Search Count: 32
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Cryo-Em Structure Of Vvd-908 Nlrp3 Complex
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY Resolution:3.03 Å Release Date: 2026-08-19 Classification: IMMUNE SYSTEM Ligands: ADP, A1CZP, MG |
Organism: Homo sapiens
Method: ELECTRON MICROSCOPY
Release Date: 2026-08-19
Ligands: ADP, A1CZP, MG
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Crystal Structure Of E.Coli Phosphopantetheine Adenylyltransferase (Ppat/Coad) In Complex With (R)-3-(3-Chlorophenyl)-3-((5-Methyl-7-Oxo-4,7-Dihydro-[1,2,4]Triazolo[1,5-A]Pyrimidin-2-Yl)Amino)Propanenitrile
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:1.61 Å Release Date: 2018-03-14 Classification: TRANSFERASE/antibiotic Ligands: EXJ, ATP, MG, SO4 |
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: EXJ, ATP, MG, SO4
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Crystal Structure Of E.Coli Phosphopantetheine Adenylyltransferase (Ppat/Coad) In Complex With 1-Benzyl-1H-Imidazo[4,5-B]Pyridine
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:1.77 Å Release Date: 2018-03-14 Classification: TRANSFERASE/antibiotic Ligands: EXG, SO4, DMS |
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: EXG, SO4, DMS
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Crystal Structure Of E.Coli Phosphopantetheine Adenylyltransferase (Ppat/Coad) In Complex With 2-((3-Bromobenzyl)Amino)-5-Methyl-[1,2,4]Triazolo[1,5-A]Pyrimidin-7(4H)-One
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:1.79 Å Release Date: 2018-03-14 Classification: TRANSFERASE/antibiotic Ligands: EXP, SO4 |
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: EXP, SO4
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Crystal Structure Of E.Coli Phosphopantetheine Adenylyltransferase (Ppat/Coad) In Complex With (R)-2,4-Dihydroxy-N-(2-(4-Hydroxy-1H-Benzo[D]Imidazol-2-Yl)Ethyl)-3,3-Dimethylbutanamide
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:1.87 Å Release Date: 2018-03-14 Classification: TRANSFERASE/antibiotic Ligands: EXS, SO4 |
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: EXS, SO4
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Crystal Structure Of E.Coli Phosphopantetheine Adenylyltransferase (Ppat/Coad) In Complex With 3-((1S,2S)-2-(4-Hydroxy-1H-Benzo[D]Imidazol-2-Yl)Cyclopentyl)Benzoic Acid
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:1.82 Å Release Date: 2018-03-14 Classification: TRANSFERASE/antibiotic Ligands: EXV, SO4 |
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: EXV, SO4
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Crystal Structure Of E.Coli Phosphopantetheine Adenylyltransferase (Ppat/Coad) In Complex With 2-(3-Chlorophenethyl)-1H-Benzo[D]Imidazol-4-Ol
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:1.92 Å Release Date: 2018-03-14 Classification: TRANSFERASE/antibiotic Ligands: EX7, SO4 |
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: EX7, SO4
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Crystal Structure Of E.Coli Phosphopantetheine Adenylyltransferase (Ppat/Coad) In Complex With 2-(Trifluoromethyl)-1H-Benzo[D]Imidazol-4-Ol
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION Resolution:2.06 Å Release Date: 2018-03-14 Classification: TRANSFERASE/antibiotic Ligands: EXD, SO4 |
Organism: Escherichia coli (strain k12)
Method: X-RAY DIFFRACTION
Release Date: 2018-03-14
Ligands: EXD, SO4
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Crystal Structure Of Eed In Complex With 6-(2-Fluoro-5-Methoxybenzyl)-1-Isopropyl-5,6,7,8-Tetrahydroimidazo[1,5-A]Pyridin-3-Amine 6-(2-Fluoro-5-Methoxybenzyl)-1-Isopropyl-5,6,7,8-Tetrahydroimidazo[1,5-A]Pyridin-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2017-01-11 Classification: TRANSCRIPTION Ligands: 7VV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: 7VV, GOL
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Crystal Structure Of Eed In Complex With 3-(3-Methoxybenzyl)Piperidine Hydrochloride
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.33 Å Release Date: 2017-01-11 Classification: TRANSCRIPTION Ligands: FMT, 7VY |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: FMT, 7VY
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Crystal Structure Of Eed In Complex With H3K27Me3 Peptide And 3-(Benzo[D][1,3]Dioxol-4-Ylmethyl)Piperidine-1-Carboximidamide
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.60 Å Release Date: 2017-01-11 Classification: Transcription/Transferase Ligands: 7W7, YT3 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: 7W7, YT3
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Crystal Structure Of Eed In Complex With H3K27Me3 Peptide And 6-(Benzo[D][1,3]Dioxol-4-Ylmethyl)-5,6,7,8-Tetrahydroimidazo[1,5-A]Pyridin-3-Amine
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2017-01-11 Classification: Transcription/Transferase Ligands: GOL, YT3, 7WD |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2017-01-11
Ligands: GOL, YT3, 7WD
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Design, Synthesis And Structure Activity Relationship Of Potent Pan-Pim Kinase Inhibitors Derived From The Pyridyl-Amide Scaffold
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2016-04-06 Classification: Transferase/Transferase Inhibitor Ligands: PEG, 6CB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2016-04-06
Ligands: PEG, 6CB
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Identification Of N-(4-((1R,3S,5S)-3-Amino-5-Methylcyclohexyl)Pyridin-3-Yl)-6-(2,6-Difluorophenyl)-5-Fluoropicolinamide (Pim447), A Potent And Selective Proviral Insertion Site Of Moloney Murine Leukemia (Pim) 1,2 And 3 Kinase Inhibitor In Clinical Trials For Hematological Malignancies
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2015-11-11 Classification: Transferase/Transferase Inhibitor Ligands: 5H7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-11-11
Ligands: 5H7
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Rsk2 N-Terminal Kinase In Complex With Bi-D1870
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.55 Å Release Date: 2015-09-02 Classification: TRANSFERASE/TRANSFERASE Inhibitor Ligands: 584, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-02
Ligands: 584, GOL
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Rsk2 N-Terminal Kinase In Complex With Bis-Phenol Pyrazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.15 Å Release Date: 2015-09-02 Classification: TRANSFERASE/TRANSFERASE inhibitor Ligands: 583, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-09-02
Ligands: 583, GOL
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Serine/Threonine-Protein Kinase Pak1 Complexed With A Dibenzodiazepine: Identification Of An Allosteric Site On Pak1
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2015-08-05 Classification: Transferase/transferase inhibitor Ligands: 4PV, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-08-05
Ligands: 4PV, GOL
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Erk2 Complexed With N-Benzylpyridone Tetrahydroazaindazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2015-07-15 Classification: Transferase/Transferase inhibitor Ligands: 4V8, NI |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-15
Ligands: 4V8, NI
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Erk2 Complexed With 2-Pyridiyl Tetrahydroazaindazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.12 Å Release Date: 2015-07-15 Classification: Transferase/Transferase inhibitor Ligands: NI, 4V9 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-15
Ligands: NI, 4V9
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Erk2 Complexed With A N-H Tetrahydroazaindazole
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.85 Å Release Date: 2015-07-15 Classification: Transferase/Transferase inhibitor Ligands: 4VB |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2015-07-15
Ligands: 4VB
