Search Count: 34
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Mineralocorticoid Receptor In Complex With Acylurea Antagonists.
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.46 Å Release Date: 2026-02-18 Classification: TRANSCRIPTION Ligands: MPD, NHE, A1IJ6 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2026-02-18
Ligands: MPD, NHE, A1IJ6
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Mineralocorticoid Receptor In Complex With (S)-13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.54 Å Release Date: 2019-01-09 Classification: TRANSCRIPTION Ligands: GOL, EWN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-09
Ligands: GOL, EWN
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Mineralocorticoid Receptor In Complex With (S)-13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2019-01-09 Classification: TRANSCRIPTION Ligands: MPD, EY8 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-09
Ligands: MPD, EY8
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Mineralocorticoid Receptor In Complex With (S)-13
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.71 Å Release Date: 2019-01-09 Classification: TRANSCRIPTION Ligands: CL, EYN |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2019-01-09
Ligands: CL, EYN
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Pi3Kg In Complex With Azd6482
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.90 Å Release Date: 2014-10-22 Classification: TRANSFERASE Ligands: A82 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2014-10-22
Ligands: A82
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Bace-1 In Complex With Hea-Type Macrocyclic Inhibitor, Mv078571
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2013-09-04 Classification: Hydrolase/Hydrolase inhibitor Ligands: 0XA, ACT, GOL |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2013-09-04
Ligands: 0XA, ACT, GOL
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Design And Synthesis Of Potent Hydroxyethylamine (Hea) Bace-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-10-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 996 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-31
Ligands: 996
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Design And Synthesis Of Potent Hydroxyethylamine (Hea) Bace-1 Inhibitors
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-10-31 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 916 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-10-31
Ligands: 916
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Bace-1 In Complex With A Hea-Macrocyclic Type Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.80 Å Release Date: 2012-07-11 Classification: Hydrolase/Hydrolase inhibitor Ligands: 0LG |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-11
Ligands: 0LG
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Bace-1 In Complex With Hea-Macrocyclic Inhibitor, Mv078512
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:1.90 Å Release Date: 2012-07-11 Classification: Hydrolase/Hydrolase inhibitor Ligands: 0N1 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2012-07-11
Ligands: 0N1
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Bace-1 In Complex With A Norstatine Type Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2010-12-29 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 038 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-12-29
Ligands: 038
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Potent Beta-Secretase 1 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-09-08 Classification: HYDROLASE Ligands: 929 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-09-08
Ligands: 929
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Potent Beta-Secretase 1 Hydroxyethylene Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.10 Å Release Date: 2010-06-02 Classification: HYDROLASE Ligands: MV7 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-06-02
Ligands: MV7
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Hcv Ns3/Ns4A Complexed With Non-Covalent Macrocyclic Compound Tmc435
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.40 Å Release Date: 2010-03-09 Classification: HYDROLASE Ligands: 30B, ZN, GOL |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2010-03-09
Ligands: 30B, ZN, GOL
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The Hcv Ns3/Ns4A Protease Apo Structure
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION Resolution:2.50 Å Release Date: 2010-03-09 Classification: HYDROLASE Ligands: ZN |
Organism: Hepatitis c virus
Method: X-RAY DIFFRACTION
Release Date: 2010-03-09
Ligands: ZN
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Crystal Structure Of Beta-Secretase 1 In Complex With Selective Beta-Secretase 1 Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.20 Å Release Date: 2010-03-02 Classification: HYDROLASE/HYDROLASE INHIBITOR Ligands: 586, SO4 |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2010-03-02
Ligands: 586, SO4
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Beta-Secretase 1 Complexed With Statine-Based Inhibitor
Organism: Homo sapiens
Method: X-RAY DIFFRACTION Resolution:2.60 Å Release Date: 2008-12-16 Classification: HYDROLASE Ligands: 757, IPA |
Organism: Homo sapiens
Method: X-RAY DIFFRACTION
Release Date: 2008-12-16
Ligands: 757, IPA
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Novel Plasmepsin Ii-Inhibitor Complex
Organism: Plasmodium falciparum
Method: X-RAY DIFFRACTION Resolution:2.24 Å Release Date: 2006-07-05 Classification: HYDROLASE Ligands: TIT |
Organism: Plasmodium falciparum
Method: X-RAY DIFFRACTION
Release Date: 2006-07-05
Ligands: TIT
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Plasmepsin Ii-Pepstatin A Complex
Organism: Plasmodium falciparum, Streptomyces argenteolus subsp. toyonakensis
Method: X-RAY DIFFRACTION Resolution:2.70 Å Release Date: 2006-07-05 Classification: HYDROLASE/HYDROLASE INHIBITOR |
Organism: Plasmodium falciparum, Streptomyces argenteolus subsp. toyonakensis
Method: X-RAY DIFFRACTION
Release Date: 2006-07-05
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Crystal Structure Of Rv1284 From Mycobacterium Tuberculosis In Complex With Thiocyanate
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION Resolution:2.00 Å Release Date: 2005-03-08 Classification: UNKNOWN FUNCTION Ligands: ZN, SCN |
Organism: Mycobacterium tuberculosis
Method: X-RAY DIFFRACTION
Release Date: 2005-03-08
Ligands: ZN, SCN
