (Ala190 Upa)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.63 Å Release Date: 2004-09-21 Classification: BLOOD CLOTTING, hydrolase Ligands: CR9, CIT |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-09-21
Ligands: CR9, CIT
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Dissecting And Designing Inhibitor Selectivity Determinants At The S1 Site Using An Artificial Ala190 Protease (Ala190 Upa)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.05 Å Release Date: 2004-09-21 Classification: BLOOD CLOTTING, hydrolase Ligands: CR9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-09-21
Ligands: CR9
 |
Dissecting And Designing Inhibitor Selectivity Determinants At The S1 Site Using An Artificial Ala190 Protease (Ala190 Upa)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.75 Å Release Date: 2004-09-21 Classification: serine protease, hydrolase Ligands: 132 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-09-21
Ligands: 132
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Dissecting And Designing Inhibitor Selectivity Determinants At The S1 Site Using An Artificial Ala190 Protease (Ala190 Upa)
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.78 Å Release Date: 2004-09-21 Classification: serine protease, hydrolase Ligands: CR9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2004-09-21
Ligands: CR9